100
Views
12
CrossRef citations to date
0
Altmetric
Drug Profile

Tapentadol immediate-release for acute pain

Pages 861-869 | Published online: 09 Jan 2014

References

  • Shavit Y, Fridel K, Beilin B. Postoperative pain management and proinflammatory cytokines: animal and human studies. J. Neuroimmune Pharmacol.1(4), 443–451 (2006).
  • Pogatzki-Zahn EM, Zahn PK. From preemptive to preventive analgesia. Curr. Opin. Anaesthesiol.19(5), 551–555 (2006).
  • Moore RA, McQuay HJ. Prevalence of opioid adverse events in chronic non-malignant pain: systematic review of randomized trials of oral opioids. Arthritis Res. Ther.7, R1046–R1051 (2005).
  • Pergolizzi J, Böger RH, Budd K et al. Opioids and the management of chronic severe pain in the elderly: consensus statement of an International Expert Panel with focus on the six clinically most often used World Health Organization Step III opioids (buprenorphine, fentanyl, hydromorphone, methadone, morphine, oxycodone). Pain Pract.8(4), 287–313 (2008).
  • Hartrick CT. Multimodal postoperative pain management. Am. J. Health Syst. Pharm.61(Suppl. 1), S4–S10 (2004).
  • Wheeler M, Oderda GM, Ashburn MA, Lipman AG. Adverse effects associated with postoperative opioid analgesia: a systematic review. J. Pain3, 159–180 (2002).
  • Gaskell H, Derry S, Moore RA, McQuay HJ. Single dose oral oxycodone and oxycodone plus paracetamol (acetaminophen) for acute postoperative pain in adults. Cochrane Database Syst. Rev.3, CD002763 (2009).
  • Toms L, Derry S, Moore RA, McQuay HJ. Single dose oral paracetamol (acetaminophen) with codeine for postoperative pain in adults. Cochrane Database Syst. Rev.1, CD001547 (2009).
  • Myers RP, Shaheen AA, Li B, Dean S, Quan H. Impact of liver disease, alcohol abuse, and unintentional ingestions on the outcomes of acetaminophen overdose. Clin. Gastroenterol. Hepatol.6(8), 918–925 (2008).
  • Gan TJ, Lubarsky DA, Flood EM et al. Patient preferences for acute pain treatment. Br. J. Anaesth.92(5), 681–688 (2004).
  • Revees RR, Burke RS. Tramadol: basic pharmacology and emerging concepts. Drugs Today (Barc.)44(11), 827–836 (2008).
  • Raffa RB, Friderichs E. The basic science aspect of tramadol hydrochloride. Pain Rev.3, 249–271 (1996).
  • Epstein DH, Preston KL, Jasinski DR. Abuse liability, behavioral pharmacology, and physical-dependence potential of opioids in humans and laboratory animals: lessons from tramadol. Biol. Psychol.73, 90–99 (2006).
  • Poulsen L, Arendt-Nielsen L, Brosen K, Sindrup SH. The hypoalgesic effect of tramadol in relation to CYP2D6. Clin. Pharmacol. Ther.60, 636–644 (1996).
  • Zhou SF. Polymorphism of human cytochrome P450 2D6 and its clinical significance: part II. Clin. Pharmacokinet.48(12), 761–804 (2009).
  • Foster A, Mobley E, Wang Z. Complicated pain management in a CYP450 2D6 poor metabolizer. Pain Pract.7(4), 352–356 (2007).
  • Tzschentke TM, De Vry J, Terlinden R et al. Tapentadol hydrochloride: analgesic mu-opioid receptor agonist noradrenaline reuptake inhibitor. Drugs Future31(12), 1053–1061 (2006).
  • Tzschentke TM, Christoph T, Kögel B et al. (-)-(1R,2R)-3-(3-dimethylamino-1-ethyl-2-methyl-propyl)-phenol hydrochloride (tapentadol HCl): a novel mu-opioid receptor agonist/norepinephrine reuptake inhibitor with broad-spectrum analgesic properties. J. Pharmacol. Exp. Ther.323(1), 265–276 (2007).
  • Hartrick CT. Tapentadol immediate release for the relief of moderate-to-severe acute pain. Expert Opin. Pharmacother.10(16), 2687–2696 (2009).
  • Monory K, Greiner E, Sartania N et al. Opioid binding profiles of new hydrazone, oxime, carbazone and semicarbazone derivatives of 14-alkoxymorphinans. Life Sci.64(22), 2011–2020 (1999).
  • Terlinden R, Ossig J, Fliegert F, Lange C, Göhler K. Absorption, metabolism, and excretion of 14C-labeled tapentadol HCl in healthy male subjects. Eur. J. Drug Metab. Pharmacokinet.32(3), 163–169 (2007).
  • Lötsch J, Weiss M, Ahne G, Kobal G, Geisslinger G. Pharmacokinetic modeling of M6G formation after oral administration of morphine in healthy volunteers. Anesthesiology90(4), 1026–1038 (1999).
  • Kneip C, Terlinden R, Beier H, Chen G. Investigations into drug–drug interaction potential of tapentadol in human liver microsomes and fresh human hepatocytes. Drug Metab. Lett.2, 67–75 (2008).
