391
Views
20
CrossRef citations to date
0
Altmetric
Original Articles

Development of egg PC/cholesterol/α-tocopherol liposomes with ionic gradients to deliver ropivacaine

, , , , , & show all
Pages 1-10 | Received 24 Oct 2014, Accepted 20 Feb 2015, Published online: 26 Mar 2015

References

  • Barbosa RM, da Silva CMG, Bella TS, et al. (2013a). Cytotoxicity of solid lipid nanoparticles and nanostructured lipid carriers containing the local anesthetic dibucaine designed for topical application. J Phys Conf Ser 429:1–8
  • Barbosa RM, Klassen A, Marcato PD, et al. (2013b). Validation of an HPLC method for the determination of dibucaine encapsulated in solid lipid nanoparticles and nanostructured lipid carriers. Lat Am J Pharm 32:1362–9
  • Barenholz Y, Haran G. (1993). Method of amphiphatic drug loading in liposomes by pH gradient. US Patent # 5, 192, 549
  • Barenholz Y, Haran G. (1994). Method of amphiphatic drug loading in liposomes by ammonium ion gradient. US Patent # 5, 316, 771
  • Boogaerts JG, Lafond ND, Declercq AG, et al. (1994). Epidural administration of liposome-associated bupivacaine for the management of postsurgical pain: a first study. J Clin Anesth 6:315–20
  • Boogaerts J, Lafont N, Donnay M, et al. (1995). Motor blockade and absence of local nerve toxicity induced by liposomal bupivacaine injected into the brachial plexus of rabbits. Acta Anaesthesiol Belg 46:19–24
  • Catterall W, Mackie K. (2011). Local anesthetics. In: Goodman LS, Gilman AG, eds. The pharmacological basis of therapeutics. New York: McGraw-Hill, 1732–4
  • Celano M, Calvagno MG, Bullota S, et al. (2004). Cytotoxic effects of gemcitabine-loaded liposomes in human anaplastic thyroid carcinoma cells. BMC Cancer 4:1–5
  • Cereda CM, Brunetto GB, Araújo DR, de Paula E. (2006). Liposomal formulations of prilocaine, lidocaine and mepivacaine prolong analgesia duration. Can J Anaesth 53:1092–7
  • Cereda CM, de Araújo DR, Brunetto GB, de Paula E. (2004). Liposomal prilocaine: preparation, characterization and in vivo evaluation. J Pharm Pharm Sci 7:235–40
  • Cereda CM, Franz-Montan M, Silva CMG, et al. (2013). Transdermal delivery of butamben from elastic and conventional liposomes. J Liposome Res 23:228–34
  • Cern A, Golbraikh A, Sedykh A, et al. (2012). Quantitative structure–property relationship modeling of remote liposome loading of drugs. J Control Release 160:147–57
  • Chen PS, Toribara TY Jr, Warner H. (1956). Microdetermination of phosphorus. Anal Chem 28:1756–8
  • Cohen R, Kanaan H, Grant GJ, Barenholz Y. (2012). Prolonged analgesia from bupisome and bupigel formulations: from design and fabrication to improved stability. J Control Release 160:346–52
  • Davidson EM, Barenholz Y, Cohen R, et al. (2010). High-dose bupivacaine remotely loaded into multivesicular liposomes demonstrates slow drug release without systemic toxic plasma concentrations after subcutaneous administration in humans. Anesth Analg 110:1018–23
  • de Araújo DR, Cereda CM, Brunetto GB, et al. (2004). Encapsulation of mepivacaine prolongs the analgesia provided by sciatic nerve blockade in mice. Can J Anaesth 51:566–72
  • de Araújo DR, Cereda CM, Brunetto GB, et al. (2008). Pharmacological and local toxicity studies of a liposomal formulation for the novel local anaesthetic ropivacaine. J Pharm Pharmacol 60:1449–57
  • de Paula E, Cereda CM, Fraceto LF, et al. (2012). Micro and nanosystems for delivering local anesthetics. Expert Opin Drug Deliv 9:1505–24
  • de Paula E, Cereda CM, Tofoli GR, et al. (2010). Drug delivery systems for local anesthetics. Recent Pat Drug Deliv Formul 4:23–34
  • de Paula E, Schreier S. (1995). Use of a novel method for determination of partition coefficients to compare the effect of local anesthetics on membrane structure. Biochim Biophys Acta 1240:25–33
  • Franz-Montan M, Baroni D, Brunetto G, et al. (2015). Liposomal lidocaine gel for topical use at the oral mucosa: characterization, in vitro assays and in vivo anesthetic efficacy in humans. J Liposome Res 25:11–19
  • Franz-Montan M, Cereda CM, Gaspari A, et al. (2013). Liposomal-benzocaine gel formulation: correlation between in vitro assays and in vivo topical anesthesia in volunteers. J Liposome Res 23:54–60
