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Review

Prasugrel for the treatment of patients with acute coronary syndrome

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Pages 321-324 | Published online: 06 Apr 2009

References

  • RuggeriZMPlatelets in atherothrombosisNat Med200281227123412411949
  • GurbelPABlidenKPGuyerKPlatelet reactivity in patients and recurring events post-stenting. Results of the PREPARE POST-STENTING studyJ Am Coll Cardiol2005461820182616286165
  • SteinhublPBBergerJTMannIIIEarly and sustained dual oral antiplatelet therapy following percutaneous coronary intervention: A randomized controlled trialJAMA20022882411242012435254
  • MehtaSRYusufSPetersRJEffects of pretreatment with clopidogrel and aspirin followed by long-term therapy in patients undergoing percutaneous coronary intervention: The PCI-CURE studyLancet200135852753311520521
  • BilletNHAntiplatelet agents and arterial thrombosisCardiol Clin20082618920118406994
  • HochholzerWTrenkDBestehornHPImpact of the degree of peri-interventional platelet inhibition after loading with clopidogrel on early clinical outcome of elective coronary stent placementJ Am Coll Cardiol2006481742175017084243
  • BuonamiciPMarcucciRMiglioriniAImpact of platelet reactivity after clopidogrel administration on drug-eluting stent thrombosisJ Am Coll Cardiol2007492312231717572245
  • NiitsuYJakubowskiJASugidachiAAsaiFPharmacology of CS-747 (prasugrel, LY640315), a novel, potent antiplatelet agent with in vivo P2Y12 receptor antagonist activitySemin Thromb Hemost20053118419415852222
  • SugidachiAAsaiFOgawaTInoueTKoikeHThe in vivo pharmacological profile of CS-747, a novel antiplatelet agent with platelet ADP receptor antagonist propertiesBr J Pharmacol20001291439144610742300
  • FaridNASmithRLGillespieTAThe disposition of prasugrel, a novel thienopyridine, in humansDrug Metab Dispos2007351096110417403916
  • RehmelJLEcksteinJAFaridNAInteractions of two major metabolites of prasugrel, a thienopyridine antiplatelet agent with the cytochromes P450Drug Metab Dispos20063460060716415119
  • BrandtJTCloseSLIturriaSJCommon polymorphisms of CYP2C19 and CYP2C9 affect the pharmacokinetic and pharmacodynamic response to clopidogrel but not prasugrelJ Thromb Haemost200752429243617900275
  • FaridNAPayneCDSmallDSCytochrome P450 3A inhibition by ketoconazole affects prsaugrel and clopidogrel pharmacokinetics and pharmacodynamics differentlyClin Pharmacol Ther20078173574117361128
  • AsaiFJakubowskiJANaganumaHPlatelet inhibitory activity and pharmacokinetics of prasugrel (CS-747) a novel thienopyridine P2Y12 inhibitor: A single-ascending dose study in healthy humansPlatelets20061720921716769598
  • JakubowskiJAMatsushimaNAsaiFA multiple dose study of prasugrel (CS-747), a novel thienopyridine P2Y12 inhibitor, compared with clopidogrel in healthy humansBr J Clin Pharm200663421430
  • MatsushimaNJakubowskiJAAsaiFPlatelet inhibitory activity and pharmacokinetics of prasugrel (CS-747) a novel thienopyridine P2Y12 inhibitor: A multiple-dose study in healthy humansPlatelets20061721822616769599
  • BrandtJTPayneCDWiviottSDA comparison of prasugrel and clopidogrel loading doses on platelet function: Magnitude of platelet inhibition is related to active metabolite formationAm Heart J200715366.e9e1617174640
  • JakubowskiJAPayneCDWeerakkodyGJDose-dependent inhibition of human platelet aggregation by prasugrel and its interaction with aspirin in healthy subjectsJ Cardiovasc Pharmocol200749167173
  • JernbergTPayneCDWintersKJPrasugrel achieves greater inhibition of platelet aggregation and a lower rate of non-responders compared with clopidogrel in aspirin-treated patients with stable coronary artery diseaseEur Heart J2006271166117316621870
  • WiviottSDAntmanEMWintersKJRandomized comparison of prasugrel (CS-747,LY640315), a novel thienopyridine P2Y12 antagonist, with clopidogrel in percutaneous coronary intervention: Results of the Joint Utilizationì of Medications to Block Platelets Optimally (JUMBO)-TIMI 26 trialCirculation20051113366337315967851
  • WiviottSDBraunwaldEMcCabeCHA clinical trial of prasugrel vs. clopidogrel in patients with acute coronary syndromesN Engl J Med20073572001201517982182
  • WiviottSDTrenkDFrelingerALPRINCIPLE-TIMI 44 InvestigatorsPrasugrel compared with high loading- and maintenance-dose clopidogrel in patients with planned percutaneous coronary intervention: the Prasugrel in Comparison to Clopidogrel for Inhibition of Platelet Activation and Aggregation-Thrombolysis in Myocardial Infarction 44 trialCirculation20071162923293218056526