66
Views
0
CrossRef citations to date
0
Altmetric
Original Research

Novel N-phenylcarbamothioylbenzamides with anti-inflammatory activity and prostaglandin E2 inhibitory properties

, , , , &
Pages 883-892 | Published online: 28 Aug 2013

References

  • Gülkok Y Biçer T Kaynak Onurdag F Özgen S Şahin MF Doğruer DS Synthesis of some new urea and thiourea derivatives and evaluation of their antimicrobial activities Turkish Journal of Chemistry 2012 36 279 291
  • Struga M Rosolowski S Kossakowski J Stefanska J Synthesis and microbiological activity of thiourea derivatives of 4-azatricyclo[5.2.2.0(2,6)]undec-8-ene-3,5-dione Arch Pharm Res 2010 33 1 47 54 20191342
  • Liav A Angala SK Brennan PJ Jackson M N-D-aldopentofuranosyl-N′-[p-(isoamyloxy)phenyl]-thiourea derivatives: potential anti-TB therapeutic agents Bioorg Med Chem Lett 2008 18 8 2649 2651 18362068
  • Walchshofer N Delabre-Defayolle I Paris J Petavy AF In vivo morphological damage induced by a new benzimidazole prodrug in Echinococcus multilocularis metacestodes J Pharm Sci 1990 79 7 606 608 2118956
  • Mishra A Srivastava K Tripathi R Puri SK Batra S Search for new pharmacophores for antimalarial activity. Part III: synthesis and bioevaluation of new 6-thioureido-4-anilinoquinazolines Eur J Med Chem 2009 44 11 4404 4412 19586687
  • Çıkla P Küçükgüzel ŞG Küçükgüzel I Synthesis and evaluation of antiviral, antitubercular and anticancer activities of some novel thioureas derived from 4-aminobenzohydrazide hydrazones Marmara Eczacılık Dergisi [Marmara Pharmaceutical Journal] 2010 14 1 13 20
  • Patel RB Chikhalia KH Pannecouque C de Clercq E Synthesis of novel PETT analogues: 3,4-dimethoxy phenyl ethyl 1,3,5-triazinyl thiourea derivatives and their antibacterial and anti-HIV studies J Braz Chem Soc 2007 18 2 312 321
  • Kayser H Eilinger P Metabolism of diafenthiuron by microsomal oxidation: procide activation and inactivation as mechanisms contributing to selectivity Pest Manag Sci 2001 57 10 975 980 11695192
  • Ramadas K Suresh G Janarthanan N Masilamani S Antifungal activity of 1,3-disubstituted symmetrical and unsymmetrical thioureas Pest Manag Sci 1998 52 2 145 151
  • Ke SY Xue SJ Synthesis and herbicidal activity of N-(o-fluoro-phenoxy-acetyl) thioureas derivatives and related fused heterocyclic compounds Arkivoc 2001 10 63 68
  • Kumar S Awasthi V Kanwar JK Influence of growth regulators and nitrogenous compounds on in vitro bulblet formation and growth in oriental lily Horticultural Science (Prague) 2007 34 2 77 83
  • Lee J Kim J Kim SY N-(3-Acyloxy-2-benzylpropyl)-N′-(4-hydroxy-3-methoxybenzyl) thiourea derivatives as potent vanilloid receptor agonists and analgesics Bioorg Med Chem 2001 9 1 19 32 11197340
  • Liu W Zhou J Zhang T Design and synthesis of thiourea derivatives containing a benzo[5,6]cyclohepta[1,2-b]pyridine moiety as potential antitumor and anti-inflammatory agents Bioorg Med Chem Lett 2012 22 8 2701 2704 22450132
  • Cherala S Lingabathula H Ganta R Ampati S Manda S Synthesis and anti-inflammatory activity of a novel series of diphenyl-1,2,4-triazoles and related derivatives J Chem 2012 9 4 2510 2515
  • Amr AE Sabry NM Abdulla MM Synthesis, reactions, and anti-inflammatory activity of heterocyclic systems fused to a thiophene moiety using citrazinic acid as synthon Monatshefte für Chemie – Chemical Monthly 2007 138 7 699 707
