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Patent Evaluation

Fused thiazole derivatives having affinity for the histamine H3 receptor

Glaxo Group Limited: WO2006097691

Pages 129-131 | Published online: 03 Jan 2007

Bibliography

  • ARRANG JM, GARBURG M, SCHWARTZ JC: Autoinhibition of brain histamine release mediated by a novel class (H3) of histamine receptor. Nature (1983) 302:832-837.
  • LEURS R, BLANDINA P, TEDFORD C, TIMMERMAN H: Therapeutic potential of histamine H3 receptor agonists and antagonists. Trends Pharm. Sci. (1998) 19(5):177-183.
  • GIOVANNINI MG, BARTOLINI L, BACCIOTTINI L, GRECO L, BLANDINA P: Effects of histamine H3 receptor agonists and antagonists on cognitive performance and scopolamine- induced amnesia. Behav. Brain Res. (1999) 104:147-155.
  • SMIT MJ, TIMMERMAN H, HIJZELENDOORN JC, LEURS R: Regulation of the human histamine H1 receptor stably expressed in Chinese hamster ovary cells. Br. J. Pharmacol. (1996) 117(6):1071-1080.
  • FUKUI H, FUJIMOTO K, MIZUGUCHI et al.: Molecular cloning of the human histamine H1 receptor gene. Biochem. Biophys. Res. Commun. (1994) 201(2):894-901.
  • SULLIVAN E, TUCKER E, DALE I: Measurement of [Ca2+] using the fluorometric imaging plate reader (FLIPR). In: Methods in Molecular Biology: Calcium Signaling Protocols. Lambert DG (Ed.). Humana Press, New Jersey, (1999):125-136.
  • AXE FU, BEMBENEK SD, SZALMA S: Three-dimensional models of histamine H3 receptor antagonist complexes and their pharmacophore. J. Mol. Graphics Mod. (2006) 24(6):456-464.
  • DEESCH IJ, MILLS JEJ, PERKINS TD et al.: Development of a pharmacophore model for histamine H3 receptor antagonists, using the newly developed molecular modeling program SLATE. J. Med. Chem. (2001) 44(11):1666-1674.
  • WILSON D: The discovery of a novel series of potent, orally active histamine H3 receptor antagonists. Proceedings of the 13th RSC-SCI Medicinal Chemistry Symposium. Cambridge, UK (2005).
  • CURRENT PATENTS GAZETTE: Thomson Scientific (2005) Issue 0538:13.
  • HOWARD HR: 7-Phenylsulfonyl- tetrahydro-3-benzazepine derivatives as antipsychotic agents. Exp. Opin. Ther. Patents (2005) 15(12):1811-1815.

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