330
Views
16
CrossRef citations to date
0
Altmetric
Research Article

Preparation of naproxen–ethyl cellulose microparticles by spray-drying technique and their application to textile materials

, , , , &
Pages 654-666 | Received 04 Sep 2013, Accepted 04 Apr 2014, Published online: 27 May 2014

References

  • Aquacoat® ECD leaflet. Available at: http://www.fmcbiopolymer.com/Portals/bio/content/Docs/AquaCoat%20ECD%207706%20.pdf. Accessed 9 March 2014
  • Argemí A, Ellis JL, Saurina J, Tomasko DL. Development of a polymeric patch impregnated with naproxen as a model of transdermal sustained release system. J Pharm Sci, 2011;100:992–1000
  • Baypret Nano-PU Handout. Available at: http://www.triochem.co.th/file_upload/pdf/file/Baypret%20NANO-PU%20handout-07.pdf. Accessed 9 March 2014
  • Beetge E, du Plessis J, Müller DG, Goosen C, van Rensburg FJ. The influence of the physicochemical characteristics and pharmacokinetic properties of selected NSAID’s on their transdermal absorption. Int J Pharm, 2000;193:261–4
  • Bettinetti G, Mura P, Faucci MT, Sorrenti M, Setti M. Interaction of naproxen with noncrystalline acetyl beta- and acetyl gamma-cyclodextrins in the solid and liquid state. Eur J Pharm Sci, 2002;15:21–9
  • Bhise KS, Dhumal RS, Paradkar AR, Kadam SS. Effect of drying methods on swelling, erosion and drug release from chitosan-naproxen sodium complexes. AAPS PharmSciTech, 2008;9:1–12
  • Blanco MD, Bernardo MV, Sastre RL, Olmo R, Muñiz E, Teijón JM. Preparation of bupivacaine-loaded poly(ε-caprolactone) microspheres by spray drying: Drug release studies and biocompatibility. Eur J Pharm Biopharm, 2003;55:229–36
  • Block JH, Beale JM. 1986. Wilson and Gisvold’s textbook of organic medicinal and drug pharmaceutical chemistry. Philadelphia: Haven Press, p. 759
  • Bodmeier R, Chen H. Preparation and characterization of microspheres containing the anti-inflammatory agents, indomethacin, ibuprofen, and ketoprofen. J Control Release, 1989;10:167–75
  • Bonina FP, Puglia C, Barbuzzi T, de Caprariis P, Palagiano F, Rimoli MG, Saija A. In vitro and in vivo evaluation of polyoxyethylene esters as dermal prodrugs of ketoprofen, naproxen and diclofenac. Eur J Pharm Sci, 2001;14:123–34
  • Brain KR, Walters KA, Watkinson AC. 2002. Methods for studying percutaneous absorption. In: Kenneth AW, ed. Dermatological and transdermal formulations. New York: CRC Press, pp. 197–269
  • Broadhead J, Rouan SKE, Rhodes CT. The spray drying of pharmaceuticals. Drug Dev Ind Pharm, 1992;18:1169–206
  • Canbolat MF, Celebioglu A, Uyar T. Drug delivery system based on cyclodextrin-naproxen inclusion complex incorporated in electrospun polycaprolactone nanofibers. Colloids Surf B Biointerfaces, 2013;115C:15–21
  • Chen H, Mou D, Du D, Chang X, Zhu D, Liu J, Xu H, Yang X. Hydrogel-thickened microemulsion for topical administration of drug molecule at an extremely low concentration. Int J Pharm, 2007;341:78–84
  • Costa P, Sousa Lobo JM. Modelling and comparison of dissolution profiles. Eur J Pharm Sci, 2001;13:123–33
  • Dahl TC. 2006. Ethylcellulose. In: Rowe RC, Sheskey PJ, Owen SC, eds. Handbook of pharmaceutical excipients. London: Pharmaceutical Press
  • Desai KGH, Park HJ. Preparation and characterization of drug-loaded chitosan-tripolyphosphate microspheres by spray drying. Drug Dev Res, 2005;64:114–28
  • Dürig T, Harcum WW, Lusvardi KM, Skinner GW. Compaction characteristics of high ethoxyl, low viscosity ethylcellulose. Pharmaceutical Technology Report 2003. 024. Wilmington, DE: Hercules Incorporated, Aqualon Division
  • Esposito E, Roncarati R, Cortesi R, Cervellati F, Nastruzzi C. Production of Eudragit microparticles by spray-drying technique: Influence of experimental parameters on morphological and dimensional characteristics. Pharm Dev Technol, 2000;5:267–78
  • Fisher G. Medical and hygiene textiles – continuing in good health. Tech Textil Int 2002;11:10–16
  • Ghorab MM, Zia H, Luzzi LA. Preparation of controlled release anticancer agents. I: 5-Fluorouracil-ethyl cellulose microspheres. J Microencapsul, 1990;7:447–54
  • Gouin S. Microencapsulation: Industrial appraisal of existing technologies and trends. Trends Food Sci Tech, 2004;15:330–47
  • Guy RH, Hadgraft J. 1989. Selection of drug candidates for transdermal delivery. In: Hadgraft J, Guy RH, eds. Transdermal drug delivery. Developmental issues and research initiatives. New York: Marcel Dekker, pp. 59–81
