Effect of particle size on oral absorption of carvedilol nanosuspensions: in vitro and in vivo evaluation

References

• KawabataYWadaKNakataniMYamadaSOnoueSFormulation design for poorly water-soluble drugs based on biopharmaceutics classification system: basic approaches and practical applicationsInt J Pharm2011420111021884771
   PubMed Web of Science ®Google Scholar
• ChenHKhemtongCYangXChangXGaoJNanonization strategies for poorly water-soluble drugsDrug Discov Today201116735436020206289
   PubMed Web of Science ®Google Scholar
• LipinskiCAPoor aqueous solubility-an industry wide problem in ADME screeningAm Pharm Rev200258285
   Google Scholar
• LipinskiCALombardoFDominyBWFeeneyPJExperimental and computational approaches to estimate solubility and permeability in drug discovery and development settingsAdv Drug Deliv Rev201264417
   Web of Science ®Google Scholar
• PaudelAWorkuZAMeeusJGunsSVan den MooterGManufacturing of solid dispersions of poorly water soluble drugs by spray drying: formulation and process considerationsInt J Pharm2013453125328422820134
   PubMed Web of Science ®Google Scholar
• YanY-DSungJHKimKKNovel valsartan-loaded solid dispersion with enhanced bioavailability and no crystalline changesInt J Pharm2012422120221022085435
   PubMedGoogle Scholar
• ShakeelFFaisalMSNanoemulsion: a promising tool for solubility and dissolution enhancement of celecoxibPharm Dev Technol2010151535619552546
   PubMed Web of Science ®Google Scholar
• TaoTZhaoYWuJZhouBPreparation and evaluation of itraconazole dihydrochloride for the solubility and dissolution rate enhancementInt J Pharm2009367110911418930795
   PubMedGoogle Scholar
• BreitenbachJMelt extrusion: from process to drug delivery technologyEur J Pharm Biopharm200254210711712191680
   PubMed Web of Science ®Google Scholar
• LakshmanJPCaoYKowalskiJSerajuddinATApplication of melt extrusion in the development of a physically and chemically stable high-energy amorphous solid dispersion of a poorly water-soluble drugMol Pharm200856994100219434852
   PubMed Web of Science ®Google Scholar
• FenskeDBChonnACullisPRLiposomal nanomedicines: an emerging fieldToxicol Pathol2008361212918337218
   PubMed Web of Science ®Google Scholar
• MohammedAWestonNCoombesAFitzgeraldMPerrieYLiposome formulation of poorly water soluble drugs: optimisation of drug loading and ESEM analysis of stabilityInt J Pharm20042851233415488676
   PubMedGoogle Scholar
• ZhuangCYLiNWangMPreparation and characterization of vinpocetine loaded nanostructured lipid carriers (NLC) for improved oral bioavailabilityInt J Pharm20103941–217918520471464
   PubMed Web of Science ®Google Scholar
• LinCChenFYeTA novel oral delivery system consisting in “drug-in cyclodextrin-in nanostructured lipid carriers” for poorly water-soluble drug: vinpocetineInt J Pharm20144651–2909624530388
   PubMedGoogle Scholar
• LukyanovANTorchilinVPMicelles from lipid derivatives of water-soluble polymers as delivery systems for poorly soluble drugsAdv Drug Deliv Rev20045691273128915109769
   PubMed Web of Science ®Google Scholar
• LuYParkKPolymeric micelles and alternative nanonized delivery vehicles for poorly soluble drugsInt J Pharm2013453119821422944304
   PubMed Web of Science ®Google Scholar
• PatravaleVBDateAAKulkarniRMNanosuspensions: a promising drug delivery strategyJ Pharm Pharmacol200456782784015233860
   PubMed Web of Science ®Google Scholar
• NoyesAAWhitneyWRThe rate of solution of solid substances in their own solutionsJ Am Chem Soc18971912930934
   Google Scholar
• ScholzAAbrahamssonBDieboldSMInfluence of hydrodynamics and particle size on the absorption of felodipine in labradorsPharm Res2002191424611837699
   PubMed Web of Science ®Google Scholar
• HintzRJJohnsonKCThe effect of particle size distribution on dissolution rate and oral absorptionInt J Pharm1989511917
   Web of Science ®Google Scholar
• XiaDCuiFPiaoHEffect of crystal size on the in vitro dissolution and oral absorption of nitrendipine in ratsPharm Res20102791965197620585842
   PubMed Web of Science ®Google Scholar
• SunWMaoSShiYLiLCFangLNanonization of itraconazole by high pressure homogenization: Stabilizer optimization and effect of particle size on oral absorptionJ Pharm Sci201110083365337321520089
   PubMed Web of Science ®Google Scholar
• WenHJiangHLuZCarvedilol ameliorates sympathetic nerve sprouting and electrical remodeling after myocardial infarction in ratsBiomed Pharmacother201064744645020359859
   PubMed Web of Science ®Google Scholar
• MorganTClinical pharmacokinetics and pharmacodynamics of carvedilolClin Pharmacokinet19942653353467914479
   PubMed Web of Science ®Google Scholar
• HokamaNHobaraNKameyaHOhshiroSSakanashiMRapid and simple micro-determination of carvedilol in rat plasma by high-performance liquid chromatographyJ Chromatogr B Biomed Sci Appl1999732123323810517241
   PubMedGoogle Scholar
• LiuDXuHTianBFabrication of carvedilol nanosuspensions through the anti-solvent precipitation-ultrasonication method for the improvement of dissolution rate and oral bioavailabilityAAPS Pharm Sci Tech2012131295304
   PubMed Web of Science ®Google Scholar
• MosharrafMNyströmCThe effect of particle size and shape on the surface specific dissolution rate of microsized practically insoluble drugsInt J Pharm199512213547
   Google Scholar
• JunghannsJ-UAMüllerRHNanocrystal technology, drug delivery and clinical applicationsInt J Nanomed200833295
   PubMed Web of Science ®Google Scholar
• MüllerRJacobsCKayserONanosuspensions as particulate drug formulations in therapy: rationale for development and what we can expect for the futureAdv Drug Deliv Rev200147131911251242
   PubMed Web of Science ®Google Scholar
• PorterCJTrevaskisNLCharmanWNLipids and lipid-based formulations: optimizing the oral delivery of lipophilic drugsNat Rev Drug Discov20076323124817330072
   PubMed Web of Science ®Google Scholar
• AnderbergEKArturssonPEpithelial transport of drugs in cell culture. VIII: effects of sodium dodecyl sulfate on cell membrane and tight junction permeability in human intestinal epithelial (Caco-2) cellsJ Pharm Sci19938243923988468683
   PubMed Web of Science ®Google Scholar
• LiuDYuSZhuZControlled delivery of carvedilol nanosuspension from osmotic pump capsule: in vitro and in vivo evaluationInt J Pharm20144751–249650325219321
   PubMed Web of Science ®Google Scholar