The use of single-sample clearance estimates to probe hepatic drug metabolism in rats. IV. A model for possible application to phenotyping xenobiotic influences on human drug metabolism

References

• Bachmann K., Yang C., Jahn D., Schwartz J. The use of single sample clearance estimates to probe hepatic drug metabolism in rats. I. Xenobiotica 1988a; 18: 149–157
   Google Scholar
• Bachmann K., Jahn D., Yang C., Schwartz J. The use of single sample clearance estimates to probe hepatic drug metabolism in rats. II. Xenobiotica 1988b; 18: 161–167
   PubMed Web of Science ®Google Scholar
• Bachmann K., Jahn D., Yang C., Schwartz J. Ethosuximide disposition kinetics in rats. Xenobiotica 1988c; 18: 373–380
   PubMed Web of Science ®Google Scholar
• Baille T., Rettenmeir A. W. Valproate: biotransformation. Antiepileptic Drugs, R. H. Levy, F. Dreifuss, R. Mattson, B. Meldrum, J. K. Penry. Raven Press, New York 1989
   Google Scholar
• Boobis A., Davies D. Human cytochromes P-450. Xenobiotica 1984; 14: 151–185
   PubMed Web of Science ®Google Scholar
• Burke M., Wolf R. Substrates and inhibitors as probes of individual forms of drug metabolizing systems. Drug Metabolism—from Molecules to Man, D. Benford, J. Bridges, G. Gibson. Taylor & Francis, London 1987; 219–243
   Google Scholar
• Conney A. Pharmacological implications of microsomal enzyme induction. Pharmacological Reviews 1967; 36: 317–366
   Google Scholar
• Conney A. Induction of microsomal cytochrome P-450 enzymes: The first Bernard B. Brodie lecture at Pennsylvania State University. Life Sciences 1986; 39: 2493–2518
   PubMed Web of Science ®Google Scholar
• Dandliker W., Kelly R. Fluorescence polarization immunoassay: theory and experimental method. Immunochemistry 1973; 10: 219–227
   PubMedGoogle Scholar
• Dickinson R., Harland R., Ilias A., Rodgers R., Kaufman S., Lynn R., Gerber N. Disposition of valproic acid in the rat: dose-dependent metabolism, distribution, enterohepatic recirculation and choleretic effect. Journal of Pharmacology and Experimental Therapeutics 1979; 211: 583–595
   PubMed Web of Science ®Google Scholar
• Døssing M., Poulsen H., Andreasen P. B., Tygstrup N. A simple method for determination of antipyrine clearance. Clinical Pharmacology and Therapeutics 1982; 32: 392–396
   PubMed Web of Science ®Google Scholar
• Eichelbaum M., Tomson T., Tybring G., Bertilsson L. Carbamazepine metabolism in man: induction and pharmacogenetic aspects. Clinical Pharmacokinetics 1985; 10: 80–90
   PubMed Web of Science ®Google Scholar
• Fournel S., Magdalou J., Pinon P., Siest G. Differential induction profile of drug-metabolizing enzymes after treatment with hypolipidemic agents. Xenobiotica 1987; 17: 445–457
   PubMed Web of Science ®Google Scholar
• Gelboin H. Benzo (a) pyrene metabolism, activation, and carcinogenesis: Role and regulation of the mixed-function oxidases and related enzymes. Physiological Reviews 1980; 60: 1107–1166
   PubMed Web of Science ®Google Scholar
• Gibson G., Orton T., Tamurini P. Cytochrome P-450 induction by clofibrate. Biochemical Journal 1982; 303: 161–168
   Google Scholar
• Halpert J. Multiplicity of steroid-inducible cytochromes P-450 in rat liver microsomes. Archives of Biochemistry and Biophysics 1988; 263: 59–68
   PubMed Web of Science ®Google Scholar
• Hardy B., Schentag J. Lack of effect of cimetidine on the metabolism of quinidine: effect on renal clearance. International Journal of Clinical Pharmacology Therapy and Toxicology 1988; 26: 388–391
   PubMed Web of Science ®Google Scholar
• Heinemeyer G., Nau H., Hildebrandt A., Roots I. Oxidation and glucuronidation of valproic acid in male rats—influence of phenobarbital, 3-methylcholanthrene, β-naphthoflavone and clofibrate. Biochemical Pharmacology 1985; 34: 133–139
   PubMed Web of Science ®Google Scholar
• Hjelle J., Klaassen C. Glucuronidation and biliary excretion of acetaminophen in rats. Journal of Pharmacology and Experimental Therapeutics 1984; 228: 407–413
   PubMed Web of Science ®Google Scholar
• Ioannides C., Parke D. V. The cytochromes P-448-A unique family of enzymes involved in chemical toxicity and carcinogenesis. Biochemical Pharmacology 1987; 36: 4197–4207
   PubMed Web of Science ®Google Scholar
• Jolley M. Fluorescence polarization immunoassay for the determination of therapeutic drug levels in human plasma. Journal of Analytical Toxicology 1981; 5: 236–240
   PubMed Web of Science ®Google Scholar
• Jusko W. Guidelines for collection and analysis of pharmacokinetic data. Applied Pharmacokinetics, W. Evans, J. Schentag, W. Jusko. Applied Therapeutics, Spokane 1986; 9–54
   Google Scholar
• Muller-Enoch D., Guengerich F. P. Oxidation of quinidine by human liver cytochrome P-450. Drug Metabolism—from Molecules to Man, D. Benford, J. Bridges, G. Gibson. Taylor & Francis, London 1987; 115–120
   Google Scholar
• Nebert W., Gonzalez F. P450 genes: structure, evolution, and regulation. Annual Reviews of Biochemistry 1987; 56: 945–993
   PubMed Web of Science ®Google Scholar
• Onhaus E., Brockmeyer N., Dylewicz P., Habicht H. The effect of antipyrine and rifampin on the metabolism of diazepam. Clinical Pharmacology and Therapeutics 1987; 42: 148–156
   PubMed Web of Science ®Google Scholar
• Pilsgaard H., Poulsen H. A one-sample method for antipyrine clearance determination in rats. Pharmacology 1984; 29: 110–116
   PubMed Web of Science ®Google Scholar
• Sharma R., Lake B., Foster J., Gibson G. Microsomal cytochrome P-452 induction and peroxisome proliferation by hypolipidaemic agents in rat liver: a mechanistic inter-relationship. Biochemical Pharmacology 1988; 37: 1193–1201
   PubMed Web of Science ®Google Scholar
• Sheiner L., Beal S. Some suggestions for measuring predictive performance. Journal of Pharmacokinetics and Biopharmaceutics 1981; 9: 503–512
   PubMedGoogle Scholar
• Shumaker R. PKCALC: A BASIC interactive computer program for statistical and pharmacokinetic analysis of data. Drug Metabolism Review 1986; 17: 331–348
   PubMed Web of Science ®Google Scholar
• Steele R., Torrie J. Principles and Procedures of Statistics. McGraw-Hill, New York 1960; 404–406
   Google Scholar