References
- Affolter H., Hertel C., Jaeggi K., Portenier M., Staehelin M. (‐)‐S‐‘3H’CGP‐12177 and its use to determine the rate constants of unlabeled β‐adrenergic antagonists. Proceedings of the National Academy of Sciences 1985; 82: 925–929
- Bai S. A., Wilson M. J., Walle U. K., Walle T. Stereoselective increase in propranolol bioavailability during chronic dosing in the dog. Journal of Pharmacology and Experimental Therapeutics 1983; 227: 360–364
- Bailey J. M. G., Heppleston C., Richmond S. J. Comparison of the in vitro activities of ofloxacin and tetracycline against Chiamydia trachomatis as assessed by indirect immunofluorescence. Antimicrobial Agents and Chemotherapy 1984; 26: 13–16
- Borner K., Lode H. Biotransformation von ausgewählten Gyrasehemmern. Infection 1984; 14(Suppl. 1)54–59
- Brown N. A., Jahnchen E., Mulles W. E., Wollert U. Optical studies on the mechanism of the interaction on the enantiomers of the anticoagulant drugs phenprocoumon and warfarin with human serum albumin. Molecular Pharmacology 1977; 13: 70–79
- Buckpitt A. R., Castagnoli N., Jr., Nelson S. D., Jones A. D., Bahnson L. S. Stereoselectivity of naphthalene epoxidation by mouse, rat, and hamster pulmonary, hepatic, and renal microsomal enzymes. Drug Metabolism and Disposition 1987; 15: 491–498
- Fujii T., Furukawa H., Yoshida K., Miyazaki H., Hashimoto M. Disposition and metabolism of ‘14C’AT‐2266, I. Single administration. Chemotherapy, Tokyo 1984; 32(Suppl. 3)117–135
- Hayakawa I., Atarashi S., Yokohama S., Imamura M., Sakano K., Furukawa M. Synthesis and antibacterial activities of optically active ofloxacin. Antimicrobial Agents and Chemotherapy 1986; 29: 163–164
- Küpfer A., Desmond P. V., Schenker S., Branch R. A. Stereoselective metabolism and disposition of the enantiomers of mephenytoin during chronic oral administration of the racemic drug in man. Journal of Pharmacology and Experimental Therapeutics 1982; 221: 590–597
- Lefkowitz R. J., Williams L. T. Catecholamine binding to the β‐adrenergic receptor. Proceedings of the National Academy of Sciences 1977; 74: 515–519
- Lennard M. S., Tucker G. T., Silas J. H., Freestone S., Lamsey L. E., Woods H. F. Differential stereoselective metabolism of metoprolol in extensive and poor debrisoquine metabolizers. Clinical Pharmacology and Therapeutics 1983; 34: 732–737
- Mayer J. M., Bartolucci C., Maitre J. M., Testa B. Metabolic chiral inversion of antiinflammatory 2‐arylpropionates: lack of reaction in liver homogenates, and study of methine proton acidity. Xenobiotica 1988; 18(5)533–543
- Okazaki O., Kurata T., Hashimoto K., Sudo K., Tsumura M., Tachizawa H. Metabolic disposition of DL‐8280. The second report: absorption, distribution and excretion of 14C‐DL‐8280 in various animal species. Chemotherapy, Tokyo 1984; 32(Suppl. 1)1185–1202
- Osada Y., Ogawa H. Antimycoplasmal activity of ofloxacin (DL‐8280). Antimicrobial Agents and Chemotherapy 1983; 23: 509–511
- Sato K., Matsuura Y., Inoue M., Une T., Osada Y., Ogawa H., Mitsuhashi M. In vitro and in vivo activity of DL‐8280, a new oxazine derivative. Antimicrobial Agents and Chemotherapy 1982; 22: 548–553
- Silber B., Holford N. H. G., Riegelman S. Stereoselective disposition and glucuroni‐dation of propranolol in human. Journal of Pharmaceutical Sciences 1982; 71: 699–703
- Sudo K., Okazaki O., Tsumura M., Tachizawa H. Isolation and identification of metabolites of ofloxacin in rats, dogs and monkeys. Xenobiotica 1986; 16: 725–732
- Sudo K., Hashimoto K., Kurata T., Okazaki O., Tsumura M., Tachizawa H. Metabolic disposition of DL‐8280. The third report: metabolism of 14C‐DL‐8280 in various animal species. Chemotherapy, Tokyo 1984; 32(Suppl. 1)1203–1210
- Sugeno K., Okabe H., Norikura R., Koike M., Kawamoto K. Absorption, distribution, metabolism and excretion of cinoxacin. The second report: comparative metabolism and disposition of cinoxacin in dog, rhesus monkey, rabbit and guinea pig. Chemotherapy, Tokyo 1980; 28(Suppl. 4)90–103
- Vermeulen N. P. E. Stereoselectivity in the enzymatic biotransformation of drugs and other xenobiotics. Drug Metabolism‐From Microbes to Man, D. Benford, J. W. Bridges, G. G. Gibson. Taylor & Francis, London 1987; 615–640
- Wade D. N., Mearrick P. T., Morris J. L. Active transport of L‐dopa in the intestine. Nature 1973; 242: 463–465
- Walle T. Stereochemistry of the in vivo disposition and metabolism of propranolol in dog and man using deuterium‐labeled pseudoracemates. Drug Metabolism and Disposition 1985; 13: 279–282
- Walle U. K., Walle T., Bai S. A. Stereoselective binding of propranolol to human plasma, alpha1‐acid glycoprotein, and albumin. Clinical Pharmacology and Therapeutics 1983; 34: 718–723
- Weiland G. A., Oswald R. E. The mechanism of binding of dihydropyridine calcium channel blockers to rat brain membranes. Journal of Biological Chemistry 1985; 260: 8456–8464
- Yamaoka K., Tanigawara Y., Nakagawa T., Uno T. A pharmacokinetic analysis program (MULTI) for microcomputer. Journal of Pharmacology and Dynamics 1981; 4: 879–885