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Research Article

Formulation studies on ibuprofen sodium–cationic dextran conjugate: effect on tableting and dissolution characteristics of ibuprofen

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Pages 39-59 | Received 16 Sep 2014, Accepted 23 Feb 2015, Published online: 31 Mar 2015

References

  • Han LH, Elliott JA, Bentham AC, et al. A modified Drucker–Prager Cap model for die compaction simulation of pharmaceutical powders. Int J Solids Struct 2008;45:3088–106
  • Prescott JK, Barnum RA. On powder flowability. Pharm Technol 2000;10:60–84.
  • British National Formulary. Musculoskeletal and joint diseases. September ed. UK: Pharmaceutical Press; 2013
  • Nokhodchi A, Amire O, Jelvehgari M. Physico-mechanical and dissolution behaviours of ibuprofen crystals crystallized in the presence of various additives. DARU 2010;18:74–83
  • Abioye A, Kola-Mustapha A, Ruparelia K. Impact of insitu granulation and temperature quenching on crystal habit and micromeritic properties of ibuprofen-cationic dextran conjugate crystanules. Int J Pharm 2014;462:83–102
  • Abioye A, Kola-Mustapha A, Chi GT, Iliya S. Quantification of in situ granulation-induced changes in pre-compression, solubility, dose distribution and intrinsic in vitro release characteristics of ibuprofen-cationic dextran conjugate crystanules. Int J Pharm 2014;471:453–77
  • Rasenack N, Muller BW. Crystal habit and tablet behaviour of ibuprofen. Int J Pharm 2002;244:45–57
  • Nada HA, Al-Saidan MS, Mueller WB. Crystal modification for improving the physical and chemical properties of ibuprofen. Pharm Technol 2005;29:90–101
  • Rasenack N, Muller BW. Ibuprofen crystals with optimized properties. Int J Pharm 2002;245:9–24
  • Lerk C, Lagas M, Fell J, Nauta P. Effect of hydrophilization of hydrophobic drugs on release rate from capsules. J Pharm Sci 1978;67:935–9
  • Ehlers H, Antikaninen O, Heinamaki J, Yliruusi J. Improving flow properties of Ibuprofen by fluidized bed particle thin-coating. Int J Pharm 2009;368:165–70
  • Genina N, Raikkonen H, Ehlers H, et al. Thin coating as an alternative approach to improve flow properties of Ibuprofen powder. Int J Pharm 2010;387:65–70
  • Kachimanis K, Nikolakakis I, Malamataris S. Tensile strength and disintegration of tableted silicified microcrystalline cellulose: influences on interparticle bonding. J Pharm Sci 2003;92:1489–501
  • Khan MA, Bolton S, Kislalioglu MS. Optimization of Process variables for the preparation of Ibuprofen coprecipitates with Eudragit S100. Int J Pharm 1994;102:185–92
  • Kachrimanis K, Ktistis G, Malamataris S. Crystallization conditions and physicochemical properties of ibuprofen-Eudragit S100 spherical crystal agglomerates prepared by solvent-change technique. Int J Pharm 1998;173:61–74
  • Pawar A, Paradkar A, Kadam S, Mahadik K. Agglomeration of ibuprofen with talc by novel crystallo-co-agglomeration technique. AAPS PharmSciTech 2004;5:Article 55
  • Dhaneshwar SS, Kandpal M, Gairola N, Kadam SS. Dextran: a promising macromolecular drug carrier. Indian J Pharm Sci 2006;68:705–14
  • Di Martino P, Beccerica M, Joiris E, et al. Influence of crystal habit on the compression and densification mechanism of ibuprofen. J Cryst Growth 2002;243:345–55
  • Duckworth WH. Discussion of Ryshkewitch paper by Winston Duckworth. J Am Ceram Soc 1953;36:68
  • Maarschalk KV, Vromans H, Groenendijk W, et al. Effect of water on deformation and bonding of pregelatinized starch compacts. Eur J Pharm Biopharm 1997;44:253–60
  • Heckel RW. Density-Pressure relationships in powder compaction. Trans Metall Soc AIME 1961;221:671–5
  • Heckel RW. An analysis of powder compaction phenomena. Trans Metall Soc AIME 1961;221:1001–8
