Key References
- Biziére, K Gueudet, C Worms, P Further evidence for a cholinomimetic activity of minaprine. Br. J. Pharmacol. 1986 87 31 (suppl)
- Worms, P Kan, JP Steinberg, R Terranova, JP Pério, A Bizière, K Cholinomimetic activities of minaprine. Naunyn-Schmiedeberg's Arch. Pharmacol. 1989 340 411–418.
- Wermuth, CG Bourguignon, JJ Hoffmann, R Kan, JP Worms, P Design and development of selective muscarinic M1 agonists starting from 3-amino-pyridazines. Scientia Pharmaceutica (Wien) 1990 58 169–172.
- Wermuth, CG Bourguignon, JJ Hoffmann, R Novel aminopyridazine-derived selective muscarinic agonists as potential drugs for senile dementia Trends in Medicinal Chemistry 90. Sarel, S, Mechoulam, R, Agranat, I Blackwell Scientific Publications Oxford 1992 135–142.
- Hoffmann, R Bourguignon, JJ Wermuth, CG The active analog approach applied to the identification of the central muscarinic pharmacophore QSAR: Rational Approaches to the Design of Bioactive Compounds. Silipo, C, Vittoria, A Elsevier Science Publishers B.V. Amsterdam 1991 283–292.
- Wermuth, CG Bourguignon, JJ Hoffmann, R Boigegrain, R Brodin, R Kan, JP Soubrié, P SR 46559 and related aminopyridazines are potent muscarinic agonists with no cholinergic syndrome Bio. Med. Chem. Lett in press.
- Schumacher, C Steinberg, R Kan, JP Michaud, JC Bourguignon, JJ Wermuth, CG Feltz, P Worms, P Bizière, K Pharmacological characterization of the aminopyridazine SR 95639A a selective M1 muscarinic agonist. Eur. J. Pharmacol. 1989 166 139–147.
- Kan, JP Steinberg, R Michaud, JC Thurneyssen, O Terranova, JP Gueudet, C Souilhac, J Brodin, R Boigegrain, R Wermuth, CG Worms, P Soubrié, P Le Fur, G SR 46559A: A novel and potent muscarinic agonist with no cholinergic syndrome. Psychopharmacology 1992 In press.
- Boast, CA Leveuter, S Sabb, A Abelson, M Beuder, R Giacomo, D Maurer, S McArthur, S Mehta, O Morris, H Moyer, J Storch, F Biochemical and behavioral characterization of a novel cholinergic agonist, SR 95639. Pharmacol. Biochem. Behav. 1991 39 2 287–292.
- Jenkins, SM Wadsworth, HJ Bromidge, S Orlek, BS Wyman, PA Riley, GJ Hawkins, J Substituent variation in azabicyclic triazole- and tetrazole-based muscarinic receptor ligands. J. Med. Chem. 1992 35 2392–2406.
- Sanofi EP -251937-B.
- Sanofi EP -429344-A.
- Sanofi EP -401333-A.
- Yoshitomi JO 333816.