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Research

Streptogramin analogues

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Pages 115-131 | Published online: 03 Mar 2008

References

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  • The first review on streptogramins.
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  • The reference article on the properties of yirginiamycin-like antibi-otics.
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  • An overview on the chemistry of streptogramins.
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  • A recent review on RP 59500 and pristinamycins.
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  • An important contribution in reviewing the properties of the strep-togramins.
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  • A molecular explanation of the synergistic action of yirginiamycin antibiotics in vim is given.
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  • A relevant article on the biological importance of the 3-hydroxy picolinic acid residue in group B streptogramins.
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  • MOERMAN MC, ANTEUNIS MJO: Partial synthesis of five analogues of the peptido lactone Virginiamycin modified in the fifth and/or sixth position ([Xxx5]-VS1 with Xxx = Ala, Asp, Asn and Lys and [A1a5,G1y61-VS1). Int. J. Peptide Protein Res. (1993) 41:102–117.
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  • ARCHER G, AUGER P, DOERS G, FERRARO MJ, FUCHS P, JORGENSEN J, LOW D, MURRAY P, RELLER LB, STRATTON C, WENNERSTEN, MOELLERING RC: RP 59500, a new streptogramin highly active against recent isolates of North American staphylococcL Diagn. Microbiol. Infect. Dis.(1993) 16(3):223–226.
  • An important contribution to the evaluation of RP 59500
  • FREMAUX A, SISSIA G, COHEN R, GESLIN P: In vitroactivity of RP 59500, a new setnisynthetic strepto-gramin, against Streptococcus pneumoniae. J. Antimi-crob. Chemother. (1992) 30 (Suppl. A):19–24.
  • APPELBAUM PC, SPANGLER SK, JACOBS MR: Susceptibilityof 139 penicillin-susceptible and resistant isolates of Streptococcus pneumoniae to RP 59500, erythromycin, vancomycin, temafloxacin, ciprofloxacin and oflox-acin. 31st International Conference On Antimicrobial Agents And Chemotherapy Chicago, (1991) Abstr. 893.
  • VERBIST L, VERHAEGEN J: Comparative in vitro activityof RP 59500. J. Antimicrob. Chemother. (1992) 30(Suppl. A):39–44.
  • COLLINS L, MALANOSKI G, WENNERSTEN C, ELIOPOULOS MG, FERRARO MJ, MOELLERING RC: In vitro activity of RP 59500 an injectable streptogramin antibiotic, against vancomycin-resistant grain-positive organisms. 32nd International Conference On Antimicrobial Agents And Che-motherapy Anaheim, (1992), Abstr. 1311.
  • SCRIVER SR, TYRRELL G, WILLEY BM, KREISWIRTH BN,LOW DE: In vitro assessment of RP 59500 (RP) against vancomycin-resistant enterococci 33rd International Conference On Antimicrobial Agents And Chemotherapy New Orleans, (1993), Abstr. 1057.
  • COOPER B, ROBINSON A, FREEMAN C, QUINTILIANI II R,MAZENS-SULLTVAN M, NIGHTINGALE C, QUINTILIANI R: Antimicrobial susceptibility of vancomycin-resistant enterococci. 33rd International Conference On Antimicro-bial Agents And Chemotherapy New Orleans, (1993), Abstr. 1053.
  • CASEWELL MW, SEYED-A/CHAVANI M, WADE J: In vitroactivity of RP 59500 against vancomycin-resistant En-terococcus faecium also resistant to 512mg/1 of gen-tamycin. 33rd International Conference On Antimicrobial Agents And Chemotherapy New Orleans,( 1993), Abstr. 1058.
