304
Views
14
CrossRef citations to date
0
Altmetric
Original Article

Physicochemical studies of binary eutectic of ibuprofen and ketoprofen for enhanced transdermal drug delivery

&
Pages 1168-1176 | Received 08 Jun 2009, Accepted 11 Feb 2010, Published online: 05 Apr 2010

References

  • Lawrence RC, Helmick CG, Arnett FC, Deyo RA, Felson DT, Giannini EH, . (1998). Estimates of the prevalence of arthritis and selected musculoskeletal disorders in the United States. Arthritis Rheum, 41(5):778–99.
  • Centers for Disease Control and Prevention (CDC), National Center for Chronic Disease Prevention and Health Promotion. (2002). The national arthritis action plan: A public health strategy (NAAP), Atlanta, GA: CDC.
  • Rovensky J, Micekova D, Gubzova Z, Fimmers R, Lenhard G, Vogtle-Junkert U, . (2001). Treatment of knee osteoarthritis with a topical non-steroidal antiinflammatory drug. Results of a randomized, double-blind, placebo-controlled study on the efficacy and safety of a 5% ibuprofen cream. Drugs Exp Clin Res, 27(5–6):209–21.
  • Vaile JH, Davis P. (1998). Topical NSAIDs for musculoskeletal conditions. A review of the literature. Drugs, 56(5):783–99.
  • Chlud K. (1991). Percutaneous therapy of painful arthritis. Ther Umsch, 48(1):42–5.
  • Valenta C, Wanka M, Heidlas J. (2000). Evaluation of novel soya-lecithin formulations for dermal use containing ketoprofen as a model drug. J Control Release, 63(1–2):165–73.
  • Calpena AC, Blanes C, Moreno J, Obach R, Domenech J. (1994). A comparative in vitro study of transdermal absorption of antiemetics. J Pharm Sci, 83(1):29–33.
  • Kasting GB, Smith RL, Cooper ER. (1987). Effects of lipid solubility and molecular size on percutaneous absorption. Basel: Karger, Pharmacol Skin, 1(1):138–53.
  • Touitou E, Chow DD, Chaw JR. (1994). Chiral β-blockers for transdermal delivery. Int J Pharm, 104(1):19–28.
  • Grant DJW, Abougela IKA, Liversidge GG, Padfield JM, Dooren AAV, Hardy MJ, . (1982). Applications of thermal methods of analysis in the pharmaceutical industry. Anal Proc, 19(12):545–9.
  • Ford JL, Timmins P. (1989). Pharmaceutical thermal analysis: Techniques and applications (Ellis Horwood Series in Pharmaceutical Technology). New York: Ellis Horwood Ltd, 47–67.
  • Brodin A, Nyqvist-Mayer A, Wadsten T, Forslund B, Broberg F. (1984). Phase diagram and aqueous solubility of the lidocaine-prilocaine binary system. J Pharm Sci, 73(4):481–4.
  • Nyqvist-Mayer AA, Brodin AF, Frank SG. (1985). Phase distribution studies on an oil-water emulsion based on a eutectic mixture of lidocaine and prilocaine as the dispersed phase. J Pharm Sci, 74(11):1192–5.
  • Nyqvist-Mayer AA, Brodin AF, Frank SG. (1986). Drug release studies on an oil-water emulsion based on a eutectic mixture of lidocaine and prilocaine as the dispersed phase. J Pharm Sci, 75(4):365–73.
  • Ke GM, Wang L, Wang P, Lu WL, Wang SM, Zhang Q, . (2005). In vitro transdermal permeation of lidocaine-dodecanol binary eutectic system. Yao Xue Xue Bao, 40(8):764–8.
  • Yong CS, Jung SH, Rhee JD, Choi HG, Lee BJ, Kim DC, . (2003). Improved solubility and in vitro dissolution of ibuprofen from poloxamer gel using eutectic mixture with menthol. Drug Deliv, 10(3):179–83.
  • Stott PW, Williams AC, Barry BW. (1998). Transdermal delivery from eutectic systems: Enhanced permeation of a model drug, ibuprofen. J Control Release, 50(1–3):297–308.
  • Yuan X, Capomacchia AC. (2005). The binary eutectic of NSAIDs and two phase liquid system for enhanced membrane penetration. Pharm Dev Technol, 10(1):1–10.
  • Garner ST, Israel BJ, Ahmed H, Capomacchia AC. (2007). Transdermal permeability of N-acetyl-D-glucosamine. Pharm Dev Technol, 12(2):169–74.
  • Moghimi HR, Barry BW, Williams AC. (1999). Stratum corneum and barrier performance. In: Bronaugh RL, Maibach HI, eds. Percutaneous absorption. 3rd ed. New York: Marcel Dekker, 518–22.
  • Itoh T, Xia J, Magavi R, Nishihata T, Rytting JH. (1990). Use of shed snake skin as a model membrane for in vitro percutaneous penetration studies: Comparison with human skin. Pharm Res, 7(10):1042–7.
  • Higuchi T, Konishi R. (1987). In vitro testing and transdermal delivery. Proceedings of the 2nd Transdermal Therapeutic Symposium. Ther Res, 6:280–8.
  • Ngawhirunpat T, Panomsuk S, Opanasopit P, Rojanarata T, Hatanaka T. (2006). Comparison of the percutaneous absorption of hydrophilic and lipophilic compounds in shed snake skin and human skin. Pharmazie, 61(4):331–5.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.