Design and characterization of cefuroxime axetil biphasic floating minitablets

References

• Abdelkader H, Abdalla OY, Salem H. (2008). Formulation of controlled-release Baclofen matrix tablets II: influence of some hydrophobic excipients on the release rate and in vitro evaluation. AAPS Pharm Sci Tech 9:675–83
   PubMed Web of Science ®Google Scholar
• Abdul S, Chandeswar AV, Jaiswal SB. (2010). A flexible technology for modified-release drugs: multiple-unit pellet system (MUPS). J Controlled Release 147:2–16
   PubMed Web of Science ®Google Scholar
• Bandari S, Eaga CM, Thadishetty A, Yamsani MR. (2010). Formulation and evaluation of multiple tablets as a biphasic gastroretentive floating drug delivery system for fenoverine. Acta Pharm 60:89–97
   PubMed Web of Science ®Google Scholar
• Barker SA, Yap SP, Yuen KH, et al. (2003). An investigation into the structure and bioavailability of a-tocopherol dispersion in gelucire 44/14. J Controlled Release 91:477–88
   PubMed Web of Science ®Google Scholar
• Bomma R, Veerabrahma K. (2012). Development of gastroretentive drug delivery system for cefuroxime axetil: in vitro and in vivo evaluation in human volunteers. Pharm Dev Technol 18:1230--37
   Google Scholar
• Bourne DW. (2002). Pharmacokinetics. In: Banker GS, Rhodes CT, eds. Modern pharmaceutics, 4th ed. New York: Marcel Dekker Inc, 67–92
   Google Scholar
• Chauhan B, Shimpi S, Mahadik KR, Paradkar A. (2005). Preparation and evaluation of floating risedronate sodium–gelucire 1 43/01 formulations. Drug Dev Ind Pharm 31:851–60
   PubMed Web of Science ®Google Scholar
• Dhumal RS, Rajmane ST, Dhumal ST, Pawar AP. (2006). Design and evaluation of bilayer floating tablets of cefuroxime axetil for bimodal release. J Sci Ind Res 65:812–6
   Web of Science ®Google Scholar
• Fuji Chemical Industry co. Ltd. (2008). Technical News letter, May, Available from: www.fujichemical.co.jp/english/neusilin.html [last accessed 11 Dec 2011]
   Google Scholar
• Govender S, Pillay V, Chetty DJ, et al. (2005). Optimisation and characterisation of bioadhesive controlled release tetracycline microspheres. Int J Pharm 306:24–40
   PubMed Web of Science ®Google Scholar
• Govikari KR, Mandapalli PK, Manthri R, Reddy VP. (2013). Development and in vivo evaluation of gastroretentive delivery systems for cefuroxime axetil. Saudi Pharm J 21:53–9
   Web of Science ®Google Scholar
• Hardman JG, Limbird LE. (2001). In: Goodman & Gilman’s, 10th ed. Pharmacological basis of therapeutics. McGraw Hill, 1938
   Google Scholar
• Higuchi T. (1963). Mechanism of sustained action medication. J Pharm Sci 52:1145–9
   PubMed Web of Science ®Google Scholar
• Jain SK, Gupta A. (2009). Development of gelucire 43/01 beads of metformin hydrochloride for floating delivery. AAPS Pharm Sci Tech 10:1128–36
   PubMed Web of Science ®Google Scholar
• Jain SK, Jangde M. (2009). Lectin conjugated gastro-retentive multiparticulate delivery system of clarithromycin for the effective treatment of helicobacter pylori. Mol Pharm 6:295–304
   PubMed Web of Science ®Google Scholar
• Khan CA, Rhodes CT. (1975). The concept of dissolution efficiency. J Pharm Pharmacol 27:48–9
   PubMed Web of Science ®Google Scholar
• Korsmeyer RW, Gurny R, Docler E, et al. (1983). Mechanism of solute release from porous hydrophilic polymers. Int J Pharm 15:25–35
   Web of Science ®Google Scholar
• Mahmoud EB, Gihan F, Mohamed F. (2009). Improvement of solubility and dissolution rate of indomethacin by solid dispersions in gelucire 50/13 and PEG4000. Saudi Pharm J 17:217–25
   Google Scholar
• Maurya SK, Bali V, Pathak K. (2012). Bilayered transmucosal drug delivery system of pravastatin sodium: statistical optimization, in vitro, ex vivo, in vivo and stability assessment. Drug Deliv 19:45–57
   PubMed Web of Science ®Google Scholar
• McEvoy GK. (1994). Cephalosporins: cefuroxime sodium and cefuroxime axetil. In: AHFS Drug Information. Bethesda, USA: American Society of Hospital Pharmacists, 99–108
   Google Scholar
• Meka L, Thadisetty A, Vobalaboina V, Yamsani MR. (2008). Design and evaluation of a novel matrix type multiple units as biphasic gastroretentive drug delivery systems. AAPS Pharm Sci Tech 9:1253–61
