1,137
Views
8
CrossRef citations to date
0
Altmetric
Research Article

Predictable pulsatile release of tramadol hydrochloride for chronotherapeutics of arthritis

, , , &
Pages 273-281 | Received 29 Jul 2009, Accepted 16 Feb 2010, Published online: 07 Jun 2010

References

  • Ahrabi, S.F., Madsen, G., Dyrstad, K., Sande, S.A., Graffner, C. (2000). Development of pectin matrix tablets for colonic delivery of model drug ropivacaine. Eur J Pharm Sci. 10:43–52.
  • Amsden, T., Cheng, L. (1995). A generic protein delivery system based on osmotically rupturable monoliths. J Contr Rel. 33:99–105.
  • Bajpai, S.K., Bajpai, M., Dengree, R. (2003). Chemically treated hard gelatin capsules for colon-targeted drug delivery: a novel approach. J Appl Polym Sci. 89:2277–82.
  • Bussemer, T., Otto, I., Bodmeier, R. (2001). Pulsatile drug-delivery systems. Crit Rev The Drug Carrier Syst. 18:433–58.
  • Cheng, G., An, F., Zou, M., Sun, J., Hao, X., He, Y. (2004). Time and pH-dependent colon-specific drug delivery for orally administered diclofenac sodium and 5-aminosalicylic acid. World J Gastroenterol. 10:1769–74.
  • Chourasia, M.K., Jain, S.K. (2004). Potential of Guar Gum microspheres for target specific drug release to colon. J Drug Target. 12:435–42.
  • Conte, U., Magg, L., Torre, M.L., Giunchedi, P., La Manna, A. (1993). Press-coated tablets for time-programmed release of drugs. Biomaterials. 14:1017–23.
  • Davis, S.S., Hardy, J.G., Fara, J.W. (1986). Transit of pharmaceutical dosage forms through the small intestine. Gut. 27:886–92.
  • Evans, D.F., Pye, G., Bramley, R., Clark, A.G., Dyson, T.J., Hardcastle, J.D. (1998). Measurement of gastrointestinal pH profiles in normal ambulant human subjects. Gut. 29:1035–41.
  • Fernandez-Hervas, M.J., Fell, J.T. (1998). Pectin:chitosan mixtures as coatings for colon-specific drug delivery: an in vitro evaluation. Int J Pharm. 169:115–9.
  • Fukui, E., Miyamura, N., Uemura, K., Kobayash, M. (2000). Preparation of enteric coated timed-release press-coated tablets and evaluation of their function by in vitro and in vivo tests for colon targeting. Int J Pharm. 204:7–15.
  • Gang, C., Feng, A., Mei-Juan, Z., Jin, S., Xiu-Hua, H., Yun-Xia, H. (2004). Time and pH-dependent colon- specific drug delivery for orally administred diclofenac sodium and 5- amino salicylic acid. Worid J Gastroenterol. 10:1769–74.
  • Gazzaniga, A., Iamartino, P., Maffione, G., Sangalli, M.E. (1994a). Oral delayed-release system for colonic specific delivery. Int J Pharm. 108:77–83.
  • Gazzaniga, A., Sangalli, M.E., Giordano, F. (1994b). Oral chronotopic drug delivery systems: achievement of time and/or site specificity. Eur J Pharm Biopharm. 40:246–50.
  • Gonzalez-Rodriguez, M.L., Maestrelli, F., Mura, P., Rabasco, A.M. (2003). In vitro release of sodium diclofenac from a central core matrix tablet aimed for colonic drug delivery. Eur J Pharm Sci. 20:125–31.
  • Halsas, M., Hietala, J., Veski, P., Jurjenson, H., Marvola, M. (1999). Morning versus evening dosing of ibuprofen using conventional and time controlled release formulations. Int J Pharm. 189:179–85.
  • Halsas, M., Penttinen, T., Veski, P., Jurjenson, H., Marvola, M. (2001). Time controlled release pseudoephedrine tablets: bioavailability and in vitro/in vivo correlations. Pharmazie. 56:718–23.
  • Kinget, R., Kalala, W., Vervoort, L., Van den Mooter, G. (1998). Colonic drug targeting. J Drug Target. 6:129–49.
  • Kopecek, J.P., Kopeckova, H., Brondsted, R., Rathi, B., Rihova Yeh, P.-Y., Ikesue, K. (1992). Polymers for colon specific drug delivery. J Contr Rel. 19:121–30.
  • Kowanko, I.C., Pownall, R., Knapp, M.S., Swannel, E.J., Mahoney, P.G. (1981). Circadian variations in the signs and symptoms of rheumatoid arthritis and in the therapeutic effectiveness of flurbiprofen at different times of the day. Br J Clin Pharmacol. 11:477–84.
  • Krishnaiah, Y.S.R., Satyanarayana, S., Rama Prasad, Y.V. (1999). Studies of Guar Gum compression-coated 5-aminosalicylic acid tablets for colon-specific drug delivery. Drug Dev Ind Pharm. 25:651–7.
  • Krishnaiah, Y.S.R., Satyanarayana, S., Rama Prasad, Y.V., Narasimha Rao, S. (1998). Evaluation of guar gum as a compression coat for drug targeting to colon, Int J Pharm. 71:137–46.
