223
Views
25
CrossRef citations to date
0
Altmetric
Research Article

Liposomal solubilization of new 3-hydroxy-quinolinone derivatives with promising anticancer activity: a screening method to identify maximum incorporation capacity

, , , , &
Pages 272-278 | Received 02 Sep 2010, Accepted 01 Dec 2010, Published online: 17 Feb 2011

References

  • Bangham, A. D., Horne, R. W. (1964). Negative staining of phospholipids and their structural modification by surface active agents as observed in the electron microscope. J Mol Biol 8:660–668.
  • Brandl, M. (2003). Liposomal drug carriers for cancer diagnosis and therapy. In: Budman, D. R., Calvert, A. H., Rowinsky, E. K. (Eds.), Handbook of anticancer drug development (pp 225–237). Philadelphia, Pennsylvania, USA: Lippincott Williams & Wilkins.
  • Brouwers, J., Brewster, M. E., Augustijns, P. (2009). Supersaturating drug delivery system: the answer to solubility-limited oral bioavailability? J Pharm Sci 98:2549–2572.
  • Drummond, D. C., Meyer, O., Hong, K., et al. (1999). Optimizing liposomes for delivery of chemotherapeutic agents to solid tumors. Pharmacol Rev 5:691–743.
  • Frantzen, C. B., Ingebrigtsen, L., Skar, M., Brandl, M. (2003). Assessing the accuracy of routine photon correlation spectroscopy analysis of heterogeneous size distributions. AAPS PharmSciTech [online]. Available at: http://www.springerlink.com/content/a7v263809141313x. Last date of access: August 10th 2010.
  • Gabizon, A., Papahadjopoulos, D. (1988). Liposome formulations with prolonged circulation time in blood and enhanced uptake by tumors. Proc Natl Acad Sci U S A 85:6949–6953.
  • Grohganz, H., Ziroli, V., Massing, U., Brandl, M. (2003). Quantification of various phosphatidylcholines in liposomes by enzymatic assay. AAPS PharmSciTech [online]. Available at: http://www.aapspharmscitech.org/articles/pt0404/pt040463/pt040463. Last date of access: August 2010.
  • Gulati, M., Grover, M., Singh, S., Singh, M. (1997). Lipophilic drug derivatives in liposomes. Int J Pharm 165:129–168.
  • Hradil, P., Hlaváč J., Soural M., et al (2009). 3-Hydroxy-2-phenyl-4(1H)-quinolinones as promising biologically active compounds. Mini Rev Med Chem, 9: 696–702.
  • Sætern, A. M., Flaten, G. E., Brandl, M. (2004). A method to determine the incorporation capacity of camptothecin in liposomes. AAPS PharmSciTech [online]. Available at: http://www.springerlink.com/content/c83715622732v278/fulltext. Last date of access: August 2010.
  • Schwendener, R., Schott, H. (2010). Liposome formulations of hydrophobic drugs. Meth Mol Biol 605:129–138.
  • Soural, M., Hlavác, J., Hradil, P., et al. (2006). 3-hydroxy-2-phenyl-4(1H)-quinolinones as promising biologically active compounds. Eur J Med Chem 41:467–474.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.