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Xenobiotica
the fate of foreign compounds in biological systems
Volume 20, 1990 - Issue 6
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Original Article

The alpha carbon oxidation of some phencyclidine analogues by rat tissue and its pharmacological implications

M. Stefek Department of Pharmacology and the Jonsson Comprehensive Cancer Center, UCLA School of Medicine, Center for the Health Sciences, Los Angeles, California, 90024-1735, USA
,
R. W. Ransom Merck, Sharp and Dohme Research Laboratories, W26A-3025 West PointPA, 19486, USA
,
E. W. Distefano Department of Pharmacology and the Jonsson Comprehensive Cancer Center, UCLA School of Medicine, Center for the Health Sciences, Los Angeles, California, 90024-1735, USA
&
A. K. Cho Department of Pharmacology and the Jonsson Comprehensive Cancer Center, UCLA School of Medicine, Center for the Health Sciences, Los Angeles, California, 90024-1735, USA
Pages 591-600 | Received 04 Aug 1989, Accepted 10 Feb 1990, Published online: 27 Aug 2009

References

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  • Weber E., Sonders M., Quarum M., McLean S., Pou S., Keana J. F. W. 1,3-Di(2-[5,-3H]-toly)guanidine: a selective ligand that labels sigma-type receptors for psychotomimetic opiates and antipsychotic drugs. Proceedings of the National Academy of Sciences, USA 1986; 83: 8784–8788
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