  • Hadzija BW, Ruddy SB, Ballenger ES. Effect of freezing on iontophoretic transport through hairless rat skin. J Pharm Pharmacol, 1992;44:387–90
  • Hawkins GS, Reifenrath WG. Development of an in vitro model for determining the fate of chemicals applied to skin. Fund Appl Toxicol, 1984;4:S133–44
  • Higuchi T. Physical chemical analysis of percutaneous absorption process from creams and ointments. J Soc Cosmet Mater, 1960;11:85–97
  • Hippler UC, Elsner P. 2006. Biofunctional textiles and the skin. Current problems in dermatology. Basel: S. Karger AG
  • Horrocks AR, Anand SC. 2003. Teknik Tekstiller El Kitabı (Technical textiles handbook). Istanbul: The Textile Institute, Türk Tekstil Vakfı
  • Huang J, Wigent RJ, Schwartz JB. Drug-polymer interaction and its significance on the physical stability of nifedipine amorphous dispersion in microparticles of an ammonio methacrylate copolymer and ethylcellulose binary blend. J Pharm Sci, 2008;97:251–62
  • Johnson ME, Blankschtein D, Linger R. Evaluation of solute permeation through the stratum corneum: Lateral bilayer diffusion as the primary transport mechanism. J Pharm Sci, 1997;86:1162–72
  • Kenawy el-R, Bowlin GL, Mansfield K, Layman J, Simpson DG, Sanders EH, Wnek GE. Release of tetracycline hydrochloride from electrospun poly(ethylene-co-vinylacetate), poly(lactic acid), and a blend. J Control Release, 2002;81:57–64
  • Kiliçarslan M, Baykara T. The effect of the drug/polymer ratio on the properties of the verapamil HCl loaded microspheres. Int J Pharm, 2003;252:99–109
  • Kim JC, Lee HY, Kim MH, Lee HJ, Kang HY, Kim SM. Preparation and characterization of chitosan/gelatin microcapsules containing triclosan. Colloids Surf B Biointerfaces, 2006;52:52–6
  • Korsmeyer RW, Gurny R, Docler E, Buri P, Peppas NA. Mechanism of solute release from porous hydrophilic polymers. Int J Pharm, 1983;15:25–35
  • Liu J, Liu C, Liu Y, Chen M, Hu Y, Yang Z. Study on the grafting of chitosan-gelatin microcapsules onto cotton fabrics and its antibacterial effect. Colloids Surf B Biointerfaces, 2013;109:103–8
  • Ma ZH, Yu DG, Branford-White CJ, Nie HL, Fan ZX, Zhu LM. Microencapsulation of tamoxifen: Application to cotton fabric. Colloids Surf B Biointerfaces, 2009;69:85–90
  • Marinković SS, Bezbradica D, Škundrić P. Microencapsulation in the textile industry. Chem Ind Chem Eng Q, 2006;12:58–62
  • Masters K. 1972. Spray drying: An introduction to principles, operational practice and applications. London: Leonard Hill Books
  • Mukherjee B, Mahapatra S, Gupta R, Patra B, Tiwari A, Arora P. A comparison of povidone-ethylcellilose and povidone-eidragit transdermal dexamethasone matrix patches based on in vitro skin permeation. Eur J Pharm Biopharm, 2005;59:475–83
  • Mura P, Zerrouk N, Mennini N, Maestrelli F, Chemtob C. Development and characterization of naproxen-chitosan solid systems with improved drug dissolution properties. Eur J Pharm Sci, 2003;19:67–75
  • Nelson G. Application of microencapsulation in textiles. Int J Pharm, 2002;242:55–62
  • Nierstrasz VA. 2007. Textile-based drug release systems. In: Langenhove LV, ed. Smart textiles for medicine and healthcare: Materials, systems and applications. Cambridge: Woodhead Publishing Ltd and CRC Press, pp. 50–74
  • Okonogi S, Yonemochi E, Oguchi T, Puttipipatkhachorn S, Yamamoto K. Enhanced dissolution of ursodeoxycholic acid from the solid dispersion. Drug Dev Ind Pharm, 1997;23:1115–21
  • Okyar A, Özsoy Y, Güngör S. 2012. Novel formulation approaches for dermal and transdermal delivery of non-steroidal anti-inflammatory drugs. In: Lemmey A, ed. Rheumatoid arthritis – Treatment. Rijeka: InTech, pp. 25–48
  • Ozyazici M, Sevgi F, Pekcetin C, Sarpas B, Sayin S. Sustained release spherical agglomerates of polymethacrylates containing mefenamic acid: In vitro release, micromeritic properties and histological studies. Pharm Dev Technol, 2012;17:483–93
  • Paudel A, Van den Mooter G. Influence of solvent composition on the miscibility and physical stability of naproxen/PVP K 25 solid dispersions prepared by cosolvent spray-drying. Pharm Res, 2012;29:251–70
  • Peppas NA. Analysis of Fickian and non-Fickian drug release from polymers. Pharm Acta Helv, 1985;60:110–11
