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Original Article

Preparation, Characterisation and Biodistribution of 99mTc-labeled Liposome Encapsulated Cyclosporine

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Pages 187-196 | Received 16 Jun 2003, Published online: 21 Jun 2010

References

  • Adler, M., Jill, P.E., Williams, A., (1997) “Pharmaceutical formulation and process”, U.S.Patent. # 5,688,525.
  • Aoki, H., Sun, C., Fuji, K. and Miyajima, K. (1995) “Disposition kinetics of liposomes modified with synthetic aminoglycolipids in rats”, Int. J. Pharm. 115, 183–191.
  • Aoki, H., Tottori, T., Sakurai, F., Fuji, K. and Miyajima, K. (1997) “Effect of positive charge density on the liposomal surface on the disposition kinetics of liposomes in rats”, Int. J. Pharm. 156, 163–174.
  • Borel, J.F. (1988) “Immunosuppression: building on Sandimmune (Cyclosporine)”, Transplant. Proc. 20, 149–153.
  • Caride, V.J. (1990) “Technical and biological considerations on the use of radiolabeled liposomes for diagnostic imaging”, Nucl. Med. Biol. 17, 35–39.
  • Crowe, J.H., Crowe, L.M. and Carpenter, J.K. (1988) “Interactions of sugars with membranes”, Biochim. Biophys. Acta 947, 367–384.
  • Damen, J., Regts, J. and Scherphof, G. (1981) “Transfer and exchange of phospholipids between small unilamellar liposomes and rat plasma high density lipoproteins. Dependence on cholesterol content and phospholipid composition”, Biochim. Biophys. Acta 665, 538–542.
  • Dowling, R.D., Zenati, M. and Burckart, G.J. (1990) “Aerosolized cyclosporine as single agent immunotherapy in canine lung allografts”, Surgery 108, 198–199.
  • Gregoriadis, G.N. (1976) “The carrier potential of liposomes in biology and medicine”, N. Engl. J. Med. 295, 704–705.
  • Gregoriadis, G. and Neerunjun, D.E. (1974) “Control of the rate of hepatic uptake and catabolism of liposome-entrapped proteins injected into rats: possible therapeutic applications”, Eur. J. Biochem. 47, 179–185.
  • Gregoriadis, G., Kirby, C. and Senior, J. (1983) “Optimization of liposomal behaviour in vivo”, Biol. Cell. 47, 11–18.
  • Hardy, J.G., Kellway, I.W. and Rogers, H. (1980) “The distribution and fate of I-131 labeled liposomes”, J. Pharm. Pharmacol. 32, 309–313.
  • Kao, Y.J. and Juliano, R.L. (1981) “Interactions of liposomes with reticuloendothelial system: effects of RE-blockade on the clearance of large unilamellar vesicles”, Biochim. Biophys. Acta 677, 453–461.
  • Kirby, C., Clarke, J. and Gregoriadis, G. (1980) “Effect of the cholesterol content of small unilamellar liposomes on their stability in vivo and in vitro”, Biochem. J. 186, 591–592.
  • Klibanov, A.L., Maruyama, K., Beckerleg, A.M., Torchilin, V.P. and Huang, L. (1991) “Activity of amphipathic poly (ethylene glycol) 5000 to prolong the circulation time of liposomes depends on the liposome size and is unfavourable for immunoliposome binding to target”, Biochim. Biophys. Acta 1062, 142–148.
  • Lopez-Berestein, G., Hopfer, R.L., Mehta, R., Mehta, R., Hersh, E.M. and Juliano, R.L. (1984) “Liposome encapsulated amphotericin-B for treatment of disseminated candidiasis in neutropenic mice”, J. Infect. Dis. 150, 278–283.
  • Luke, D.R., Kasiske, B.L., Matzke, G.R. and Keane, W.F. (1987) “Effects of cyclosporine on the isolated perfused rat kidney”, Transplantation 43, 795–799.
