Design, formulation and optimization of valsartan transdermal gel containing iso-eucalyptol as novel permeation enhancer: preclinical assessment of pharmacokinetics in Wistar albino rats

Bibliography

• Guo R, Du X, Zhang R, et al. Bioadhesive film formed from a novel organic-inorganic hybrid gel for transdermal drug delivery system. Eur J Pharm Biopharm 2011;79(3):574-83
   PubMed Web of Science ®Google Scholar
• Langer R. Transdermal drug delivery: past progress, current status, and future prospects. Adv Drug Deliv Rev 2004;56(5):557-8
   PubMed Web of Science ®Google Scholar
• Ahad A, Al-Jenoobi FI, Al-Mohizea AM, et al. Systemic delivery of beta-blockers via transdermal route for hypertension. Saudi Pharm J 2014. [ Epub ahead of print]
   Google Scholar
• Ahad A, Al-Jenoobi FI, Al-Mohizea AM, et al. Transdermal delivery of calcium channel blockers for hypertension. Expert Opin Drug Deliv 2013;10(8):1137-53
   PubMed Web of Science ®Google Scholar
• Ahad A, Raish M, Al-Mohizea AM, et al. Enhanced anti-inflammatory activity of carbopol loaded meloxicam nanoethosomes gel. Int J Biol Macromol 2014;67C:99-104
   Google Scholar
• Batheja P, Sheihet L, Kohn J, et al. Topical drug delivery by a polymeric nanosphere gel: formulation optimization and in vitro and in vivo skin distribution studies. J Control Release 2011;149(2):159-67
   PubMed Web of Science ®Google Scholar
• Brown MB, Martin GP, Jones SA, Akomeah FK. Dermal and transdermal drug delivery systems: current and future prospects. Drug Deliv 2006;13(3):175-87
   PubMed Web of Science ®Google Scholar
• Prausnitz MR, Mitragotri S, Langer R. Current status and future potential of transdermal drug delivery. Nat Rev Drug Discov 2004;3(2):115-24
   PubMed Web of Science ®Google Scholar
• Benson HA. Transdermal drug delivery: penetration enhancement techniques. Curr Drug Deliv 2005;2(1):23-33
   PubMedGoogle Scholar
• Smith EW, Maibach HI. Percutaneous penetration enhancers. CRC Press, Florida, Boca Raton; 1995
   Google Scholar
• Smith EW, Maibach HI. Percutaneous penetration enhancers. CRC Press, Florida, Boca Raton; 2005
   Google Scholar
• Ahad A, Aqil M, Kohli K, et al. Chemical penetration enhancers: a patent review. Expert Opin Ther Pat 2009;19(7):969-88
   PubMed Web of Science ®Google Scholar
• Ahad A, Aqil M, Kohli K, et al. Role of novel terpenes in transcutaneous permeation of valsartan: effectiveness and mechanism of action. Drug Dev Ind Pharm 2011;37(5):583-96
   PubMed Web of Science ®Google Scholar
• Sapra B, Jain S, Tiwary AK. Percutaneous permeation enhancement by terpenes: mechanistic view. Aaps J 2008;10(1):120-32
   PubMed Web of Science ®Google Scholar
• Jain R, Aqil M, Ahad A, et al. Basil oil is a promising skin penetration enhancer for transdermal delivery of labetolol hydrochloride. Drug Dev Ind Pharm 2008;34(4):384-9
   PubMed Web of Science ®Google Scholar
• Ahad A, Aqil M, Kohli K, et al. Interactions between novel terpenes and main components of rat and human skin: mechanistic view for transdermal delivery of propranolol hydrochloride. Curr Drug Deliv 2011;8(2):213-24
   PubMed Web of Science ®Google Scholar
• Hassan N, Ahad A, Ali M, Ali J. Chemical permeation enhancers for transbuccal drug delivery. Expert Opin Drug Deliv 2010;7(1):97-112
   PubMed Web of Science ®Google Scholar
• Aqil M, Ahad A, Sultana Y, Ali A. Status of terpenes as skin penetration enhancers. Drug Discov Today 2007;12(23-24):1061-7
   PubMed Web of Science ®Google Scholar
• Palamakula A, Nutan MT, Khan MA. Response surface methodology for optimization and characterization of limonene-based coenzyme Q10 self-nanoemulsified capsule dosage form. AAPS PharmSciTech 2004;5(4):e66
   PubMedGoogle Scholar
• Chang JS, Huang YB, Hou SS, et al. Formulation optimization of meloxicam sodium gel using response surface methodology. Int J Pharm 2007;338(1-2):48-54
   PubMed Web of Science ®Google Scholar
• Govender S, Pillay V, Chetty DJ, et al. Optimisation and characterisation of bioadhesive controlled release tetracycline microspheres. Int J Pharm 2005;306(1-2):24-40
   PubMedGoogle Scholar
• Ahad A, Aqil M, Kohli K, et al. Formulation and optimization of nanotransfersomes using experimental design technique for accentuated transdermal delivery of valsartan. Nanomedicine 2012;8(2):237-49
