Advanced search
Publication Cover
Expert Opinion on Therapeutic Patents Volume 4, 1994 - Issue 4
Submit an article Journal homepage
9
Views
9
CrossRef citations to date
0
Altmetric
Research Article

Overview Central & Peripheral Nervous System: Recent developments in serotonin reuptake inhibitors

Gregory M Shutske Neuroscience Strategic Business Unit, Hoechst-Roussel Pharmaceuticals Inc, Route 202-206, PO Box 2500, Somerville, NJ, 08876-1258, USA
Pages 335-341 | Published online: 03 Mar 2008

References to Primarv Literaturess

  • BURTON SW: Int. Clin. Psycbopharmacol. (1991) 6 (Suppl3): 1–17.
  • STOKES PE: Clin. Ther. (1993) 15: 216–43.
  • MILNE RJ, GOA ICI: Drugs (1991) 41: 450–477.A good review of preclinical pharmacology and clinical effects of citalopram as well as SSRIs as a class.
  • MURDOCH D, MCTAVISH D: Drugs (1992) 44: 604–624.
  • DECHANT KL, CLISSOLD SP: Drugs (1991) 41: 225–253.
  • •Good review of paroxetine; good discussion of adaptive changes in serotonin receptors following long-term SSRI administration.
  • FULLER RW, WONG DT, ROBERTSON DW: Med. Res. Rev.(1991) 11: 17–34. Reviews structure-activity relationships for fluoxetine and summa-rizes therapeutic indications other than depression.
  • RUDORFER MV, POTTER WZ: Drugs (1989) 37: 713–738.
  • CHUMPRADIT S, KUNG MP, PANYACHOTIPUN C, PRAPAN-SIRI V, FOULON C, BROOKS BP, SZABO SA, TEJANI-BUIT S, FRAZER A, KUNG HF: J. Med. Chem. (1992) 35: 4492–4497.
  • KUNG MP, CHUMPRADIT S, BILLINGS J, KUNG H: Life Sci. (1992) 51: 95–106.
  • WONG DT, BYMASTER FP, MAYLE DA, REID LR, ICRUSHIN-SKI JH, ROBERTSON DW: Neuropsychopharmacol. (1993) 8: 23–33.
  • VALENTA V, VLKOVA M, VALCHAR M, DOBROVSKY K, POLIVKA Z: Collect. Czech. Chem. Commun. (1991) 56: 1525–1533.
  • MICHALS DR, SMITH HE: Chirality (1993) 5: 20–23.
  • JILEK J, SINDELAR K, POMYKACEK J, ICMONICEK V, SEDIVY Z, Hrubantova M, HOLUBEK J, SVATEK E, RYSKA M, KORUNA I, VALCHAR M, DLABAC A, METYSOVA J, DLOHOZKOVA N, PROTIVA M: Collect. Czech. Cbem. Com-mun. (1989) 54: 3294–3338.
  • SINDELAR K, KMONICEK V, TIRUBANTOVA M, POLIVKA Z:Collect. Czech. Chem. Commun. (1992) 57: 194–203.
  • SINDELAR K, POMYKACEK J, HOLUBEK J, SVATEK E, VALCHAR M, DOBROVSKY K, METYSOVA J, POLIVKA Z: Collect. Czech .Chem. Commun. (1991) 56: 459–477.
  • LEMBERGER L, FULLER RW, ZERBE RE: Clin. Pharmacol.(1985) 8: 299–317.
  • HOGBERG T, ROSS SB, STROM P, BRUNEWALD GL, CREESE MW, BUNCE JD: J. Med. Chem. (1988) 31: 913–919.
  • HANSCH C, CALDWELL J: J. Comput. Aided Mol. Des. (1991) 5: 441–453.
  • MARCUSSON JO, NORINDER U, HOGBERG T, ROSS SB: Eur.J. Pharmacol. (1992) 215: 191–198. QSAR analysis of zimeldine analogues.
