Formulation of wax oxybenzone microparticles using a factorial approach

References

• Albertini B, Mezzena M, Passerini N, Rodriguez L, Scalia S. Evaluation of spray congealing as technique for the preparation of highly loaded solid lipid microparticles containing the sunscreen agent, avobenzone. J Pharm Sci 2009; 98: 2759–69
   PubMed Web of Science ®Google Scholar
• Bhavsar MD, Tiwari SB, Amiji MM. Formulation optimization for the nanoparticles-in-microsphere hybrid oral delivery system using factorial design. J Control Release 2006; 110: 422–30
   PubMed Web of Science ®Google Scholar
• Denet AR, Vanbever R, Préat V. Skin electroporation for transdermal and topical delivery. Adv Drug Deliv Rev 2004; 56: 659–74
   PubMed Web of Science ®Google Scholar
• Dorgan PD. Waxes in cosmetics. Drug Cosmet Ind 2002; 133: 30–3
   Google Scholar
• Felton LA, Wiley CJ, Godwin DA. Influence of hydroxypropyl-beta-cyclodextrin on the transdermal permeation and skin accumulation of oxybenzone. Drug Dev Ind Pharm 2002; 28: 1117–24
   PubMed Web of Science ®Google Scholar
• Felton LA, Wiley CJ, Godwin DA. Influence of cyclodextrin complexation on the in vivo photoprotection effects of oxybenzone. Drug Dev Ind Pharm 2004; 30: 95–102
   PubMed Web of Science ®Google Scholar
• Furniss BS, Hannaford AJ, Smith PWG, Tatchell AR. Specroscopic methods and the interpretation of spectra. Vogel's textbook of practical organic chemistry. Longman Group UK LTD, England 1989; 254–316
   Google Scholar
• Gogna D, Jain SK, Yadav AK, Agrawal GP. Microsphere based improved sunscreenformulation of ethylhexyl methoxycinnamate. Curr Drug Deliv 2007; 14: 153–9
   Google Scholar
• Gomaa YA, El-Khordagui LK, Boraei NA, Darwish IA. Chitosan microparticles incorporating a hydrophilic sunscreen agent. Carbohydr Polym 2010; 81: 234–42
   Web of Science ®Google Scholar
• González H, Farbrot A, Larkö O, Wennberg AM. Percutaneous absorption of the sunscreen benzophenone-3 after repeated whole-body applications, with and without ultraviolet irradiation. Br J Dermatol 2006; 154: 337–40
   PubMed Web of Science ®Google Scholar
• González S, Fernández-Lorente M, Gilaberte-Calzada Y. The latest on skin photoprotection. Clin Dermatol 2008; 26: 614–26
   PubMed Web of Science ®Google Scholar
• Gulbake A, Jain A, Khare P, Sanjay KJ. Solid lipid nanoparticles bearing oxybenzone: In vitro and in vivo evaluation. J Microencapsul 2010; 27: 226–33
   PubMed Web of Science ®Google Scholar
• Guyot M, Fawaz F. Nifedipine loaded-polymeric microspheres: Preparation and physical characteristics. Int J Pharm 1998; 17: 61–74
   Google Scholar
• Iannuccelli V, Sala N, Tursilli R, Coppi G, Scalia S. Influence of lipospheres preparation on butyl-methoxydibenzoylmethane photostability. Eur J Pharm Biopharm 2006; 63: 140–45
   PubMed Web of Science ®Google Scholar
• Jain SK, Jain NK. Multiparticulate carriers for sun-screening agents. Int J Cosmet Sci 2010; 32: 89–98
   PubMedGoogle Scholar
• Janjua NR, Mogensen B, Andersson AM, Petersen JH, Henriksen M, Skakkebaek NE, Wulf HC. Systemic absorption of the sunscreens benzophenone-3, octylmethoxycinnamate, and 3-(4-methyl-benzylidene) camphor after whole-body topical application and reproductive hormone levels in humans. J Invest Dermatol 2004; 123: 57–61
