660
Views
12
CrossRef citations to date
0
Altmetric
Research Article

A material sparing test to predict punch sticking during formulation development

&
Pages 1054-1060 | Received 27 Jul 2011, Accepted 01 Nov 2011, Published online: 19 Dec 2011

References

  • Roberts M, Ford JL, MacLeod GS, Fell JT, Smith GW, Rowe PH. (2003). Effects of surface roughness and chrome plating of punch tips on the sticking tendencies of model ibuprofen formulations. J Pharm Pharmacol, 55:1223–1228.
  • Wang JL, Tonglei L, Bateman SD, Erck R, Morris KR. (2003). Modeling of adhesion in tablet compression-I. Atomic force microscopy and molecular simulation. J Pharm Sci, 92:798–814.
  • Gordon RE, VanKoevering CL, and Reits DJ. (1984). Utilization of differential scanning calorimetry in the compatibility screening of ibuprofen with the stearate lubricants and construction of phase diagrams. Int J Pharm, 21:99–105.
  • Danjo K, Kojimo S, Chen CY, Sunada H, Otsuka A. (1997). Effect of water content on sticking during compression. Chem Pharm Bull, 45:706–709.
  • Roberts M, Ford JL, MacLeod GS, Fell JT, Smith GW, Rowe PH et al. (2004). Effect of lubricant type and concentration on the punch tip adherence of model ibuprofen formulations. J Pharm Pharmacol, 56:299–305.
  • Waimer F, Krumme M, Danz P, Tenter U, Schmidt PC. (1999). A novel method for the detection of sticking of tablets. Pharm Dev Technol, 4:359–367.
  • Matoba H, Yoshikawa T, Makino T, Sato K. (2000). Crystalline transition and interaction of drugs and the phenomenon of sticking to the punch during preparation procedures. Pharm Tech Japan, 16:1057–1067.
  • Riepma KA, Vromans H, Lerk CF. (1993). A coherent matrix model for the consolidation and compaction of an excipient with magnesium stearate. Int J Pharm, 97:195–203.
  • Vromans H, Bolhuis GK, Lerk CF. (1988). The evaluation of the magnesium stearate susceptibility of directly compressible materials as an indication for fragmentation properties. Powder Technol, 54:39–44.
  • Roberts M, Ford JL, MacLeod GS, Fell JT, Smith GW, Rowe PH et al. (2004). Effect of punch tip geometry and embossment on the punch tip adherence of a model ibuprofen formulation. J Pharm Pharmacol, 56:947–950.
  • Newton, JM, Haririan I, and Podzeck F. (2000). The influence of punch curvature on the mechanical properties of compacted powders. Powder Tech, 107:79–83.
  • Sixsmith D, McCluskey D. (1981). The effect of punch tip geometry on powder movement during the tableting process. J Pharm Pharmacol, 33:79–81.
  • Matsumoto R, Kawakami K, Aoki S. (2007). Impact of compression pressure on tablet appearance. Int J Pharm, 341:44–49.
  • Waimer F, Krumme M, Danz P, Tenter U, Schmidt PC. (1999). The influence of engravings on the sticking of tablets. Investigations with an instrumented upper punch. Pharm Dev Technol, 4:369–375.
  • Mitrevej KT, Augsbuger LL. (1982). Adhesion of tablets in a rotary tablet press II. Effects of blending time, running time, and lubricant concentration. Drug Dev Ind Pharm, 8:237–282.
  • Ando T, Kanaya Y, Yajima Y, Hiura M. (1990). Prevention of sticking to punches by coating with lactose in tableting of bencyclane fumarate. Yakuzaigaku, 50:300–306.
  • Schumann S, Searle GD. (1992). The effects of Chromium nitride ion bombardment treatment of tablet tooling on tablet adherence. Drug Dev Ind Pharm, 18:1037–1061.
  • Watanabe Y, Endo K, Koizumi K, Matsumoto M. (1998). A new compression tableting method using a punch coated with amorphous alloys. J Pharm Sci Technol, 58:147–154.
  • Toyoshima K, Yasumura M, Ohnishi N, Ueda Y. (1988). Quantitative evaluation of tablet sticking by surface roughness measurement. Int J Pharm, 46:211–215.
  • Sendall FE, Staniforth JN. (1986). A study of powder adhesion to metal surfaces during compression of effervescent pharmaceutical tablets. J Pharm Pharmacol, 38:489–493.
  • Narayan P, Hancock BC. (2003). The relationship between the particle properties, mechanical behaviour, and surface roughness of some pharmaceutical excipient compacts. Mat Sci Eng, A355:24–36.
  • Wang JJ, Guillot MA, Bateman SD, Morris KR. (2004). Modeling of adhesion in tablet compression. II. Compaction studies using a compaction simulator and an instrumented tablet press. J Pharm Sci, 93:407–417.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.