281
Views
13
CrossRef citations to date
0
Altmetric
Non-themed Articles

Physicochemical properties and mechanisms of drug release from melt-extruded granules consisting of chlorpheniramine maleate and Eudragit FS

Pages 563-571 | Received 03 Mar 2015, Accepted 21 May 2015, Published online: 11 Jun 2015

References

  • Zhang F, McGinity JW. Properties of sustained release tablets prepared by hot-melt extrusion. Pharm Dev Technol 1999;4:241–50
  • Sprockel OL, Price JC, Jennings R, et al. In vitro/in vivo evaluation of a liquid sustained-release dosage form of chlorpheniramine. Drug Dev Ind Pharm 1989;15:1393–404
  • Bruce DL, Koleng JJ, McGinity JW. The influence of polymeric subcoat and pellet formulation on the release of chlorphenarime maleate from enteric coated pellets. Drug Dev Ind Pharm 2003;29:909–25
  • Kassem AA, El-Assasy AE, Said SA, El-Kady SF. Sustained release chlorpheniramine maleate tablets. Bull Faculty Pharmacy 1976;14:75–84
  • Friesen D, Shanker R, Crew M, Smithey D. Hydroxypropyl methylcellulose based spray-dried dispersions: an overview. Mol Pharm 2008;5:1003–19
  • Laarhoven JAHv, Kruft MAB, Vromans H. Effect of supersaturation and crystallization phenomena on the release properties of a controlled release device based on EVA copolymer. J Control Release 2002;82:309–19
  • Follonier N, Doelker E, Cole E. Evaluation of hot-melt extrusion as a new technique for the production of polymer-based pellets for sustained-release capsules containing high loading of freely water soluble drugs. Drug Dev Ind Pharm 1994;20:1323–39
  • Zhu Y, Shah NH, Malick AW, et al. Controlled release of a poorly water-soluble drug from hot-melt extrudates containing acrylic polymers. Drug Dev Ind Pharm 2006;32:569–83
  • Ma D, Djemai A, Gendorn C, et al. Development of a HPMC-based controlled release formulation with hot melt extrusion. Drug Dev Ind Pharm 2013;39:1070–83
  • Loreti G, Maroni A, Del Curto MD, et al. Evaluation of hot-melt extrusion technique in the preparation of HPC matrices for prolonged release. Eur J Pharm Sci 2014;52:77–85
  • Yang R, Wang Y, Zheng X, et al. Preparation and evaluation of ketoprofen hot-melt extruded enteric and sustained-release tablets. Drug Dev Ind Pharm 2008;34:83–9
  • Bouman J, Belton P, Venema P, et al. The development of direct extrusion-injection moulded zein matrices as novel oral controlled drug delivery systems. Pharm Res 2015. [Epub ahead of print]. doi: 10.1007/s11095-015-1663-9
  • Crowley MM, Schroeder B, Fredersdorf A, et al. Physicochemical properties and mechanism of drug release from ethyl cellulose matrix tablets prepared by direct compression and hot-melt extrusion. Int J Pharm 2004;269:509–22
  • Dvorracckova K, Rabiskova M, Muselik J, et al. Coated hard capsules as pH-dependent drug transport systems to ileo-colonic compartment. Drug Dev Ind Pharm 2011;37:1131–40
  • Kulthe SS, Bahekar JK, Godhani CC, et al. Modulated release of 5-fluorouracil from pH-sensitive and colon targeted pellets: an industrially feasible approach. Drug Dev Ind Pharm 2013;39:138–45
  • Young C, Dietzsch C, McGinity JW. Compression of controlled-release pellets produced by hot-melt extrusion and spheronization process. Pharm Dev Technol 2005;10:133–9
  • Higuchi T. Mechanism of sustained-action medication. Theoretical analysis of rate of release of solid drugs dispersed in solid matrices. J Pharm Sci 1963;52:1145–9
  • Siepmann J, Peppas NA. Higuchi equation: derivation, applications, use and misuse. Int J Pharm 2011;418:6–12
  • Carli F, Motta A. Particle size and surface area distributions of pharmaceutical powders by microcomputerized mercury porosimetry. J Pharm Sci 1984;73:197–203