   PubMed Web of Science ®Google Scholar
• Jaspart S, Bertholet P, Piel G, Dogne JM, Delattre L, Evrard B. Solid lipid microparticles as a sustained release system for pulmonary drug delivery. Eur J Pharm Biopharm 2007; 65: 47–56
   PubMed Web of Science ®Google Scholar
• Jaspart S, Piel G, Delattre L, Evrard B. Solid lipid microparticles: formulation, preparation, characterization, drug release and applications. Expert Opin Drug Deliv 2005; 2: 75–87
   PubMedGoogle Scholar
• Jenning V, Gohla S. Comparison of wax and glyceride solid lipid nanoparticles (SLN®). Int J Pharm 2000; 196: 219–22
   PubMed Web of Science ®Google Scholar
• Labouta HI, El-Khordagui LK, Molokhia AM, Ghaly GM. Multivariate modeling of encapsulation and release of an ionisable drug from polymer microspheres. J Pharm Sci 2009; 89: 4603–15
   Google Scholar
• Lamprecht A, Yamamoto H, Takeuchi H, Kawashima Y. Microsphere design for the colonic delivery of 5-fluorouracil. J Control Release 2003; 90: 313–22
   PubMed Web of Science ®Google Scholar
• Larsson K. Classification of glycerides crystal forms. Acta Chem Scand 1996; 20: 2255–60
   Google Scholar
• Mao S, Shi Y, Li L, Xu J, Schaper A, Kissel T. Effects of process and formulation parameters on characteristics and internal morphology of poly (D,L-lactide-co-glycolide) microspheres formed by the solvent evaporation method. Eur J Pharm Biopharm 2008; 68: 214–23
   PubMed Web of Science ®Google Scholar
• Martinez-Sancho C, Herrero-Vanrell R, Negro S. Optimization of aciclovir poly (D,L-lactide-co-glycolide) microspheres for intravitreal administration using a factorial design study. Int J Pharm 2004; 273: 45–56
   PubMed Web of Science ®Google Scholar
• Montgomery DC. Experiments with a single factor: The analysis of variance. Design and analysis of experiments. John Wiley & Sons, New York 1997; 63–117
   Google Scholar
• Ohba N. Hydrophile-lipophile balance values for O/W emulsions stabilized by nonionic surfactants. II. Required HLB hydrophile-lipophile balance values of the oil mixture. Bull Chem Soc Jpn 1962; 35: 1021–5
   Google Scholar
• Pardeike J, Hommoss A, Müller RH. Lipid nanoparticles (SLN, NLC) in cosmetic and pharmaceutical dermal products. Int J Pharm 2009; 366: 170–84
   PubMed Web of Science ®Google Scholar
• Pasquali RC, Taurozzi MP, Bregni C. Some considerations about the hydrophilic-lipophilic balance system. Int J Pharm 2008; 356: 44–51
   PubMed Web of Science ®Google Scholar
• Passerini N, Perissuti B, Moneghini M, Voinovich D, Albertini B, Cavallari C, Rodriguez L. Characterization of carbamazepine-Gelucire 50/13 microparticles prepared by a spray congealing process using ultrasounds. J Pharm Sci 2002; 91: 699–707
   PubMed Web of Science ®Google Scholar
• Patel M, Jain SK, Yadav AK, Gogna D, Agrawal GP. Preparation and characterization of oxybenzone-loaded gelatin microspheres for enhancement of sunscreening efficacy. Drug Deliv 2006; 13: 323–30
   PubMed Web of Science ®Google Scholar
• Roberts M, Cespi M, Ford JL, Dyas AM, Downing J, Martini LG, Crowley PJ. Influence of ethanol on aspirin release from hypremellose matrices. Int J Pharm 2007; 332: 31–7
   PubMed Web of Science ®Google Scholar