  • NEU HC, CHIN N, GU J: The in vitro activity of newstreptogramins, RP 59500, RP 57669 and RP 54476, alone and in combination. J. Antimicrob. Chemother. (1992) 30(Suppl. A):83–94.
  • DABERNAT H, SEGUY, DELMAS C: In vitro activity of RP59500, a semi-synthetic streptogramin, against Haemo-pbilus influenzae. 33rd International Conference On An-timicrobial Agents And Chemotherapy New Orleans, (1993), Abstr. 226.
  • ANDREW JM, BASWELL F, WISE R: In vitro activity of RP59500 against staphylococci and respiratory patho-gens. 33rd International Conference On Antimicrobial Agents and Chemotherapy New Orleans, US (1993): Abstr. 1044. 72. cc
  • DUBOIS J, JOLY JR: In vitro activity of RP 59500, a new synergistic antibacterial agent, against Legionella spp. J. Antimicrob. Chemother. (1992) 30(Suppl. A):77–82.
  • SOUSSY CJ, ACAR JF, CLUZEL R, COURVALIN P, DUVAL J, FLEURETTE J, MEGRAUD, MEYRAN M, THABAUT A: A collaborative study of the in vitro sensitivity to RP 59500 of bacteria isolated in seven hospitals in France. J. Antimicrob. Chemother. (1992) 30(Suppl. A):53–58.
  • RENAUDIN H, BOUSSENS B, BEBEAR C: In vitro activity of RP 59500 against Mycoplasnsa. 31st International Conference On Antimicrobial Agents And Chemotherapy Chicago, (1991), Abstr. 897.
  • BOUANCHAUD DH: unpublished data.
  • WISE R: unpublished data.
  • LECLERCQ R, NANTAS L, SOUSSY CJ, DUVAL J: Activity of RP 59500, a new parenteral sennlsynthetic strepto-gramin, against staphylococci with various mecha-nisms of resistance to macrolide-lincosamide-streptogramki antibiotics. J. Antimicrob. Chemother. (1992) 30(Suppl. A):67–76.
  • EL SOLH N, LONCLE V, AUBERT S, CASETTA A, ALLIGNET J: Analysis of Staphylococcal elements conferring resis-tance to streptogramin A (RP 54476). 33rd International Conference On Antimicrobial Agents And Chemotherapy New Orleans, (1993), Abstr. 217.
  • HOBAN DJ, WESNOWESKI B, PALATNICK L, ZHANEL CJ, DAVIDSON RJ: In vitro activity of streptogramin RP 59500 against staphylococci, including bactericidal ki-netic studies. J. Antimicrob. Chemother. (1992) 30(Suppl. A):59–66.
  • BRUMEIIT W, HAMILTON-MILLER JMT, SHAH S: In vitro activity of RP 59500, a new semisynthetic strepto-gramin, against Gram-positive bacteria. J. Antimicrob. Chemother. (1992) 30(Suppl. A):29–38.
  • PASCULLE AW, LINDEN PK, MCDEVITT DA, WAGENER JL, MCKNIGHT JL, PAPAFRANGAS EA: Susceptibility of van-comycin-resistant Enterococcus faecium (VREF) to al-ternative antimicrobial agents singly and in combination. 33rd International Conference On Antimicro-bial Agents And Chemotherapy New Orleans, (1993), Abstr. 1060.
  • BOUANCHAUD DH: /n vitro and in vivo synergic activity and fractional inhibitory concentration (FIC) of the components of a sernisynthetic streptogramin, RP
  • J. Antimicrob. Chemother. (1992) 30(Suppl. A):95-99. A reference article on synergistic activity of streptogramin compo-nents
  • CRAIG W, EBERT S: Pharmacodynamyc activities of RP59500 in an animal infection modeL 33rd International Conference On Antimicrobial Agents And Chemotherapy, New Orleans, (1993), Abstr. 470.
  • CHIN NX, NEU HC: Post-antibiotic effect of RP 59500 against gram-positive bacteria compared to other agents. 31st International Conference On Antimicrobial Agents And Chemotherapy, Chicago, (1991), Abstr. 899.
  • A relevant article on post-antibiotic effect
