References
- Atchison, R. E., Gosling, J., Monteclaro, F. S., Franci, C., Digilio, L., Charo, I. F., and Goldsmith, M. 1996. Science 274:1924–1926.
- Baba, M., Nishimura, O., Kanzaki, N., Okamoto, M., Sawada, H., Iizawa, Y., Shiraishi, M., Aramaki, Y., Okonogi, K., Ogawa, Y.,Meguro, K., and Fujino, M. 1999. Proc. Natl. Acad. Sci. USA 96:5698–5703.
- Bieniassz, P. D., Fridell, R. A., Aramori, I., Ferguson, S. S., Caron, M. G., and Cullen, B. R. 1997. EMBO J. 16:2599–2609.
- Blanpain, C.,Vanderwinden, J.-M., Cihak, J.,Wittamer,V., Le Poul, E., Issafras, H., Stangassinger, M., Vassart, G., Marullo, S., Schlondorff, D., Parmentier, M., and Mack, M. 2002. Mol. Biol. Cell 13:723–737.
- Bursavich, M. G., and Rich, D. H. 2001. J. Med. Chem. 45:541–558.
- Christopolous, A., and Kenakin, T. P. 2002. Pharmacol. Rev. 54:323–374.
- Doms, R. W., and Peiper, S. C. 1997. Virol. 235:179–190.
- Doranz, B. J., Lu, Z.-H., Rucker, J., Zhang, T.-Y., Sharron, M., Cen,Y.-H.,Wang, Z.-X., Guo, H.-H., Du, J.-D., Accavitti, M. A., Doms, R. W., and Peiper, S. C. 1997. J. Virol. 71:6305–6314.
- Ehlert, F. J. 1988. Mol. Pharmacol. 33:187–194.
- Fawazi, A. B., MacDonald, D., Benbow, L. L., Smith-Torhan, A., Zhang, H., Weig, B. C., Ho, G., Tulshian, D., Linder, M. E., Graziano, M. P. 2001. Mol. Pharmacol. 59:30–37.
- Finke, G., Oates, B., Mills, S. G., MacCoss, M., Malkowitz L., Springer, M. S., Gould, S. L., DeMartino, A., Carella, A., Carver, G., et al. 2001. Bioorg. Med. Chem. Lett. 11:2475–2479.
- Frauenfelder, H., Parak, F., and Young, R. D. 1988. Ann. Rev. Biophys. Biophys. Chem. 17:451–479.
- Frauenfelder, H., Sligar, S. G., andWolynes, P. G. 1991. Science 254:1598–1603.
- Ghanouni, P., Grycynski, Z., Steenhuis, J. J., Lee,T.W., Farrens, D. L., Lakowicz, J. R., and Kobilka, B. K. 2001. J. Biol. Chem. 276: 24433–24436.
- Hall, D. A. 2000. Mol. Pharmacol. 58:1412–1423.
- Hejnova, L., Tucek, S., and El-Fakahany, E. E. 1995. Eur. J. Pharmacol. 291: 427–430.
- Heveker, N., Montes, M., Germeroth, L., Amara, A., Trautmann, A., Alizon, M., and Schneider-Mergener, J. 1998. Current Biology 8:369–376.
- Hilser, V. J., and Freire, E. 1996. J Mol. Biol. 262:756–772.
- Hilser, V. J., and Freire, E. 1997. Protein Struct. Funct. Genet. 27:171–183.
- Hilser, V. J., Townsend, B. D., and Freire, E. 1997. Biophys. Chem. 64:69–79.
- Hilser, V. J., Dowdy, D., Oas, T. G., and Freire, E. 1998. Proc. Natl. Acad. Sci. USA 95:9903–9908.
- Jakubic, J., Bacakova, L., Lisa, V., El-Fakahany, E. E., and Tucek, S. 1996. Proc. Natl. Acad. Sci USA 93:8705–8709.
- Jakubic, J., Bacakova, L., Lisa, V., El-Fakahany, E. E., and Tucek, S. 1997. Mol. Pharmacol. 52:172–179.
- Kazmierski,W. M., Boone, L., Lawrence,W.,Watson, C., andKenakin, T. 2002. Current Drug Targets-Infectious Disorders 2:265–278.
- Kenakin, T. P. 2002a. Ann. Rev. Pharmacol. Toxicol. 42:349–379.
- Kenakin, T. P. 2002b. Nature Reviews (Drug Discovery) 1:103–109.
- Kenakin, T. P. 2003. Trends Pharmacol. Sci. 24:346–354.
- Kenakin, T. P., and Onaran, O. 2002. Trends Pharmacol. Sci. 23:275–280.