• Roth W, Setnik B, Zietsch M, Burst A, Breitenbach J, Sellers E, Bernnan D. Ethanol effects on drug release from verapamil meltrex, an innovative melt extruded formulation. Int J Pharm 2009; 368: 72–5
   PubMed Web of Science ®Google Scholar
• Schauder S, Ippen H. Contact and photocontact sensitivity to sunscreens. Review of a 15-year experience and of the literature. Contact Derm 1997; 37: 221–32
   PubMed Web of Science ®Google Scholar
• Schmid-Wendtner MH, Korting HC. The pH of the skin surface and its impact on the barrier function. Skin Pharmacol Physiol 2006; 19: 296–302
   PubMed Web of Science ®Google Scholar
• Schwartz JB, Simonelli AP, Higuchi WI. Drug release from wax matrices. II. Application of a mixture theory to the sulfanilamide-wax system. J Pharm Sci 1968; 57: 280–2
   Google Scholar
• Shah V, Elkins J, Skelly J. Relationship between in vivo skin blanching and in vitro release rate foe betametahsone valerate creams. J Pharm Sci 2006; 81: 104–6
   Google Scholar
• Torrado S, Torrado J, Cadórniga R. Topical application of albumin microspheres containing vitamin A: Drug release and availability. Int J Pharm 1992; 86: 147–52
   Web of Science ®Google Scholar
• Tursilli R, Piel G, Delattre L, Scalia S. Solid lipid microparticles containing the sunscreen agent, octyl-dimethylaminobenzoate: Effect of the vehicle. Eur J Pharm Biopharm 2007; 66: 483–7
   PubMed Web of Science ®Google Scholar
• Varshosaz J, Keihanfar M. Development and evaluation of sustained-release propranolol wax microspheres. J Microencapsul 2001; 18: 277–84
   PubMed Web of Science ®Google Scholar
• Villalobos-Hernández JR, Müller-Goymann CC. Novel nanoparticulate carrier system based on carnauba wax and decyl oleate for the dispersion of inorganic sunscreens in aqueous media. Eur J Pharm Biopharm 2005; 60: 113–22
   PubMed Web of Science ®Google Scholar
• Villalobos-Hernández JR, Müller-Goymann CC. Physical stability, centrifugation tests, and entrapment efficiency studies of carnauba wax-decyl oleate nanoparticles used for the dispersion of inorganic sunscreens in aqueous media. Eur J Pharm Biopharm 2006; 63: 115–27
   PubMed Web of Science ®Google Scholar
• Villalobos-Hernández JR, Müller-Goymann CC. In vitro erythemal UV-A protection factors of inorganic sunscreens distributed in aqueous media using carnauba wax-decyl oleate nanoparticles. Eur J Pharm Biopharm 2007; 65: 122–5
   PubMed Web of Science ®Google Scholar
• Wang L, Ando S, Ishida Y, Ohtani H, Tsuge S, Nakayama T. Quantitative and discriminative analysis of carnauba waxes by reactive pyrolysis-GC in the presence of organic alkali using vertical microfurnance pyrolyzer. J Anal Appl Pyrolysis 2001; 58–59: 525–37
   Web of Science ®Google Scholar
• Wissing SA, Müller RH. The development of an improved carrier system for sunscreen formulations based on crystalline lipid nanoparticles. Int J Pharm 2002; 242: 373–5
   PubMed Web of Science ®Google Scholar
• Xia Q, Saupe A, Müller RH, Souto EB. Nanostructured lipid carriers as novel carrier for sunscreen formulations. Int J Cosmet Sci 2008; 29: 473–82
   Google Scholar
• Yener G, Incegul T, Yener N. Importance of using solid lipid microspheres as carriers for UV filters on the example octyl methoxycinnamate. Int J Pharm 2003; 258: 203–7
   PubMed Web of Science ®Google Scholar