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Original Research

Oral fondaparinux: use of lipid nanocapsules as nanocarriers and in vivo pharmacokinetic study

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Pages 2941-2951 | Published online: 21 Nov 2011

References

  • De CaterinaRHustedSWallentinLAnticoagulants in heart disease: current status and perspectivesEur Heart J200728788091317426080
  • WeitzDSWeitzJIUpdate on heparin: what do we need to know?J Thromb Thrombolysis201029219920719882363
  • MotlekarNAYouanBBThe quest for non-invasive delivery of bioactive macromolecules: a focus on heparinsJ Control Release200611329110116777255
  • WeitzJINew oral anticoagulants in developmentThromb Haemost20101031627020062934
  • GarciaDLibbyECrowtherMAThe new oral anticoagulantsBlood20101151152019880491
  • MavrakanasTBounameauxHThe potential role of new oral anti-coagulants in the prevention and treatment of thromboembolismPharmacol Ther20111301465821185864
  • TurpieAGDirect Factor Xa and direct thrombin inhibitors: a clinical trial updateCurr Opin Drug Discov Devel2009124497508
  • ThanouMHendersonSKydonieusAElsonCN-sulfonato-N,O-carboxymethylchitosan: a novel polymeric absorption enhancer for the oral delivery of macromoleculesJ Control Release2007117217117817184870
  • Bernkop-SchnurchAKastCEGuggiDPermeation enhancing polymers in oral delivery of hydrophilic macromolecules: thiomer/GSH systemsJ Control Release20039329510314636716
  • VetterAPereraGLeithnerKKlimaGBernkop-SchnurchADevelopment and in vivo bioavailability study of an oral fondaparinux delivery systemEur J Pharm Sci2010413–448949720705133
  • Khafagyel-SMorishitaMOnukiYTakayamaKCurrent challenges in non-invasive insulin delivery systems: a comparative reviewAdv Drug Deliv Rev200759151521154617881081
  • LamprechtAUbrichNMaincentPOral low molecular weight heparin delivery by microparticles from complex coacervationEur J Pharm Biopharm200767363263817540548
  • JiaoYUbrichNMarchand-ArvierMIn vitro and in vivo evaluation of oral heparin-loaded polymeric nanoparticles in rabbitsCirculation2002105223023511790706
  • HoffartVUbrichNLamprechtAMicroencapsulation of low molecular weight heparin into polymeric particles designed with biodegradable and nonbiodegradable polycationic polymersDrug Deliv20031011712554358
  • PorterCJPoutonCWCuineJFCharmanWNEnhancing intestinal drug solubilisation using lipid-based delivery systemsAdv Drug Deliv Rev200860667369118155801
  • MartinsSSarmentoBFerreiraDCSoutoEBLipid-based colloidal carriers for peptide and protein delivery – liposomes versus lipid nanoparticlesInt J Nanomedicine20072459560718203427
  • ChakrabortySShuklaDMishraBSinghSLipid – an emerging platform for oral delivery of drugs with poor bioavailabilityEur J Pharm Biopharm200973111519505572
  • GotoTMorishitaMNishimuraKNovel mucosal insulin delivery systems based on fusogenic liposomesPharm Res200623238439116382280
  • TakeuchiHMatsuiYYamamotoHKawashimaYMucoadhesive properties of carbopol or chitosan-coated liposomes and their effectiveness in the oral administration of calcitonin to ratsJ Control Release2003862–323524212526820
  • HeurtaultBSaulnierPPechBProustJEBenoitJPA novel phase inversion-based process for the preparation of lipid nanocarriersPharm Res200219687588012134960
  • LacoeuilleFHindreFMoalFIn vivo evaluation of lipid nanocapsules as a promising colloidal carrier for paclitaxelInt J Pharm20073441–214314917646066
  • HureauxJLagarceFGagnadouxFLipid nanocapsules: ready-to-use nanovectors for the aerosol delivery of paclitaxelEur J Pharm Biopharm200973223924619560538
  • PeltierSOgerJMLagarceFCouetWBenoitJPEnhanced oral paclitaxel bioavailability after administration of paclitaxel-loaded lipid nanocapsulesPharm Res20062361243125016715372
  • RogerELagarceFBenoitJPThe gastrointestinal stability of lipid nanocapsulesInt J Pharm2009379226026519524655
  • CoonJSKnudsonWClodfelterKLuBWeinsteinRSSolutol HS 15, nontoxic polyoxyethylene esters of 12-hydroxystearic acid, reverses multidrug resistanceCancer Res19915138979021988130
  • RogerELagarceFGarcionEBenoitJPLipid nanocarriers improve paclitaxel transport throughout human intestinal epithelial cells by using vesicle-mediated transcytosisJ Control Release2009140217418119699246
  • HureauxJLagarceFGagnadouxFToxicological study and efficacy of blank and paclitaxel-loaded lipid nanocapsules after i.v. administration in micePharm Res201027342143020054705
  • TurpieAGErikssonBILassenMRBauerKAFondaparinux, the first selective factor Xa inhibitorCurr Opin Hematol200310532733212913785
  • DonatFDuretJPSantoniAThe pharmacokinetics of fondaparinux sodium in healthy volunteersClin Pharmacokinet200241Suppl 21912383039