  • NOUGAYREDE A, BERTHAUD N, BOUANCHAUD DH: Post-antibiotic effects of RP 59500 with Staphylococcus aureus. J. Antimicrob. Chemother. (1992) 30(Suppl. A):101–106.
  • ROLIN O, BOUANCHAUD DH: in vivo efficacy of RP59500, a new synergistic antibacterial agent, in Staphy- lococcus aureus and in Streptococcus pneumoniae mouse experimental infections. 30th International Con-ference On Antimicrobial Agents And Chemotherapy, Atlanta, (1991), Abstr. 787.
  • AZOULAY-DUPUIS E, VALLEE E, VEBER B, POCIDALO JJ: Activity of RP 59500, a new semisynthetic strepto-gramin, in mouse pneumonia induced by a macrolide-resistant strain of streptococcus pneumoniae. 31st International Conference On Antimicrobial Agents And Che-motherapy, (1991) Chicago, Abstr. 902.
  • AZOULAY-DUPUIS E, VALLEE E, POCIDALO JJ: Efficacy of RP 59500, a new semisynthetk streptogramin, against penicillin-resistant and multiresistant strains of strep-tococcus pneumoniae. 32nd International Conference On Antimicrobial Agents And Chemotherapy, Anaheim, (1992), Abstr. 1311.
  • CHAMBERS FIF: Studies of RP 59500 in vitro and in a rabbit model of aortic valve endocarditis caused by methicillin-resistant Staphylococcus aureus. j Antimi-crob. Chemother. (1992) 30 (Suppl. A):117–122.
  • FANTIN B., VALLOIS DM., OTTAVIANI M, MAZLERE B, GARRY L, POCIDALO B, CARBON C: Autoradiographic pattern of diffusion of 14C RP 59500 throughout infected cardiac vegetation in rabbits. 33rd International Confer-ence On Antimicrobial Agents And Chemotherapy New Or-leans, (1993), Abstr. 161.
  • BERTHAUD N, MONTAY G, HUET Y, BOURGUES A, BUS-SIERE JC, SAUTEDE M, SELINGUE M, DESNOTTES JF: RP 59500, in vivo bactericidal activity in a model of S. aureus mouse infection: influence of varying the dos-age and the number of treatments. 32nd International Conference On Antimicrobial Agents And Chemotherapy Anaheim, (1992), Abstr. 1315.
  • BERTHAUD N, ROMBI C, HURT Y, BOURGUES A, BUSSIERE JC, SAUTEDE M, SELINGUE M, DESNOTrES JF: RP 59500: In vivo bactericidal activity in Streptococcus pneumo-niae mouse septicemia. 33rd International Conference On Antimicrobial Agents And Chemotherapy New Orleans, (1993), Abstr. 1157.
  • TURCO'I h A, BERGERON MG: Pharmacodynamic inter-action between RP 59500 and Gram-positive bacteria Infecting fibrin dots. Antimicrob. Agents Chemother. (1992) 36(10):2211–2215
  • DESNOTTES JF, DIALLO N: RP 59500:In vitro antistaphy-lococcal bactericidal activity across platelet-fibrin ma-trices compared to that of vancomycin. 33rd International Conference On Antimicrobial Agents And Che-motherapy New Orleans, (1993), Abstact 763.
  • GEORGOPOULOS A, BREYER S, FEISTANER S, STAUFFER F, MARKRISTATHIS A, GEORGOPOULOS M., GRANINGER W: Bactericidal effect of RP 59500 against staphylococci with different phenotypes in a diffusion chamber model in rabbits. 32nd International Conference On An-timicrobial Agents And Chemotherapy Anaheim, (1992), Abstr. 1309.
  • DESNOITIS JF, DIALLO N: Cellular uptake and intracel-lular bactericidal activity of RP 59500 in murine macro-phages. J. Antimicrob. Chemother. (1992) 30(Suppl. A):107–115.
  • ETIENNE SD, MONTAY G, LE LIBOUX A, FRYDMAN A, GARAUD JJ: A phase I, double-blind, placebo-controlled study of the tolerance and phannacokinetic behaviour of RP 59500. J. Antimicrob. Chemother. (1992) 30(Suppl. A):123–131.
  • The first study published on tolerance and pharmacokinetics of RP 59500 in man.

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