  • Wang JY Yamasaki S Takeuchi K Okabe S Delayed healing of acetic acid-induced gastric ulcers in rats by indomethacin Gastroenterology 1989 96 2 Pt 1 393 402 2910759
  • Konturek PK Brzozowski T Konturek SJ Dembiński A Role of epidermal growth factor, prostaglandin, and sulfhydryls in stress-induced gastric lesions Gastroenterology 1990 99 6 1607 1615 2227276
  • Takeuchi K Pathogenesis of NSAID-induced gastric damage: importance of cyclooxygenase inhibition and gastric hypermotility World J Gastroenterol 2012 18 18 2147 2160 22611307
  • Limban C Missir AV Chirita IC Neagu AF Draghici C Chifiriuc MC Synthesis and antimicrobial evaluation of some new 2-(4-fluoro-phenoxymethyl) benzoic acid thioureides Revista de Chimie (Bucharest) 2011 62 168 173
  • Limban C Marutescu L Chifiriuc MC Synthesis, spectroscopic properties and antipathogenic activity of new thiourea derivatives Molecules 2011 16 9 7593 7607 21900862
  • Bahi A Sadek B Schwed SJ Walter M Stark H Influence of the novel histamine H3 receptor antagonist ST1283 on voluntary alcohol consumption and ethanol-induced place preference in mice Psychopharmacology (Berl) 2013 228 1 85 95 23474889
  • Koo HJ Lim KH Jung HJ Park EH Anti-inflammatory evaluation of gardenia extract, geniposide and genipin J Ethnopharmacol 2006 103 3 496 500 16169698
  • Komeshima N Osowa T Nishitoba T Jinno Y Kiriu T Synthesis and anti-inflammatory activity of antioxidants, 4-alkylthio-o-anisidine derivatives Chem Pharm Bull (Tokyo) 1992 40 2 351 356 1535026
  • Winter CA Risley EA Nuss GW Carrageenin-induced edema in hind paw of the rat as an assay for antiiflammatory drugs Proc Soc Exp Biol Med 1962 111 544 547 14001233
  • Ackrell J Antonio Y Franco F Synthesis and antiinflammatory activity of 6,11-dihydro-11-oxodibenzo[b,e]thiepinalkanoic acids and related compounds J Med Chem 1978 21 10 1035 1044 309946
  • Dunn JP Muchowski JM Nelson PH Antiinflammatory 5,6-dihydro-11-oxodibenz[b,e]azepine-3-acetic acids J Med Chem 1981 24 9 1097 1099 6974784
  • Erol DD Sunal R Duru S Synthesis and screening of analgesic and anti-inflammatory activity of 6-acyl-3-(4-substituted benzoylmethyl)-2(3H)-benzoxazolones Arzneimittelforschung 1990 40 4 478 480 2357250
  • Barsoum FF Hosni HM Girgis AS Novel bis(1-acyl-2-pyrazolines) of potential anti-inflammatory and molluscicidal properties Bioorg Med Chem 2006 14 11 3929 3937 16460945
  • Khayyal MT El-Ghazaly MA Abdallah DM Okpanyi SN Kelber O Weiser D Mechanisms involved in the anti-inflammatory effect of a standardized willow bark extract Arzneimittelforschung 2005 55 11 677 687 16366042
  • Edwards JC Sedgwick AD Willoughby DA The formation of a structure with the features of synovial lining by subcutaneous injection of air: an in vivo tissue culture system J Pathol 1981 134 2 147 156 7019400
  • Rasheed A Kumar CK Mishra A Synthesis, hydrolysis studies and phamacodynamic profiles of amide prodrugs of dexibuprofen with amino acids J Enzyme Inhib Med Chem 2011 26 5 688 695 21250819
  • Bekhit AA Fahmy HT Design and synthesis of some substituted 1H-pyrazolyl-oxazolidines or 1H-pyrazolyl-thiazolidines as anti-inflammatory-antimicrobial agents Arch Pharm (Weinheim) 2003 336 2 111 118 12761764