  • SchieleFFondaparinux and acute coronary syndromes: update on the OASIS 5–6 studiesVasc Health Risk Manag2010617918720407625
  • SantiRContinoLGattoSLevisAFondaparinux in major orthopedic surgical patientsIntern Emerg Med20105216720195927
  • BauerKAHawkinsDWPetersPCFondaparinux, a synthetic pentasaccharide: the first in a new class of antithrombotic agents – the selective factor Xa inhibitorsCardiovasc Drug Rev2002201375212070533
  • RosencherNBellamyLArnaoutLShould new oral antico-agulants replace low-molecular-weight heparin for thromboprophylaxis in orthopaedic surgery?Arch Cardiovasc Dis2009102432733319427610
  • FrankRDSchabbauerGHolscherTThe synthetic pentasaccharide fondaparinux reduces coagulation, inflammation and neutrophil accumulation in kidney ischemia-reperfusion injuryJ Thromb Haemost20053353154015748244
  • HeurtaultBSaulnierPPechBThe influence of lipid nanocapsule composition on their size distributionEur J Pharm Sci2003181556112554073
  • RawatAMajumderQHAhsanFInhalable large porous microspheres of low molecular weight heparin: in vitro and in vivo evaluationJ Control Release2008128322423218471921
  • KhokhlovVYSelemenevVFKhokhlovaONShcherbininRLHeparin determination by spectrophotometric and photocolorimetric methodsPharm Chem J1999338450451
  • MotlekarNASrivenugopalKSWachtelMSYouanBBModulation of gastrointestinal permeability of low-molecular-weight heparin by L-arginine: in-vivo and in-vitro evaluationJ Pharm Pharmacol200658559159816640827
  • KlaefflingCPiechottkaGDaemgen-von BrevernGDevelopment and clinical evaluation of two chromogenic substrate methods for monitoring fondaparinux sodiumTher Drug Monit200628337538116778722
  • BianchiniPBergonziniGLParmaBOsimaBRelationship between plasma antifactor Xa activity and the antithrombotic activity of heparins of different molecular massHaemostasis19952562882988586320
  • StangierJClinical pharmacokinetics and pharmacodynamics of the oral direct thrombin inhibitor dabigatran etexilateClin Pharmacokinet200847528529518399711
  • RogerELagarceFBenoitJPDevelopment and characterization of a novel lipid nanocapsule formulation of Sn38 for oral administrationEur J Pharm Biopharm201179118118821303693
  • HuynhNTPassiraniCSaulnierPBenoitJPLipid nanocapsules: a new platform for nanomedicineInt J Pharm2009379220120919409468
  • HirsjarviSQiaoYRoyereABibetteJBenoitJPLayer-by-layer surface modification of lipid nanocapsulesEur J Pharm Biopharm201076220020720656028
  • MeissnerYUbrichNEl GhazouaniFMaincentPLamprechtALow molecular weight heparin loaded pH-sensitive microparticlesInt J Pharm20073351–214715317150317
  • PeiraECarlottiMETrottaCCavalliRTrottaMPositively charged microemulsions for topical applicationInt J Pharm20083461–211912317618070
  • BaeKHMoonCWLeeYParkTGIntracellular delivery of heparin complexed with chitosan-g-poly(ethylene glycol) for inducing apoptosisPharm Res20092619310018777202
  • MoriSMatsuuraARama PrasadYVTakadaKStudies on the intestinal absorption of low molecular weight heparin using saturated fatty acids and their derivatives as an absorption enhancer in ratsBiol Pharm Bull200427341842114993814
  • MalkovDWangHZDinhSGomez-OrellanaIPathway of oral absorption of heparin with sodium N-[8-(2-hydroxybenzoyl)amino] caprylatePharm Res20021981180118412240944
  • MoazedBHiebertLMMovement of heparins across rat gastric mucosa is dependent on molecular weight and pHPharm Res200926118919518937058
  • Rama PrasadYVMinamimotoTYoshikawaYIn situ intestinal absorption studies on low molecular weight heparin in rats using labrasol as absorption enhancerInt J Pharm20042711–222523215129989
  • Scala-BertolaJRabiskovaMLecompteTBonneauxFMaincentPGranules in the improvement of oral heparin bioavailabilityInt J Pharm20093741–2121619446753
  • MousaSAZhangFAljadaAPharmacokinetics and pharmaco-dynamics of oral heparin solid dosage form in healthy human subjectsJ Clin Pharmacol200747121508152018048572
  • BerkowitzSDMarderVJKosuticGBaughmanRAOral heparin administration with a novel drug delivery agent (SNAC) in healthy volunteers and patients undergoing elective total hip arthroplastyJ Thromb Haemost2003191914191912941031
  • HoffartVLamprechtAMaincentPLecompteTVigneronCUbrichNOral bioavailability of a low molecular weight heparin using a polymeric delivery systemJ Control Release20061131384216697485
  • RogerELagarceFGarcionEBenoitJPBiopharmaceutical parameters to consider in order to alter the fate of nanocarriers after oral deliveryNanomedicine (Lond)20105228730620148639
  • StangierJRathgenKStahleHGansserDRothWThe pharmacokinetics, pharmacodynamics and tolerability of dabigatran etexilate, a new oral direct thrombin inhibitor, in healthy male subjectsBr J Clin Pharmacol200764329230317506785