  • Krishnaiah, Y.S.R., Satyanarayana, V., Kumar, B.D., Karthikeyan, R.S. (2002). In vitro drug release studies on guar gum-based colon targeted oral drug delivery systems of 5-fluorouracil. Eur J Pharm Sci. 16:185–92.
  • Maggi, L., Conte, U., Gurni, R. (1999). Delivery device for the release of active ingredient in subsequent time. Proceedings of the International Controlled Release Bioactive Materials, Boston, MA, Vol. 26.
  • Mastiholimath, V.S., Dandagi, P.M., Jain, S.S., Gadad, A.P., Kulkarni, A.R. (2007). Time and pH dependent colon specific, pulsatile delivery of theophylline for noctural asthma. Int J Pharm. 328:49–56.
  • Morita, R., Honda, R., Takahashi, Y. (2000). Development of oral controlled release preparations, a PVP swelling controlled release system (SCRS): I. Design of SCRS and its release controlling factor. J Contr Rel. 63:297–304.
  • Nykanen, P., Lempaa, S., Aaltonen, M.L., Jurjenson, H., Veski, P., Marvola, M. (2001). Citric acid as excipient in multiple-unit enteric-coated tablets for targeting drugs on the colon. Int J Pharm. 229:155–62.
  • Obaidat, A.A., Obaidat, R.M. (2001). Controlled release tramadol hydrochloride from matrices prepared using glyceryl behenate. Eur J Pharm Biopharm. 52:231–5.
  • Otsuka, M., Matsuda, Y. (1994). Controlled drug release of highly water-soluble pentoxifylline from time-imit disintegration type wax matrix tablets. Pharm Res. 11:351–4.
  • Pozzi, F., Furlani, P., Gazzaniga, A. (1994). The TIME CLOCK system: a new oral dosage form for fast and complete release of drug after a predetermined lag time. J Contr Rel. 31:99–108.
  • Sangalli, M.E., Maroni, A., Zema, L., Busetti, C., Giordano, F., Gazzaniga, A. (2001). In vitro and in vivo evaluation of an oral system for time and/or site-specific drug delivery. J Contr Rel. 73:103–10.
  • Sawada, T., Kondo, H., Nakashima, H., Sako, K., Hayashi, M. (2004). Time-release compression-coated core tablet containing nifedipine for chronopharmacotherapy. Int J Pharm. 280:103–11.
  • Schorn, D., Seymour, M.A. (1981). Indomethacin or sulindac in rheumatoid arthritis at night. S Afr Med J. 59:913–4.
  • Scott, J.T. (1960). Morning stiffness in rheumatoid arthritis. Ann Rheum Dis. 19:361–8.
  • Takeuchi, H., Yasuji, T., Yamamoto, H., Kawashima, Y. (2000). Spray-dried lactose composite particles containing an ion complex of alginate-chitosan for designing a dry-coated tablet having a time-controlled releasing function. Pharm Res. 17:94–9.
  • Tekade, A.R., Gattani, S.G. (2009). Development and evaluation of pulsatile drug delivery system using novel polymer. Pharm Dev Tech. 14:380–7.
  • Tiwari, S.B., Murthy, T.K., Pai, M.R., Mehta, P.R., Chowdaty, P.B. (2003). Controlled release formulation of Tramadol hydrochloride using hydrophilic and hydrophobic matrix system. AAPS Pharm Sci Tech. 4:1–6.
  • Turkoglu, M., Takka, S., Baran, H., Sakr, A. (1999). Pectin hydroxyl propyl methyl cellulose drug delivery system for colon targeting. Pharm Pharmacol. 51:154.
  • Turkoglu, M., Ugurlu, T. (2002). In vitro evaluation of pectin–HPMC compression coated 5-aminosalicylic acid tablets for colonic delivery. Eur J Pharm Biopharm. 53:65–73.
  • Ugurlu, T., Turkoglu, M., Gurer, U.S., Akarsu, B.G. (2007). Colonic delivery of compression coated nisin tablets using pectin/ HPMC polymer mixture. Eur J Pharm Biopharm. 67:202–10.
  • Varshosaz, J., Tavakoli, N., Kheirolahi1, F. (2006). Use of hydrophilic natural gums in formulation of sustained-release matrix tablets of tramadol hydrochloride. AAPS Pharm Sci Tech. 7:E1–7.
  • White, W.B., Black, H.R., Weber, M.A., Elliott, W.J., Bryzinski, B., Fakouhi, T.D. (1998). Comparison of effects of controlled onset extended release verapamil at bedtime and nifedipine gastrointestinal therapeutic system on arising on early morning blood pressure, heart rate, and the heart rate-blood pressure product. Am J Cardiol. 81:424–31.
  • Wilding, I.R., Davis, S.S., Pozzi, F. (1994). Enteric coated timed release system for colonic targeting. Int J Pharm. 111:99–102.
  • Zahirul Khan, M.I., Zeljko, P., Nevenka, K. (1999). A pH-dependent colon targeted oral drug delivery system using methacrylic acid copolymers I. Manipulation of drug releases using Eudragit L100-55 and Eudragit S100 combinations. J Contr Rel. 58:215–22.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.