  • Smit JW, Oh C, Rengelshausen J et al. Effects of acetaminophen, naproxen, and acetylsalicylic acid on tapentadol pharmacokinetics: results of two randomized, open-label, crossover, drug–drug interaction studies. Pharmacotherapy30(1), 25–34 (2010).
  • Mangold B, Oh C, Jaeger D et al. The pharmacokinetics of tapentadol are not affected by omeprazole: results of a 2-way crossover drug-interaction study in healthy subjects. Pain Pract.7(S1), 55 (2007).
  • Smit J, Oh C, Mangold B et al. Effects of metoclopramide on tapentadol pharmacokinetics: results of an open-label, cross-over, drug–drug interaction study. J. Clin. Pharmacol.49, 1104 (2009) (Abstract 62).
  • Smit J, Oh C, Lannie C et al. Effects of probenecid on tapentadol immediate release pharmacokinetics: results of an open-label, crossover, drug–drug interaction study. J. Clin. Pharmacol.49, 1104 (2009) (Abstract 61).
  • Gardner JS, Blough D, Drinkard CR et al. Tramadol and seizures: a surveillance study in a managed care population. Pharmacotherapy20(12), 1423–1431 (2000).
  • Kleinert R, Lange C, Steup A et al. Single dose analgesic efficacy of tapentadol in postsurgical dental pain: the results of a randomized, double-blind, placebo-controlled study. Anesth. Analg.107(6), 2048–2055 (2008).
  • Stegmann JU, Weber H, Steup A et al. The efficacy and tolerability of multiple-dose tapentadol immediate release for the relief of acute pain following orthopedic (bunionectomy) surgery. Curr. Med. Res. Opin.24(11), 3185–3196 (2008).
  • Daniels SE, Upmalis D, Okamoto A, Lange C, Häeussler J. A randomized, double-blind, Phase III study comparing multiple doses of tapentadol IR, oxycodone IR, and placebo for postoperative (bunionectomy) pain. Curr. Med. Res. Opin.25(3), 765–776, (2009).
  • Daniels S, Casson E, Stegmann JU et al. A randomized, double-blind, placebo-controlled Phase 3 study of the relative efficacy and tolerability of tapentadol IR and oxycodone IR for acute pain. Curr. Med. Res. Opin.25(6), 1551–1561 (2009).
  • Hartrick C, Van Hove I, Stegmann JU, Oh C, Upmalis D. Efficacy and tolerability of tapentadol immediate release and oxycodone HCl immediate release in patients awaiting primary joint replacement surgery for end-stage joint disease: a 10-day, Phase III, randomized, double-blind, active- and placebo-controlled study. Clin. Ther.31(2), 260–271 (2009).
  • Hale M, Upmalis D, Okamoto A, Lange C, Rauschkolb C. Tolerability of tapentadol immediate release in patients with lower back pain or osteoarthritis of the hip or knee over 90 days: a randomized, double-blind study. Curr. Med. Res. Opin.25(5), 1095–1104 (2009).
  • Upmalis D, Lange C, Okamoto A et al. A pooled analysis of the incidence of treatment-emergent adverse events in Phase 2/3 studies of tapentadol IR. Pain Pract.9(S1), 163 (2009).
  • Wesson DR, Ling W. The Clinical Opiate Withdrawal Scale (COWS). J. Psychoactive Drugs35(2), 253–259 (2003).
  • Handelsman L, Cochrane KJ, Aronson MJ et al. Two new rating scales for opiate withdrawal. Am. J. Drug Alcohol Abuse13(3), 293–308 (1987).
  • Antman EM, Bennett JS, Daugherty A, Furberg C, Roberts H, Taubert KA. Use of nonsteroidal anti-inflammatory drugs: an update for clinicians. A scientific statement from the American Heart Association. Circulation115, 1634–1642 (2007).
  • Tannenbaum H, Bombardier C, Davis P, Russell AS; Third Canadian Consensus Conference Group. An evidence-based approach to prescribing nonsteroidal anti-inflammatory drugs. Third Canadian Consensus Conference. J. Rheumatol.33, 140–157 (2006).
  • Desai SP, Solomon DH, Abramson SB et al. The American College of Rheumatology Ad Hoc Group on Use of Selective and Nonselective Nonsteroidal Anti-inflammatory Drugs. Recommendations for the use of selective and non-selective anti-inflammatory drugs: an American College of Rheumatology white paper. Arthritis Rheum.59, 1058–1073 (2008).
  • AGS Panel on the Pharmacological Management of Persistent Pain in Older Persons. Pharmacological management of persistent pain in older persons. J. Am. Geriatr. Soc.57(8), 1331–1346 (2009).
  • Kuehn BM. New pain guideline for older patients: avoid NSAIDs, consider opioids. JAMA302, 19 (2009).
  • Avouac J, Gossec L, Dougados M. Efficacy and safety of opioids for osteoarthritis: a meta-analysis of randomized controlled trials. Osteoarthritis Cartilage15, 957–965 (2007).
  • Leandro G. Meta-analysis in Medical Research. Blackwell Publishing, Ltd, Malden, MA, USA (2005).

Websites

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.