  • Humbert-Droz P, Gurny R, Mordier D, Doelker E. Densification behaviour of drugs presenting availability problems. Int J Pharm Tech Prod Mfr 1983;4:29–35
  • Doelker E. Assessment of powder compaction. In: Chulia D, Deleuil M, Pourcelot Y, eds. Powder technology and pharmaceutical process. Amsterdam: Elsevier; 1994:403
  • Costa P. An alternative method to the evaluation of similarity factor in dissolution testing. Int J Pharm 2001;220:77–83
  • Romero AJ, Savastano L, Rhodes CT. Monitoring crystal modifications in systems containing ibuprofen. Int J Pharm 1993;99:125–34
  • Wong LW, Pilpel N. The effect of particle shape on the mechanical properties of powders. Int J Pharm 1990;59:145–54
  • Coates J. Interpretation of infrared spectra: a practical approach. In: Meyers RA, ed. Encyclopedia of analytical chemistry. Chichester: Wiley; 2000:10815–37
  • Lambert JB, Shurvell HF, Lightner DA, Cooks RG. Organic structural spectroscopy. New Jersey: Prentice Hall Inc.; 1998
  • Lee T, Chen YH, Zhang CW. Solubility, polymorphism, crystallinity, crystal habit and drying scheme of (R,S)-(±)-sodium ibuprofen dehydrate. Pharm Technol 2007;31:72–87
  • Amato ME, Djedani F, Pappalardo GC, et al. Molecular modeling of β-cyclodextrin complexes with nootropic drugs. J Pharm Sci 1992;81:1157–61
  • Rodreguez R, Alvarez-Lorenzo C, Concheiro A. Interactions of ibuprofen with cationic polysaccharide in aqueous dispersions and hydrogels: rheological and diffusional implications. Eur J Pharm Sci 2003;20:429–38
  • Nokhodchi A, Rubinstein MH, Larhrib H, Gyuot JC. The effect of moisture on the properties of Ibuprofen tablets. Int J Pharm 1995;118:191–7
  • Shi L, Feng Y, Sun CC. Initial moisture content in raw material can profoundly influence high shear wet granulation process. Int J Pharm 2011;416:43–8
  • Garr JSM, Robinstein MH. The influence of moisture on consolidation and compaction properties of paracetamol. Int J Pharm 1992;81:187–92
  • Shi L, Feng Y, Sun CC. Roles of granule size in over-granulation during high shear wet granulation. J Pharm Sci 2010;99:3322–5
  • Johansson B, Alderborn G. Degree of pellets deformation during compaction and its relationship to the tensile strength of tablets formed of microcrystalline cellulose. Int J Pharm 1996;132:207–20
  • Santos H, Veiga F, Pina ME, Sousa JJ. Compaction, compression and drug release properties of diclofenac sodium and ibuprofen pellets comprising xanthan gum as a sustained release agent. Int J Pharm 2005;295:15–27
  • Adolfsson Å, Caramella C, Nyström C. The effect of milling and addition of dry binder on the interparticulate bonding mechanism in sodium chloride tablets. Int J Pharm 1998;160:187–95
  • Alderborn G, Nyström C. Studies on direct compression of tablets IV. The effect of particle size on the mechanical strength of tablets. Acta Pharm Suec 1982;19:381–90
  • Roberts RJ, Rowe RC. Brittle/ductile behaviour in pharmaceutical materials used in tabletting. Int J Pharm 1987;36:205–9
  • Ghosh LK, Ghosh NC, Chatterjee M, Gupta BK. Product development studies on the tablet formulation of ibuprofen to improve bioavailability. Drug Dev Ind Pharm 1998;24:473–7
  • Abioye A, Kola-Mustapha A. Controlled electrostatic self-assembly of ibuprofen-cationic dextran nanoconjugates prepared by low energy green process – a novel delivery tool for poorly soluble drugs. Pharm Res [Epub ahead of print]. DOI: 10.1007/s11095-014-1603-0
  • Oliveira RB, Nascimento TL, Lima EM. Design and characterization of sustained release ketoprofen-entrapped carnauba wax microparticles. Drug Dev Ind Pharm 2012;38:1–11
  • Costa P, Lobo JMS. Modelling and comparison of dissolution profiles. Eur J Pharm Sci 2001;13:123–33

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