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Xenobiotica
the fate of foreign compounds in biological systems
Volume 26, 1996 - Issue 2
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Research Article

Enantioselective binding of Casodex to the androgen receptor

A. Mukherjee Department of Pharmaceutical Sciences, College of Pharmacy, 874 Union Avenue, University of Tennessee, Memphis, TN, 32, USA
,
L. Kirkovsky Department of Pharmaceutical Sciences, College of Pharmacy, 874 Union Avenue, University of Tennessee, Memphis, TN, 32, USA
,
X. T. Yao Department of Pharmaceutical Sciences, College of Pharmacy, 874 Union Avenue, University of Tennessee, Memphis, TN, 32, USA
,
R. C. Yates Department of Pharmaceutical Sciences, College of Pharmacy, 874 Union Avenue, University of Tennessee, Memphis, TN, 32, USA
,
D. D. Miller Department of Pharmaceutical Sciences, College of Pharmacy, 874 Union Avenue, University of Tennessee, Memphis, TN, 32, USA
&
J. T. Dalton Department of Pharmaceutical Sciences, College of Pharmacy, 874 Union Avenue, University of Tennessee, Memphis, TN, 32, USA
Pages 117-122 | Received 13 Jul 1995, Published online: 22 Sep 2008

References

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  • Veldscholte J., Berrevoets C. A., Ris-Stalpers C., Kuiper G. G. J. M., Jenster G., Trapman J., Brinkmann A. O., Mulder E. The androgen receptor in LNCaP cells contains a mutation in the ligand binding domain which affects steroid binding characteristics and response to antiandrogens. Journal of Steroid Biochemistry and Molecular Biology 1992; 41: 665–669

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