   PubMed Web of Science ®Google Scholar
• Ahad A, Aqil M, Kohli K, et al. Enhanced transdermal delivery of an anti-hypertensive agent via nanoethosomes: statistical optimization, characterization and pharmacokinetic assessment. Int J Pharm 2013;443(1-2):26-38
   PubMed Web of Science ®Google Scholar
• Gannu R, Palem CR, Yamsani VV, et al. Enhanced bioavailability of lacidipine via microemulsion based transdermal gels: formulation optimization, ex vivo and in vivo characterization. Int J Pharm 2010;388(1-2):231-41
   PubMed Web of Science ®Google Scholar
• Gannu R, Yamsani VV, Yamsani SK, et al. Optimization of hydrogels for transdermal delivery of lisinopril by Box-Behnken statistical design. AAPS PharmSciTech 2009;10(2):505-14
   PubMed Web of Science ®Google Scholar
• Gannu R, Yamsani VV, Palem CR, et al. Iontophoretic delivery of lisinopril: optimization of process variables by Box-Behnken statistical design. Pharm Dev Technol 2010;15(2):169-77
   PubMed Web of Science ®Google Scholar
• Rizwan M, Aqil M, Ahad A, et al. Transdermal delivery of valsartan: I. Effect of various terpenes. Drug Dev Ind Pharm 2008;34(6):618-26
   PubMed Web of Science ®Google Scholar
• Nishida N, Taniyama K, Sawabe T, Manome Y. Development and evaluation of a monolithic drug-in-adhesive patch for valsartan. Int J Pharm 2010;402(1-2):103-9
   PubMed Web of Science ®Google Scholar
• Bhosale SS, Avachat AM. Design and development of ethosomal transdermal drug delivery system of valsartan with preclinical assessment in Wistar albino rats. J Liposome Res 2013;23(2):119-25
   PubMed Web of Science ®Google Scholar
• Ahad A, Aqil M, Ali A. Investigation of antihypertensive activity of carbopol valsartan transdermal gel containing 1,8-cineole. Int J Biol Macromol 2014;64C:144-9
   Google Scholar
• Narishetty ST, Panchagnula R. Transdermal delivery of zidovudine: effect of terpenes and their mechanism of action. J Control Release 2004;95(3):367-79
   PubMed Web of Science ®Google Scholar
• Shakeel F, Baboota S, Ahuja A, et al. Skin permeation mechanism and bioavailability enhancement of celecoxib from transdermally applied nanoemulsion. J Nanobiotechnology 2008;6:8
   PubMedGoogle Scholar
• Yamane MA, Williams AC, Barry BW. Terpene penetration enhancers in propylene glycol/water co-solvent systems: effectiveness and mechanism of action. J Pharm Pharmacol 1995;47(12A):978-89
   PubMed Web of Science ®Google Scholar
• Vaddi HK, Ho PC, Chan SY. Terpenes in propylene glycol as skin-penetration enhancers: permeation and partition of haloperidol, Fourier transform infrared spectroscopy, and differential scanning calorimetry. J Pharm Sci 2002;91(7):1639-51
   PubMed Web of Science ®Google Scholar
• Vaddi HK, Ho PC, Chan YW, Chan SY. Terpenes in ethanol: haloperidol permeation and partition through human skin and stratum corneum changes. J Control Release 2002;81(1-2):121-33
   PubMed Web of Science ®Google Scholar
• Chopra S, Patil GV, Motwani SK. Response surface methodology for optimization of losartan potassium controlled release tablets. J Control Release 2006;116(2):e102-4
   PubMed Web of Science ®Google Scholar
• Khajeh M. Application of Box-Behnken design in the optimization of a magnetic nanoparticle procedure for zinc determination in analytical samples by inductively coupled plasma optical emission spectrometry. J Hazard Mater 2009;172(1):385-9
   PubMed Web of Science ®Google Scholar
• Hughes MF, Shrivastava SP, Fisher HL, Hall LL. Comparative in vitro percutaneous absorption of p-substituted phenols through rat skin using static and flow-through diffusion systems. Toxicol In Vitro 1993;7(3):221-7
   PubMed Web of Science ®Google Scholar
• Ng SF, Rouse JJ, Sanderson FD, et al. Validation of a static Franz diffusion cell system for in vitro permeation studies. AAPS PharmSciTech 2010;11(3):1432-41
   PubMed Web of Science ®Google Scholar
• Crutcher W, Maibach HI. The effect of perfusion rate on in vitro percutaneous penetration. J Invest Dermatol 1969;53(4):264-9
   PubMed Web of Science ®Google Scholar
• Mura S, Manconi M, Sinico C, et al. Penetration enhancer-containing vesicles (PEVs) as carriers for cutaneous delivery of minoxidil. Int J Pharm 2009;380(1-2):72-9
   PubMed Web of Science ®Google Scholar
