A robust experimental design method to optimize formulations of retinol solid lipid nanoparticles

References

• Andersson E, Rosdahl I, Törmä H, Vahlquist A. Ultraviolet irradiation depletes cellular retinol and alters the metabolism of retinoic acid in cultured human keratinocytes and melanocytes. Melanoma Res 1999; 3: 339–46
   Google Scholar
• Bloomfield MS, Butler WC. Robustness testing, using experimental design, of a flow-through dissolution method for a product where the actives have markedly differing solubility properties. Int J Pharm 2000; 206(1–2): 55–61
   Google Scholar
• Bolton S. Pharmaceutical statistics: Practical and clinical applications. Marcel Dekker, 2nd ed., Revised and Expanded. New York 1990
   Google Scholar
• Borror CM, 1998. Response surface methods for experiments involving noise variables. Ph.D. Dissertation, Department of Industrial Engineering, Arizona State University, Tempe, AZ
   Google Scholar
• Choi DH, Shin SM, Truong NKV, Jeong SH, A new experimental design method to optimize formulations focusing on a lubricant for hydrophilic matrix tablets. Drug Dev Ind Pharm, 2012;38 (9):1117–27
   Google Scholar
• Del Castillo E, Montgomery D. A nonlinear programming solution to the dual response problem. J Qual Technol 1993; 25(3)199–204
   Web of Science ®Google Scholar
• Ding R, Lin DKJ, Wei D. Dual-response surface optimization: A weighed MSE approach. Qual Eng 2004; 16(3)377–85
   Google Scholar
• Fisher GJ, Voorhees JJ. Molecular mechanisms of retinoid actions in skin. FASEB J 1996; 10: 1002–13
   PubMed Web of Science ®Google Scholar
• Gonnet M, Lethuaut L, Boury F. New trends in encapsulation of liposoluble vitamins. J Control Release 2010; 146(3)276–90
   PubMed Web of Science ®Google Scholar
• Jenning V, Gysler A, Schafer-Korting M, Gohla SH. Vitamin A loaded solid lipid nanoparticles for topical use: Occlusive properties and drug targeting to the upper skin. Eur J Pharm Biopharm 2000a; 49: 211–18
   PubMed Web of Science ®Google Scholar
• Jenning V, Schafer-Korting M, Gohla S. Vitamin A-loaded solid lipid nanoparticles for topical use: Drug release properties. J Control Rel 2000b; 66: 115–26
   PubMed Web of Science ®Google Scholar
• Jenning V, Thunemann AF, Gohla SH. Characterisation of a novel solid lipid nanoparticle carrier system on binary mixtures of liquid and solid lipids. Int J Pharm 2000c; 199(2)167–77
   PubMed Web of Science ®Google Scholar
• Kincl M, Turk S, Vrecer F. Application of experimental design methodology in development and optimization of drug release method. Int J Pharm 2005; 291: 39–49
   PubMed Web of Science ®Google Scholar
• Kovacevic A, Savic S, Vuleta G, Muller RH, Keck CM. Polyhydroxy surfactants for the formulation of lipid nanoparticles (SLN and NLC): Effect on size, physical stability and particle matrix structure. Int J Pharm 2011; 406: 163–72
   PubMed Web of Science ®Google Scholar
• Lin X, Li X, Zheng LQ, Yu L, Zhang Q, Liu W. Preparation and characterization of monocaprate nanostructured lipid carriers. Colloids Surf A Physicochem Eng Asp 2007; 311(1–3)106–11
   Google Scholar
• Mehnert W, Mader K. Solid lipid nanoparticles: Production, characterization and applications. Adv Drug Deliv Rev 2001; 47(2–3)165–96
   PubMed Web of Science ®Google Scholar
• Melot M, Pudney PD, Williamson AM, Caspers PJ, Van Der Pol A, Puppels GJ. Studying the effectiveness of penetration enhancers to deliver retinol through the stratum cornum by in vivo confocal Raman spectroscopy. J Control Rel 2009; 138(1)32–9
   PubMed Web of Science ®Google Scholar
• Muller RH, Maaben S, Weyhers H, Specht F, Lucks JS. Cytotoxicity of magnetite loaded polylactide, polylactide/glycolide particles and solid lipid nanoparticles. Int J Pharm 1996; 138: 85–94
   Web of Science ®Google Scholar
• Muller RH, Mader K, Gohla S. Solid lipid nanoparticles (SLN) for controlled drug delivery – A review of the state of the art. Eur J Pharm Biopharm 2000; 50: 161–78
   PubMed Web of Science ®Google Scholar
• Pardike J, Hommoss A, Muller RH. Lipid nanoparticles (SLN, NLC) in cosmetic and pharmaceutical dermal products. Int J Pharm 2009; 366: 170–84
   PubMedGoogle Scholar
• Shigematsu T, Shingo T. Modulation of collagen-synthesis and cell-proliferation by retinoids in human skin fibroblasts. J Dermatol Sci 1995; 9: 142–5
   PubMedGoogle Scholar
• Shin SM, Cho BR. Bias-specified robust design optimization and its analytical solutions. Comput Ind Eng 2005; 48: 129–48
   Web of Science ®Google Scholar
• Siekmann B, Westesen K. Sub-micron sized parenteral carrier systems based on solid lipid. Pharm Pharmacol Lett 1992; 1: 123–6
   Google Scholar
• Sorg O, Tran C, Carraux P, Didierjean L, Saurat JH. Retinol and retinyl esters epidermal pools are not identically sensitive to UVB irradiation and anti-oxidant protective effect. Dermatology 1999; 199(4)302–27
   PubMedGoogle Scholar
• Szuts EZ, Harosi FI. Solubility of retinoids in water. Arch Biochem Biophys 1991; 287(2) 297–304
   PubMed Web of Science ®Google Scholar
• Tsunoda T, Takabashy K. Stability of all-trans-retinol in cream. J Soc Cosmet Chem 1995; 46: 191–8
   Web of Science ®Google Scholar
• Vahlquist A. What are natural retinoids?. Dermatol 1999; 1: 3–11
   Google Scholar
• Varani J, Warner JRL, Gharaee-Kermani M, Phan SH, Kang S, Chung J, Wang Z, Datta SC, Fisher GJ, Voorhees JJ. Vitamin A antagonizes decreased cell growth and elevated collagen-degrading matrix metalloproteinases and stimulates collagen accumulation in naturally aged human skin. J Invest Dermatol 2000; 114: 480–6
   PubMed Web of Science ®Google Scholar
• Vining GG, Myers RH. Combining Taguchi and response surface philosophies: A dual response approach. J Qual Technol 1990; 22: 38–45
   Web of Science ®Google Scholar
• Vitorino C, Carvalho FA, Almeida AJ, Sousa JJ, Pais AA. The size of solid lipid nanoparticles: An interpretation from experimental design. Colloids Surf B Biointerfaces 2011; 84: 117–30
   PubMed Web of Science ®Google Scholar
• Wissing SA, Muller RH. Cosmetic applications for solid lipid nanoparticles (SLN). Int J Pharm 2003; 254: 65–68
   PubMed Web of Science ®Google Scholar
• zur Muhlen A, zur Muhlen E, Niehus H, Mehnert W. Atomic force microscopy studies of solid lipid nanoparticles. Pharm Res 1996; 13(9)1411–16
   PubMedGoogle Scholar