  • Ertel KD, Zoglio MA, Ritschel WA, Carstensen JT. Physical aspects of wet granulation 4. Effect of kneading time on dissolution rate and tablet properties. Drug Dev Ind Pharm 1990;16:963–81
  • Zoglio MA, Carstensen JT. Physical aspects of wet granulation 3. Effect of wet granulation on granule porosity. Drug Dev Ind Pharm 1983;9:1417–34
  • Rubio MR, Ghaly ES. In-vitro release of acetaminophen from sodium alginate controlled-release pellets. Drug Dev Ind Pharm 1994;20:1239–51
  • Ardusso M, Manzo R, Jimenez-Kairuz A. Comparative study of three structurally related acid polyelectrolyes as carriers of basic drug. Supramol Chem 2010;22:289–96
  • Elkheshen SA. Interaction of verapamil hydrochloride with carbopol 934P and its effect on the release rate of the drug and the water uptake of the polymer matrix. Drug Dev Ind Pharm 2001;27:925–34
  • Saettone MF, Monti D, Torracca MT, et al. Muco-adhesive liquid ophthalmic vehicles – evaluation of macromolecular ionic complexes of pilocarpine. Drug Dev Ind Pharm 1989;15:2475–89
  • Petereite HU, Meier C, Gryczke A. Melt extrusion consisting of salts of active ingredients. WO03/072083 A2;2003
  • Maniruzzaman M, Boateng JS, Chowdhry BZ, et al. A review on the taste masking of bitter APIs: hot-melt extrusion (HME) evaluation. Drug Dev Ind Pharm 2014;40:145–56
  • Moustafine RI, Kabanova TV, Kemenova VA, Mooter GVd. Characteristics of interpolyelectrolyte complexes of Eudragit E100 with Eudraigt L100. J Control Release 2005;103:191–8
  • Gryczke A, Schminke S, Maniruzzaman M, et al. Development and evaluation of orally disintegrating tablets (ODTs) containing ibuprofen granules prepared by hot melt extrusion. Colloids Surf B: Biointerfaces 2011;86:275–84
  • Plaizier-Vercammen JA. Interaction of povidone with aromatic compounds. IV: effect of macromolecule molecular weight, solvent dielectric constant, and ligand solubility on complex formation. J Pharm Sci 1983;72:1042–4
  • Higuchi T, Kuramoto R. Study of possible complex formation between macromolecules and certain pharmaceuticals. I. Polyvinylpyrrolidone with sulfathiazole, procaine hydrochloride, sodium salicylate, benzyl penicillin, chloramphenicol, mandelic acid, caffeine, theophylline, and cortisone. J Am Pharm Assoc 1954;43:393–7
  • Gill SJ, Robert CH, Wymn J. Biochemical thermodynamics. 2nd edn. Amsterdam: Elsevier; 1988
  • Nogueiras-Nieto L, Sobarzo-Sánchez E, Gómez-Amoza JL, Otero-Espinar FJ. Competitive displacement of drugs from cyclodextrin inclusion complex by polypseudorotaxane formation with poloxamer: implications in drug solubilization and delivery. Eur J Pharm Biopharm 2012;80:585–95
  • Frenning G. Modelling drug release from inert matrix systems: from moving-boundary to continuous-field descriptions. Int J Pharm 2011;418:88–99
  • DiNunzio JC, Martin C, Zhang F. Melt extrusion: shaping drug delivery in the 21st century. Pharm Technol 2010;10:30–7
  • Nyström C, Alderborn G, Duberg M, Karehill P-G. Bonding of surface area and bonding mechanism – two important factors for the understanding of powder compactability. Drug Dev Ind Pharm 1993;19:2143–96
  • Caraballo I, Millan M, Rabasco AM. Relationship between drug percolation threshold and particle size in matrix tablets. Pharm Res 1996;13:387–90
  • Elarini SK, Leuenberger H. Modeling of drug-release from polymer matrices – effect of drug loading. Int J Pharm 1995;121:141–8
  • Bruce LD, Koleng JJ, McGinity JW. The influence of polymeric subcoats and pellet formulation on the release of chlorpheniramine maleate from enteric coated pellets. Drug Dev Ind Pharm 2003;29:909–24

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.