  • Morgan, J.R., Williams, K.E. and Davis, R.I. (1981) “Localisation of experimental staphylococcal abscesses by 99mTc-labeled liposomes”, J. Med. Micro. 14, 213–217.
  • Morgan, J.R., Williams, L.A. and Howard, C.B. (1985) “Technetium- labeled liposome imaging for deep-seated infection”, Br. J. Radiol. 58, 35–38.
  • Nabar, S.J. and Nadkarni, G.D. (1998) “Effect of size and charge of liposomes on biodistribution of encapsulated 99mTc-DTPa in rats”, Ind. J. Pharmacol. 30, 199–202.
  • Nacucchio, M.C., Gatto Bellora, M.J., Sordelli, D.O. and D’Aquino, M. (1985) “Enhanced liposome mediated activity of piperacillin against staphylococci”, Antimicrob. Agents Chemother. 27, 137–139.
  • Ogihara, I. and Kojimi, S. (1989) “Cholesterol enhances the delivery of liposome encapsulated gallium-67 to tumors”, Eur. J. Nucl. Med. 15, 612–619.
  • Ogihara, I., Kojimi, S. and Jay, M. (1986) “Differential uptake of gallium- 67 labeled liposomes between tumors and inflammatory lesions in rats”, J. Nucl. Med. 27, 1300–1302.
  • Ostro, M.J. and Cullis, P.R. (1989) “Use of liposomes as injectable drug delivery systems”, Am. J. Hosp. Pharm. 46, 1576–1577.
  • Perico, N. and Remuzzi, G. (1997) “Prevention of transplant rejection: current treatment guidelines and future developments”, Drugs 54, 533–570.
  • Puschett, J.B., Greenbery, A., Holley, J. and McCauley, J. (1990) “The spectrum of cyclosporine nephrotoxicity”, Am. J. Nephrol. 10, 296–299.
  • Richardson, V.J., Jeyasingh, K. and Jewkes, R.F. (1977) “Properties of [99mTc] technetium labeled liposomes in normal and tumor bearing rats”, Biochem. Soc. Trans. 5, 290–291.
  • Richardson, V.J., Jeyasingh, K., Jewkes, R.F., Ryman, B.E. and Tattersall, M.H. (1978) “Possible tumor localization of 99m Technetium labeled liposomes: effects of lipid composition, charge, and liposome size”, J. Nucl. Med. 19, 1049–1054.
  • Rudolph, A.S. (1988) “The freeze-dried preservation of liposome encapsulated hemoglobin: a potential blood substitute”, Cryobiology 25, 277–284.
  • Saha, G.B. (1993) “Methods of Radiolabeling”, In: Saha, G.B., ed, Physics and Radiobiology of Nuclear Medicine (Springer, New York), pp 100–106.
  • Stuhne-Sekalec, L. and Stanaav, N.Z. (1991) “Liposomes as carriers of Cyclosporine A”, J. Microencapsul. 18, 441–446.
  • Theobald, A.E. (1990) Chapter 7, In: Sampson, C.B., ed, Textbook of Radiopharmacy: Theory and Practice (Gordon and Breach, New York), pp 127–129.
  • Thiel, G., Mihatsch, M.J., Stahl, R.A., Hermle, M. and Brunner, F.P. (1986) “Cyclosporine nephrotoxicity in Goldblatt renovascular hypertension in rats”, Clin. Nephrol. 25, S199–S204.
  • Treat, J., Greenspan, A. and Forst, D. (1990) “Antitumor activity of liposome encapsulated doxorubicin in advanced breast cancer: phase II study”, J. Natl Cancer Inst. 82, 1706–1710.
  • Vadiei, K., Perez-Soler, R., Lopez-Berestein, G. and Luke, D.R. (1989) “Pharmacokinetic and pharmacodynamic evaluation of liposomal cyclosporine”, Int. J. Pharm. 57, 125–131.
  • Venkataramanan, R., Habucky, K., Burckart, G.J. and Ptachcinski, R.J. (1989) “Clinical pharmacokinetics in organ transplant patients”, Clin. Pharm. 16, 134–161.
  • Wu, M.S., Robbins, J.C., Ponpipom, M.M. and Shen, T.V. (1981) “Modified in vivo behaviour of liposomes containing synthetic glycolipids”, Biochim. Biophys. Acta 674, 19–29.

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