  • Puglia C, Blasi P, Rizza L, Schoubben A, Bonina F, Rossi C, Ricci M. Lipid nanoparticles for prolonged topical delivery: An in vitro and in vivo investigation. Int J Pharm, 2008;357:295–304
  • Puglia C, Bonina F, Rizza L, Cortesi R, Merlotti E, Drechsler M, Mariani P, Contado C, Ravani L, Esposito E. Evaluation of percutaneous absorption of naproxen from different liposomal formulations. J Pharm Sci, 2010;99:2819–29
  • Rattes ALR, Oliveria WP. Spray drying conditions and encapsulating composition effects on formation and properties of sodium diclofenac microparticles. Powder Technol, 2007;171:7–14
  • Ré MI, Biscans B. Preparation of microspheres of ketoprofen with acrylic polymers by a quasi emulsion solvent diffusion method. Powder Technol, 1999;101:120–33
  • Rinaki E, Valsami G, Macheras P. The power law can describe the ‘entire’ drug release curve from HPMC-based matrix tablets: A hypothesis. Int J Pharm, 2003;255:199–207
  • Rodrigues SN, Martins IM, Fernandes IP, Gomes PB, Mata VG, Barreiro MF, Rodrigues AE. Scentfashion®: Microencapsulated perfumes for textile application. Chem Eng J, 2009;149:463–72
  • Sakellariou P, Rowe RC, White EFT. The thermomechanical properties and glass transition temperatures of some cellulose derivatives used in film coatings. Int J Pharm, 1985;27:267–77
  • Saravanan M, Bhaskar K, Srinivasa Rao G, Dhanaraju MD. Ibuprofen-loaded ethylcellulose/polystyrene microspheres: An approach to get prolonged drug release with reduced burst effect and low ethylcellulose content. J Microencapsul, 2003;20:289–302
  • Sariisik M, Arici M, Topbas O, Karavana SY, Ozturk C, Ertan G. Design of orthopedic support material containing diclofenac sodium microparticles: Preparation and characterization of microparticles and application to orthopedic support material. Text Res J, 2013;83:1030–43
  • Shah VP, Elkins J, Lam SY, Skelly JP. Determination of in vitro drug release from hydrocortisone creams. Int J Pharm, 1989;53:53–9
  • Singh P, Roberts MS. Skin permeability and local tissue concentration of nonsteriodal anti-inflammatory drugs after topical application. J Pharmacol Expt Ther, 1994;268:144–51
  • Streubel A, Siepmann J, Bodmeier R. Floating microparticles based on low density foam powder. Int J Pharm, 2002;241:279–92
  • Swart H, Breytenbach JC, Hadgraft J, du Plessis J. Synthesis and transdermal penetration of NSAID glycoside esters. Int J Pharm, 2005;301:71–9
  • Thies C. 1996. A survey of microencapsulation processes. In: Benita S, ed. Microencapsulation methods and industrial applications. New York: Marcel Dekker, pp. 1–21
  • Tripathi KD. 2003. Essentials of medical pharmacology. New Delhi: Jaypee Brothers Medical Publishers, pp. 176–7
  • Ustündağ Okur N, Apaydın S, Karabay Yavaşoğlu NÜ, Yavaşoğlu A, Karasulu HY. Evaluation of skin permeation and anti-inflammatory and analgesic effects of new naproxen microemulsion formulations. Int J Pharm, 2011;416:136–44
  • Vasiliu S, Popa M, Rinaudo M. Polyelectrolyte capsules made of two biocompatible natural polymers. Eur Polym J, 2005;41:923–32
  • Walters KA, Brain KR, Green DM, James VG, Watkinson AC, Sands RH. Comparison of the transdermal delivery of estradiol from two gel formulations. Maturitas, 1998;29:189–95
  • Wang FJ, Wang CH. Sustained release of etanidazole from spray dried microspheres prepared by non-halogenated solvents. J Control Release, 2002;81:263–80
  • Won DH, Kim MS, Lee S, Park JS, Hwang SJ. Improved physicochemical characteristics of felodipine solid dispersion particles by supercritical antisolvent precipitation process. Int J Pharm, 2005;301:199–208
  • Yamada T, Onishi H, Machida Y. Sustained release ketoprofen microparticles with ethylcellulose and carboxymethylethylcellulose. J Control Release, 2001;75:271–82
  • Yiping H, Xiaolie L, Dezhu M. Ringed spherulite morphology and compatibility in the binary blends of poly(ε-caprolactone) with ethyl cellulose. Eur Polym J, 2001;37:2153–7
  • Zahedi P, Lee PI. Solid molecular dispersions of poorly water-soluble drugs in poly(2-hydroxyethyl methacrylate) hydrogels. Eur J Pharm Biopharm, 2007;65:320–8
  • Zakeri-Milani P, Barzegar-Jalali M, Tajerzadeh H, Azarmi Y, Valizadeh H. Simultaneous determination of naproxen, ketoprofen and phenol red in samples from rat intestinal permeability studies: HPLC method development and validation. J Pharm Biomed Anal, 2005;39:624–30

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.