  • Franz-Montan M, Silva ALR, Cogo K, et al. (2007). Liposome-encapsulated ropivacaine for topical anesthesia in human oral mucosa. Anesth Analg 104:1528–31
  • Gesztes A, Mezei M. (1988). Topical anesthesia of the skin by liposome-encapsulated tetracaine. Anesth Analg 67:1079–81
  • Grant SA. (2002). The holy grail: long-acting local anesthetics and liposomes. Best Pract Res Clin Anesthesiol 16:345–52
  • Grant GJ, Bansinath M. (2001). Liposomal delivery systems for local anesthetics. Reg Anesth Pain Med 26:61–3
  • Grant GJ, Barenholtz Y, Bolotin E, et al. (2004). A novel liposomal bupivacaine formulation to produce ultralong-acting analgesia. Anesthesiology 101:133–7
  • Grant GJ, Barenholtz Y, Piskoun B, et al. (2001). DRV liposomal bupivacaine: preparation, characterization, and in vivo evaluation in mice. Pharm Res 18:336–43
  • Grant GJ, Lax J, Susser L, et al. (1997). Wound infiltration with liposomal bupivacaine prolongs analgesia in rats. Acta Anaesthesiol Scand 41:204–7
  • Grant GJ, Vermeulen K, Langerman L, et al. (1994). Prolonged analgesia with liposomal bupivacaine in a mouse model. Reg Anesth 19:264–9
  • Griffith OH, Jost OP. (1976). Spin labels in biological membranes. In: Berliner LJ, ed. Spin labeling: theory and applications. New York: Academic Press, 454–523
  • Grillo R, Melo NFS, de Araújo DR, et al. (2009). Validation of an HPLC method for quantitative determination of benzocaine in PHBV microparticles and PLA-nanoparticles. Lat Am J Pharm 28:393–9
  • Gubernator J. (2011). Active methods of drug loading into liposomes: recent strategies for stable drug entrapment and increased in vivo activity. Expert Opin Drug Deliv 8:565–80
  • ICH. (2005). Validation of analytical procedures: text and methodology (Q2R1). International Conference on Harmonization; Nov 2005; Geneva
  • Jonsson JA, Andersson M, Melander C, et al. (2000). Automated liquid membrane extraction for high-performance liquid chromatography of ropivacaine metabolites in urine. J Chromatogr A 870:151–7
  • Lafont ND, Legros FJ, Boogaerts JG. (1996). Use of liposome-associated bupivacaine in a cancer pain syndrome. Anaesthesia 51:578–9
  • Lagan G, McLure HA. (2004). Review of local anaesthetic agents. Curr Anaesth Crit Care 15:247–54
  • Mohanraj VJ, Chen Y. (2006). Nanoparticles – a review. Trop J Pharm Res 5:561–73
  • Mowat JJ, Mok MJ, MacLeod BA, Madden TD. (1996). Liposomal bupivacaine extended duration nerve blockade using large unilamellar vesicles that exhibit a proton gradient. Anesthesiology 85:635–43
  • Pinto LMA, Yokaichiya DK, Fraceto LF, de Paula E. (2000). Interaction of benzocaine with biomembranes. Biophys Chem 87:213–23
  • Samad A, Sultana Y, Aqil M. (2007). Liposomal drug delivery systems: an update review. Curr Drug Deliv 4:297–305
  • Schreier S, Polnaszek CF, Smith IC. (1978). Spin labels in membranes. Problems in practice. Biochim Biophys Acta 515:395–436
  • Strichartz GR, Covino BG. (1990). Local anesthetics. In: Miller RD, ed. Anesthesia. New York: Churchill Livingstone, 437–70
  • Torchilin VP. (2005). Recent advances with liposomes as pharmaceutical carriers. Nat Rev Drug Discov 4:145–60
  • Torchilin VP. (2012). Liposomes in drug delivery. Adv Deliv Sci Technol 4:289–328
  • Tu S, McGinnis T, Krugner-Higby L, Heath TD. (2010). A mathematical relationship for hydromorphone loading into liposomes with trans-membrane ammonium sulfate gradients. J Pharm Sci 99:2672–80
  • Warren RC. (1987). Physics and architecture of cell membranes. Bristol and Philadelphia (PA): Adam-Hilger
  • Weiniger CF, Golovanevski M, Sokolsky-Papkov M, Domb AJ. (2010). Review of prolonged local anesthetic action. Exp Opin Drug Deliv 7:737–52
  • Wiles MD, Nathanson MH. (2010). Local anaesthetics and adjuvants – future developments. Anaesthesia 65:22–37
  • Yu HY, Li SD, Sun P. (2002). Kinetic and dynamic studies of liposomal bupivacaine and bupivacaine solution after subcutaneous injection in rats. J Pharm Pharmacol 54:1221–7
  • Zuo M, Duan GL, Ge ZG. (2004). Simultaneous determination of ropivacaine and antipyrine by high performance liquid chromatography and its application to the in vitro transplacental study. Biomed Chromatogr 18:752–5

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.