• Moghimi HR, Makhmalzadeh BS, Manafi A. Enhancement effect of terpenes on silver sulphadiazine permeation through third-degree burn eschar. Burns 2009;35(8):1165-70
   PubMed Web of Science ®Google Scholar
• Narishetty ST, Panchagnula R. Transdermal delivery system for zidovudine: in vitro, ex vivo and in vivo evaluation. Biopharm Drug Dispos 2004;25(1):9-20
   PubMed Web of Science ®Google Scholar
• Chisty MN, Bellantone RA, Taft DR, Plakogiannis FM. In vitro evaluation of the release of albuterol sulfate from polymer gels: effect of fatty acids on drug transport across biological membranes. Drug Dev Ind Pharm 2002;28(10):1221-9
   PubMed Web of Science ®Google Scholar
• Amin S, Kohli K, Khar RK, et al. Mechanism of in vitro percutaneous absorption enhancement of carvedilol by penetration enhancers. Pharm Dev Technol 2008;13(6):533-9
   PubMed Web of Science ®Google Scholar
• Tatar S, Saglik S. Comparison of UV- and second derivative-spectrophotometric and LC methods for the determination of valsartan in pharmaceutical formulation. J Pharm Biomed Anal 2002;30(2):371-5
   PubMed Web of Science ®Google Scholar
• Bachhav YG, Patravale VB. Microemulsion based vaginal gel of fluconazole: formulation, in vitro and in vivo evaluation. Int J Pharm 2009;365(1-2):175-9
   PubMed Web of Science ®Google Scholar
• Paget GM, Barnes JM. Interspecies dosage conversion scheme in evaluation of results and quantitative application in different species. In: Laurence DR, Bacharach AL, editors. Evaluation of drug activities: pharmacometrics. Academic press, London, New York; 1964. p. 160-2
   Google Scholar
• Piao ZZ, Lee ES, Tran HT, Lee BJ. Improved analytical validation and pharmacokinetics of valsartan using HPLC with UV detection. Arch Pharm Res 2008;31(8):1055-9
   PubMed Web of Science ®Google Scholar
• Chaudhary H, Kohli K, Amin S, et al. Optimization and formulation design of gels of Diclofenac and Curcumin for transdermal drug delivery by Box-Behnken statistical design. J Pharm Sci 2011;100(2):580-93
   PubMed Web of Science ®Google Scholar
• Chaudhary H, Rohilla A, Rathee P, Kumar V. Optimization and formulation design of carbopol loaded Piroxicam gel using novel penetration enhancers. Int J Biol Macromol 2013;55:246-53
   PubMed Web of Science ®Google Scholar
• Levison KK, Takayama K, Isowa K, et al. Formulation optimization of indomethacin gels containing a combination of three kinds of cyclic monoterpenes as percutaneous penetration enhancers. J Pharm Sci 1994;83(9):1367-72
   PubMed Web of Science ®Google Scholar
• Cornwell PA, Barry BW, Stoddart CP, Bouwstra JA. Wide-angle X-ray diffraction of human stratum corneum: effects of hydration and terpene enhancer treatment. J Pharm Pharmacol 1994;46(12):938-50
   PubMed Web of Science ®Google Scholar
• Levang AK, Zhao K, Singh J. Effect of ethanol/propylene glycol on the in vitro percutaneous absorption of aspirin, biophysical changes and macroscopic barrier properties of the skin. Int J Pharm 1999;181(2):255-63
   PubMedGoogle Scholar
• Arellano A, Santoyo S, Martin C, Ygartua P. Influence of propylene glycol and isopropyl myristate on the in vitro percutaneous penetration of diclofenac sodium from carbopol gels. Eur J Pharm Sci 1999;7(2):129-35
   PubMed Web of Science ®Google Scholar
• Krishnaiah YS, Satyanarayana V, Karthikeyan RS. Effect of the solvent system on the in vitro permeability of nicardipine hydrochloride through excised rat epidermis. J Pharm Pharm Sci 2002;5(2):123-30
   PubMed Web of Science ®Google Scholar
• Sarpotdar PP, Zatz JL. Evaluation of penetration enhancement of lidocaine by nonionic surfactants through hairless mouse skin in vitro. J Pharm Sci 1986;75(2):176-81
   PubMed Web of Science ®Google Scholar
• Lucero MJ, Vigo J, Leon MJ. A study of shear and compression deformations on hydrophilic gels of tretinoin. Int J Pharm 1994;106:25-133
   Google Scholar
• Sultana S, Bhavna Iqbal Z, et al. Lacidipine encapsulated gastroretentive microspheres prepared by chemical denaturation for pylorospasm. J Microencapsul 2009;26(5):385-93
   PubMed Web of Science ®Google Scholar
• Gannu R, Palem CR, Yamsani SK, et al. Enhanced bioavailability of buspirone from reservoir-based transdermal therapeutic system, optimization of formulation employing Box-Behnken statistical design. AAPS PharmSciTech 2010;11(2):976-85
   PubMed Web of Science ®Google Scholar