   PubMed Web of Science ®Google Scholar
• Merchant HA, Shoaib HM, Tazeen J, Yousuf RI. (2006). Once-daily tablet formulation and in vitro release evaluation of cefpodoxime using hydroxypropyl methylcellulose: a technical note. AAPS Pharm Sci Tech 7:E178–83
   Google Scholar
• Moore JW, Flanner HH. (1996). Mathematical comparison of dissolution profiles. Pharma Tech 20:64–74
   Google Scholar
• Nafiz OC, Göksel A, Hassan YAE. (2006). Determination of cefuroxime axetil in tablets and biological fluids using liquid chromatography and flow injection analysis. Anal Chim Acta 576:246–52
   PubMed Web of Science ®Google Scholar
• Patel VF, Patel NM. (2006). Intragastric floating drug delivery system of cefuroxime axetil: in vitro evaluation. AAPS Pharm Sci Tech 7:E118--E124
   Google Scholar
• Patel DM, Patel NM, Patel VF, Bhatt DA. (2007). Floating granules of ranitidine hydrochloride-gelucire 43/01: formulation optimization using factorial design. AAPS Pharm Sci Tech 8:E1–7
   PubMedGoogle Scholar
• Patra CN, Pandit HK, Singh SP, Devi MV. (2008). Applicability and comparative evaluation of wet granulation and direct compression technology to Rauwolfia serpentina root powder: a technical note. AAPS Pharm Sci Tech 9:100–4
   PubMed Web of Science ®Google Scholar
• Planinisek O, Kovacic B, Vrecer F. (2011). Carvedilol dissolution improvement by preparation of solid dispersions with porous silica. Int J Pharm 406:41–8
   PubMedGoogle Scholar
• Potluri RHK, Bandari S, Jukanti R, et al. (2011). Solubility enhancement and physicochemical characterization of carvedilol solid dispersion with gelucire 50/13. Arch Pharm Res 34:51–7
   PubMed Web of Science ®Google Scholar
• Raj KA, Yada D, Yada D, et al. (2010). Determination of cefixime trihydrate and cefuroxime axetil in bulk drug and pharmaceutical dosage forms by HPLC. Int J Chem Tech Res 2:334–6
   Google Scholar
• Rawlin EA. (2010). Bentley’s text book of pharmaceutics, 8th ed. Elsevier: Philadelphia
   Google Scholar
• Rudnic EM, Lausier JM, Chilamkurti RN, Rhodes CT. (1980). Studies of the utility of cross linked polyvinylpolypyrrolidine as a tablet disintegrant. Drug Dev Ind Pharm 6:291–309
   Web of Science ®Google Scholar
• Sanker C, Mishra C. (2003). Development and in vitro evaluations of gelatin microspheres of ketorolac tromethamine for intranasal administration. Acta Pharm 53:101–10
   PubMedGoogle Scholar
• Sheu MT, Hsia A, Ho HO. (2001). Polyglycolized saturated glycerides as carrier and enhancer for drug penetration. Chin Pharm J 53:107–18
   Google Scholar
• Shimpi S, Chauhan B, Mahadik KR, Paradkar A. (2004). Preparation and evaluation of diltiazem hydrochloride-gelucire 43/01 floating granules prepared by melt granulation. AAPS Pharm SciTech 5:51–6
   Google Scholar
• Shrivastava AR, Ursekar B, Kapadia CJ. (2009). Design, optimization, preparation and evaluation of dispersion granules of valsartan and formulation into tablets. Curr Drug Delivery 10:28–37
   Google Scholar
• Sommers DK, Van WM, Moncrieff J, Schoeman HS. (1984). Influence of food and reduced gastric acidity on the bioavailability of bacampicillin and cefuroxime axetil. Br J Clin Pharmacol 18:535–9
   PubMed Web of Science ®Google Scholar
• Srivastava AK, Ridhurkar DN, Wadhwa S. (2005). Floating microspheres of cimetidine: formulation, characterization and in vitro evaluation. Acta Pharm 55:277–85
   PubMedGoogle Scholar
• Thakkar VT, Shah PA, Soni TG, et al. (2009). Goodness-of-Fit Model-Dependent approach for release kinetics of levofloxacin hemihydrates floating tablet. Dissol Technol 16:35–9
   Web of Science ®Google Scholar
• The United States Pharmacopoeia 31. (2008). United State Pharmacopeial Convention INC: Asian edition, 1698–700
   Google Scholar
• Wells JI, Aulton ME. (2007). Pharmaceutical preformulation. In: Aulton ME, ed. Aulton’s pharmaceutics: the design and manufacture of medicines, 3rd ed. USA, Churchill Livingstone: Elsevier, 355–7
   Google Scholar
• Yamashiro M, Yuasa Y, Kawakita K. (1983). An experimental study on the relationships between compressibility, fluidity and cohesion of powder solids at small tapping numbers. Powder Technol 34:225–31
   Web of Science ®Google Scholar