- Kumar, S., Ma, B., Tsai, C. J.,Wolfson, H., and Nussinov, R. 1999. Cell Biochem. Biophys. 31: 141–164.
- Kwong, P. D.,Wyatt, R., Robinson, J., Sweet, R.W., Sodroski, J., and Hendricks, W. A. 1998. Nature 393: 648–659.
- Lee, B., Sharron, M., Blanpain, C., Doranz, B. J., Vakili, J., Setoh, P., Berg, E., Liu, G., Guy, H. R., Durell, S. R., Parmentier, M., Chang, C. N., Price, K., Tsang, M., and Doms, R. W. 1999a. J. Biol. Chem. 274:9617–9626.
- Litschig, S., Gasparini, F., Rueegg, D. F., Stoehr, N., Flor, P. J., Vranesic, I., Prézeau, L., Pin, J. P., Thomsen, C., and Kuhn, R. 1999. Mol. Pharmacol. 55:453–461.
- Ma, B., Kumar, S., Tsai, C. J., and Nussinov, R. 1999. Protein Eng. 12:713–720.
- Moore, J. P., Trkola, A., and Dragic, T. 1997. Curr. Opin. Immunol. 9:551–562.
- Nagasaw, T., Hirota, S., Tachibana, K., Takakura, N., Nishikawa, S., Kitamura, Y., Yoshida, N., Kikutani, H., and Kishimoto, T. 1996. Nature 382: 635–638.
- Onaran, H. O., and Costa, T. 1997. Ann. N.Y. Acad. Sci. 812:98–115.
- Onaran, H. O., Scheer, A., Cotecchia, S., and Costa, T. 2000. In The Pharmacology of Functional, Biochemical, and Recombinant Systems Handbook of Experimental Pharmacology, vol. 148. Eds. T. P. Kenakin and J. A. Angus. Germany: Springer, Heidelberg. pp. 217–80.
- Picard, L., Simmons, G., Power, C. A., Meyer, A., Wiess, R. A., and Clapham, P. R. 1997. J. Virol. 71:5003–5011.
- Rees, S., Morrow, D., and Kenakin, T. 2002. Receptors and Channels 8:261– 268.
- Rizzuto, C. D., Wyatt, R., Hernández-Ramos, N., Sun, Y., Kwong, P. D., Hendrickson, W. A., and Sodroski, J. 1998. Science 280:1949–1953.
- Roettger, B. F., Ghanekar, D., Rao, R., Toledo, C., Yingling, J., Pinon, D., and Miller, L. J. 1997. Mol. Pharmacol. 51:357–362.
- Ross, T., Bieniasz, P. D., and Cullen, B. R. 1999. Adv. Virus Res. 52:233–267.
- Rucker, J., Edinger, A. L., Sharron, M., Samson, M., Lee, B., Berson, J. F. Y., Collman, R. G., Doranz, B. J., Domes, R. W., and Parmentier, M. 1997. J. Virol. 71:8999–9007.
- Sachpatzidis, A., Benton, B. K., Manfredis, J. P., Wang, H., Hamilton, A., Dohlman, H. G., and Lolis, E. 2003. J. Biol. Chem. 278:896–907.
- Smyth, R. J., Yi, Y., Singh, A., and Collman, R. G. 1998. J. Virol. 72:4478–4484.
- Stephenson, R. P. 1956. Br. J. Pharmacol. 11:379–393.
- Straub, F. B. 1964. Adv. Enzymology 26:89–114.
- Strizki, J. M., Xu, S., Wagner, N. E., Wojcik, L., Jia Liu, J., Hou, Y., Endres, M., Palani, A., Shapiro, S., Clader, J. W., Greenlee, W. J., Tagat, J. R., et al. 2001. Proc. Natl. Acad. Sci. USA. 98:12718–12723.
- Tachibana, K., Hirota, S., Iizasa, H., Yoshida, H., Kawabata, K., Kataoka, Y., Kitamura, Y., Matsushima, K., Yoshida, N., Nishikawa, S., Kishimoto, T., and Nagasawa, T. 1998. Nature 393:591–594.
- Tsai, C. J., Kumar, S., Ma, B., and Nussinov, R. 1999. Protein Sci. 8:1181–1190.
- Tucek, S., and Proska, J. 1995. Trends Pharmacol. Sci. 16:205–212.
- Venter, J. C., Adams, M. D., Myers, E. M., Li, P. W., Mural, R. J., Sutton, G. G., Smith, H. O., Yandell, M., Evans, C. A., Holt, R. A., et al. 2001. Science 291:1304–1351.
- Zou, Y. R., Kottmann, A. H., Kuroda, M., Taniuchi, I., and Littman, D. R. 1998. Nature 393:595–599.