  • KAISER C, SETLER PE: Antidepressant Agents In: Burger's Medicinal Chemistry, 4th Ed. (1981). WOLFF ME, (Ed.), Wiley & Sons, New York: 1044–1045.
  • JOHNSON MP, FRESCAS SP, OBERLENDER R, NICHOLS DE:J. Med. Chem. (1991) 34: 1662–1668.
  • FULLER RW, SNODDY HD, ICRUSHINSKI JH, ROBERTSON DW: Neuropharmacol. (1992) 31: 997–1000.
  • WONG DT, BYMASTER FP, REID LR, MAYLE DA, KRUSHIN-SKI JH, ROBERTSON DW: Neuropsychopharmaca (1993) 8: 337–344.
  • WELCH WM, KRASKA AR, SARGES R, KOE BK: J. Med. Chem.(1984) 27: 1508–1515.
  • HYTTEL J, BOGESO KP, PERREGAARD J, SANCHEZ C: J.Neural. Transm. Gen. Sect. (1992) 88: 157–160.
  • SHANK RP, VAUGHT JL, PELLEY KA, SETLER PE, MCCOM-SEY DF, MARYANOFF BE: J. Pharmacol. Exp. Therap. (1988) 247: 1032–1038. Good comparative reuptake, receptor binding, and in vivo pharma-cology for a number of SSR1s.
  • MARYANOFF BE, VAUGHT JL, SHANK RP, MCCOMSEY DF, COSTANZO MJ., NORTEY SO: pled.Chem. (1990) 33: 2793–2797.
  • SMITH DF, JENSEN PN, POULSEN SH, MIKKELSEN EO,ELBAZ E, GLASER R: EurJ.Pharmacol. (1991) 196: 85–92.
  • HABERT E, GRAHAM D, TAHRAHOUI L, CLAUSTRE Y,LANGER SZ: Eur. J. Pharmacol. (1985) 118: 107–114. Evidence that paroxetine labels the 5-HT reuptake transporter, ranks potency of several SSRls.
  • BLEGON A, MATHIS C: Synapse (1993) 13: 1–9.
  • GOBBI M, CERVO L, TADDEI C, MENNINI T: Neurocbem. Int. (1993) 23: 247–251.
  • HRDINA PD, FOY B, HEPNER A, SUMMERS RJ:J. Pbarmacol, Exp. Ther. (1990) 252: 410–418.
  • SUEHIRO M, WILSON AA, SCHEFFEL U, DANNALS RE, RAVERT HT, WAGNER HN, JR: Int.J. Rad. Appl. InstrumMl. (1991) 18: 791–796.
  • MATHIS CA, GERDES JM, ENAS JD, WHITNEY JM, TAYLORSE, ZHANG Y, MCKENNA DJ, HAVLIK S, PEROUTKA SJ: Pharm. Pharmacol. (1992) 44: 801–805. Ranks methyl-substituted paroxetine derivatives for in vitro potency.
  • D'AMATO RJ, LARGENT BL, SNOWMAN AM, SNYDER SH: J. Pharmacy!. Exp. Then (1987) 242: 364–371.
  • KOE BK, LABEL LA, WELCH WM: Psychopbarmacol. (1990) 100: 470–476.
  • HASHIMOTO K, GOROMARU T: J. Pharmacol. Exp. Ther. (1990) 255: 146–153.
  • HASHIMOTO K, GOROMARU T: Eur. J. Pharmacy!. (1990) 180: 273–281.
  • HASHIMOTO K, GOROMARU T Neuropharmacol. (1991) 30:113-117. Evidence that 6-nitroquipazine labels the 5-HT reuptake transporter; ranks potency of several SSRIs.
  • HASHIMOTO K, GOROMARU T Neurophartnacol. (1992) 31: 869–874.
  • MATHIS CA, TAYLOR SE, BIEGON A, ENAS JD: Brain Res.(1993) 619: 229–235.
  • BLEGON A, MATHIS CA, HANRAHAN SM, JAGUST WJ: BrainRes. (1993) 619: 236–246.
  • SUEHIRO M, SCHEFFEL U, DANNALS RF, RAVERT HT, RICAURTE GA, WAGNER HN, JR: J. Nucl. Med. (1993) 34: 120–127.
  • WALDMETER PC, BAUMANN PA: Naunyn Schmiedeberg Arch. Pharmacol. (1983) 324: 20–26.
  • WALDMEIER PC, STOCKLIN K: Eur. J. Pharmacol. (1989) 169: 197–204.
