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Research Article

Ciprofloxacin hydrochloride-loaded glyceryl monostearate nanoparticle: factorial design of Lutrol F68 and Phospholipon 90G

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Pages 331-343 | Received 23 Jul 2011, Accepted 12 Dec 2011, Published online: 18 Jan 2012

References

  • Ahlin P, Kristl J, Smid-Korbar J. Optimization of procedure parameters and physical stability of solid lipid nanoparticles in dispersions. Acta Pharm 1998; 48: 259–67
  • Ahmad H, Yaseen M. Application of a chemical group contribution technique for calculating solubility parameters of polymers. Polymer Eng Sci 1979; 19: 858–63
  • Banker GS, Rhodes CT. Modern pharmaceutics. Informa HealthCare, New York 2002
  • Barton AFM. CRC handbook of solubility parameters and other cohesion parameters. CRC, Florida 1991
  • Barton AFM. Applications of solubility parameters and other cohesion parameters in polymer science and technology. Pure Appl Chem 1985; 57: 905–12
  • Bordes C, Fréville V, Ruffin E, Marote P, Gauvrit JY, Briançon S, Lantéri P. Determination of poly(-caprolactone) solubility parameters: Application to solvent substitution in a microencapsulation process. Int J Pharm, 2010;383:236–43.
  • Cavalli R, Caputo O, Marengo E, Pattarino F, Gasco MR. The effects of components of microemulsions on both size and crystalline structure of solid lipid nanoparticles (SLN) containing a series of model molecules. Pharmazie 1998; 53: 392–96
  • Charoo NA, Kohli K, Ali A, Anwer A. Ophthalmic delivery of ciprofloxacin hydrochloride from different polymer formulations: in vitro and in vivo studies. Drug Dev Ind Pharm 2003; 29(2)215–21
  • Chatzaeiaoannou TP. Quantitative calculations in pharmaceutical practice and research. VCH Publishers, New York 1993
  • Clausse M. Dielectric Properties of emulsions and related systems. Encyclopedia of emulsion technology, P Becher. Marcel Dekker Inc., New York 1983; 1: 481–715
  • Costa P, Sousa Lobo JM. Modeling and comparison of dissolution profiles. Eur J Pharm Biopharm 2001; 13: 123–33
  • Dillena K, Vandervoorta J, Mooterb G, Verheydenb L, Ludwig A. Factorial design, physicochemical characterisation and activity of ciprofloxacin-PLGA nanoparticles. Int J Pharm 2004; 275: 171–87
  • Egger SF, Ruckhofer J, Alzner E, Hell M, Hitz W, Grabner G. In vitro susceptibilities to topical antibiotics of bacteria isolated from the surface of clinically symptomatic eyes. Ophthalmic Res 2001; 33: 117–20
  • Ghebremeskel AN, Vemavarapu C, Lodaya M. Use of surfactants as plasticizers in preparing solid dispersions of poorly soluble API: Selection of polymer-surfactant combinations using solubility parameters and testing the processability. Int J Pharm 2007; 328: 119–29
  • Gohel MC, Panchal MK, Jogani VV. Novel mathematical method for quantitative expression of deviation from the Higuchi model. AAPS PharmSciTech 2000; 1: 43–8
  • Hansen CM. Hansen solubility parameters: A user's handbook. CRC, Florida 2007
  • Heurtault B, Saulnier P, Pech B, Proust JE, Benoit JP. Physico-chemical stability of colloidal lipid particles. Biomaterials, 2003;24:4283–300.
  • Higuchi T. Mechanism of sustained action medication. Theoretical analysis of rate of release of solid drugs dispersed in solid matrices. J Pharm Sci 1963; 52: 1145–9
  • Komatsu H, Kitajima A, Okada S. Pharmaceutical characterization of commercially available intravenous fat emulsions: estimation of average particle size, size distribution and surface potential using photon correlation spectroscopy. Chem Pharm Bull 1995; 43: 1412–15
  • Li X, Nies S, Kong J, Li N, Jue C, Pana W. A controlled release ocular delivery system for ibuprofen based on nanostructured lipid carriers. Int J Pharm 2008; 363: 177–82
  • Magdassi S, Siman-Tov A. Formation and stabilization of perfluorocarbon emulsions. Int J Pharm 1990; 59: 69–72
  • Mehnert W, Mäder K. Solid lipid nanoparticles: Production, characterization and applications. Adv Drug Deliv Rev 2001; 47: 165–96
  • Mishra GP, Bagui M, Tamboli V, Mitra AK, Recent applications of liposomes in ophthalmic drug delivery. J Drug Deliv, 2011;2011:1–14
  • Morel S, Ugazio E, Cavalli R, Gasco MR. Thymopentin in solid lipid nanoparticles. Int J Pharm 1996; 132: 259–61
  • Muller RH. Cytotoxicity of magnetite-loaded polylactide, polylactide/glycolide particles and solid lipid nanoparticles. Int J Pharm 1996; 138: 85–94
  • Muller RH. Solid lipid nanoparticles: Phagocytic uptake, in vitro cytotoxicity and in vitro biodegradation. Pharm Ind 1999; 61: 564–9
  • Muller RH, Maaben S, Weyhers H, Mehnert W. Phagocytic uptake and cytotoxicity of solid lipid nanoparticles (SLN) sterically stabilized with poloxamine 908 and poloxamer 407. J Drug Target 1996; 4: 161–70
  • Müller RH, Mäder K, Gohla S. Solid lipid nanoparticles (SLN) for controlled drug delivery – A review of the state of the art. Eur J Pharm Biopharm 2000; 50: 161–77
  • Muller RH, Ruhl D, Runge S, Schulze-Forster K, Mehnert W. Cytotoxicity of solid lipid nanoparticles as a function of the lipid matrix and the surfactant. Pharm Res 1997; 14: 458–62
  • Müller RH, Wallis K, Tröster S, Kreuter J. In vitro characterization of poly (methyl-methaerylate) nanoparticles and correlation to their in vivo fate. J Contr Release 1992; 20: 237–46
  • Olbrich C, Gessner A, Schroder W, Kayser O, Muller RH. Lipid-drug conjugate nanoparticles of the hydrophilic drug diminazene – Cytotoxicity testing and mouse serum adsorption. J Cont Release 2004a; 96: 425–35
  • Olbrich C, Muller RH, Tabatt K, Kayser O, Schulze C, Schade R. Stable biocompatible adjuvants: a new type of adjuvant based on solid lipid nanoparticles: a study on cytotoxicity, compatibility and efficacy in chicken. Altern Lab Anim 2002; 30: 443–58
  • Olbrich C, Scholer N, Tabatt K, Kayser O, Muller RH. Cytotoxicity studies of Dynasan 114 solid lipid nanoparticles (SLN) on RAW 264.7 macrophages – Impact of phagocytosis on viability and cytokine production. J Pharm Pharmacol 2004b; 56: 883–91
  • Pandita D, Ahuja A, Lather V, Dutta T, Velpandian T, Khar R. Development, characterization and in vitro assessement of stearylamine-based lipid nanoparticles of paclitaxel. Pharmazie 2011; 66: 171–7
  • Reithmeier H, Herrmann J, Gopferich A. Lipid microparticles as a parenteral controlled release device for peptides. J Contr Release 2001; 73: 339–50
  • Reza M, Quadir MA, Haider SS. Development of theophylline sustained release dosage form based on kollidon SR. Pak J Pharm Sci 2002; 15: 63–70
  • Roberts R, Rowe R. The solubility parameter and fractional polarity of microcrystalline cellulose as determined by mechanical measurement. Int J Pharm 1993; 99: 157–64
  • Schubert M, Muller-Goymann C. Characterisation of surface-modified solid lipid nanoparticles (SLN): Influence of lecithin and nonionic emulsifier. Eur J Pharm Biopharm 2005; 61: 77–86
  • Schubert MA, Harms M, Muller-Goymann CC. Structural investigations on lipid nanoparticles containing high amounts of lecithin. Eur J Pharm 2006; 27: 226–36
  • Schwarz C. Solid lipid nanoparticles (SLN) for controlled drug delivery II. Drug incorporation and physicochemical characterization. J Microencapsul 1999; 16: 205–13
  • Shi L, Li Z, Yu L, Jia H, Zheng L. Effects of surfactants and lipids on the preparation of solid lipid nanoparticles using double emulsion method. Journal of Disper Sci Tech 2011; 32: 254–9
  • Sinha VR, Srivastava S, Goel H, Jindal V. Solid lipid nanoparticles (SLN's) – Trends and implications in drug targeting. Int J Adv Pharmaceut Sci 2010; 1: 212–38
  • Swardrick J. Encyclopedia of pharmaceutical technology. Informa Healthcare, New York 2007
  • Trotta M, Debernardi F, Caputo O. Preparation of solid lipid nanoparticles by a solvent emulsification–diffusion technique. Int J Pharm 2003; 257: 153–60
  • van Krevelen DW, Hoftyzer P. Properties of polymers. Elsevier Publishing Company, New York 1976
  • Vaughan C. Using solubility parameters in cosmetics formulation. J Soc Cosmet Chem 1985; 36: 319–33
  • Verheyen S, Augustijns P, Kinget R, Van den Mooter G. Determination of partial solubility parameters of five benzodiazepines in individual solvents. Int J Pharm, 2001;228:199–207.
  • Wang Y, Deng Y, Mao S, Jin S, Wang J, Bi D. Characterization and body distribution of -elemene solid lipid nanoparticles (SLN). Drug Dev Ind Pharm 2005; 31: 769–78
  • Westesen K, Siekmann B. Investigation of the gel formation of phospholipid-stabilized solid lipid nanoparticles. Int J Pharm 1997; 151: 35–45
  • Wiacek AE. Electrokinetic properties of n-tetradecane/lecithin solution emulsions. Colloid Surface Physicochem Eng Aspect 2007; 293: 20–7
  • Zimmer A, Kreuter J. Microspheres and nanoparticles used in ocular delivery systems. Adv Drug Deliv Rev 1995; 16: 61–73
  • Yassin AEB, Anwer M, Mowafy HA, El-Bagory I, Bayomi M, Alsarra I. Optimization of 5-fluorouracil solid-lipid nanoparticles: A preliminary study to treat colon cancer. Int J Med Sci, 2010;7(6):398–408.
  • Zimmermann E, Müller RH. Electrolyte-and pH-stabilities of aqueous solid lipid nanoparticle (SLN (TM)) dispersions in artificial gastrointestinal media. Eur J Pharm Biopharm 2001; 52: 203–10

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