  • WALDMEIER PC, GRAF T, GERMER M, FELDTRAUER JJ, HOWALD H: Biol. Psychiatry (1993) 33: 373–379.
  • WALDMEIER PC: Prog. Neuropsychopharmacol. Biol. Psy-chiatry(1993) 17: 183–198.
  • ANGEL I, SCHOEMAKER H, PROU'TEAU M, GARREAU M, LANGER SZ: Surf. Pharmacol. (1993) 232: 139–145.
  • ANZINI M, CAPPELLI A, VOMERO S, CAMPIANI G., C.AG-NOTTO, A., SKORUPSKA MZ: Farmaco. (1991) 46: 1435–1447.
  • MALLERON JL, GUEREMY C, MIGNANI S, PEYRONEL JF,TRUCHON A, BLANCHARD JC, DOBLE A, LADURON P, PIOT 0, ZUNDEL JL, BETSCHART J, CANARD H, CHAILLOU P, FERRIS 0, HUON C, JUST B, KERPHIRIQUE R, MARTIN B, MOUTON P, RENAUDON A: J. Med. Chem. (1993) 36: 1194–1202.
  • EISON AS, EISON MS, TORRENTE JR, WRIGHT RN, YOCCA D: Psychopharmacol. Bull. (1990) 26: 311–315.
  • DEFRANCE R, MAREY C, KAMOUN A: Clin. Neuropharma-col. (1988) 160 (suppl. 15): S74–S82.
  • MENNINI T, MOCAER E, GARATTINI S: Naunyn Schmiede-berg Arch. Parmacol. (1987) 336: 478–482.
  • PUIG S, RIVOT JP, BESSON JM: Brain Res, (1993) 600: 219–224.
  • BROQUA P, BAUDRIE V, CHAOULOFF F: Eur. Neuropsycho-pharmacol. (1992) 2: 115–120.
  • ZOHAR J, ZOHAR-KADOUCH RC, KINDLER S: Drugs (1992) 43: 210–218.
  • SCHNEIER FR, LIEBOWITZ MR, DAVIES SO, FAIRBANKS J,HOLLANDER E, CAMPEAS R, KLEIN DF: J. Clin. Psychophar-macol. (1990) 10: 119–121.
  • WESTENBERG HG, DEN BOER JA: Pharmacopsychiatry (1993) 26 (Suppl 1): 30–33.
  • WISE SD: Am. J. Clin. Nutr. (1992) 55: 181S–184S.
  • RAMIREZ LC, ROSENSTOCK J, STROWIG S, CERCONE S, RASIUN P: Am. J. Med. (1990) 88: 540–541.
  • POTTER VAN LOON BJ, RADDER JK, FROLICH M, KRANS HM, ZWINDERMAN AU, MEINDERS AE: Int.J. Obes. (1992) 16: 79–85.
  • MEINDERS AE, PIJL H: Mt, J. Obes. (1992) 16 (Suppl 4): S35–S39.
  • BLAKELY RD, BERSON 11E, FREMEAU RT jR, CARON MG,PEEK MM, PRINCE HK, BRADLEY CC: Nature (1991) 354: 66–70. Cloning and expression of the rat 5-HT transporter in HeLa fi-broblasts and inhibition of 5-HT transport by SSRIs.
  • HOFFMAN BJ, MEZEY E, BROWNSTEIN MJ: Science (1991)254: 579–580. Cloning and expression of the rat 5-HT transporter in CV-1 cells and inhibition of 5-HT transport by SSRls.

References to Patent Literature

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Order Reprints Request Corporate Permissions

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

Request Academic Permissions

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.

Related research

People also read lists articles that other readers of this article have read.

Recommended articles lists articles that we recommend and is powered by our AI driven recommendation engine.

Cited by lists all citing articles based on Crossref citations.
Articles with the Crossref icon will open in a new tab.