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Journal of Receptor Research Volume 11, 1991 - Issue 6
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Research Article

Evaluation of 3H-CGP 12177 and 3H-DHA Binding to β2-Adrenoceptors of Rat Reticulocytes by Means of Affinity Spectra

Z. Kállay Institute of Preventive and Clinical Medicine, 833 01, Bratislava
,
J. Šmisterová Institute of Experimental Pharmacology, Slovak Academy of Sciences, 842 16, Bratislava, Czecho-Slovakia
,
L. Šoltés Institute of Experimental Pharmacology, Slovak Academy of Sciences, 842 16, Bratislava, Czecho-Slovakia
&
V. Marko Institute of Experimental Pharmacology, Slovak Academy of Sciences, 842 16, Bratislava, Czecho-Slovakia
Pages 909-917 | Published online: 26 Sep 2008

References

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  • Stahelin M., Simons P., Jaeggi K., Wigger N. CGP 12177. A hydrophilic beta-adrenergic receptor radioligand reveals high affinity binding of agonists to intact cells. J. Biol. Chem. 1983; 258: 3496–3502
  • Kaiser G., Wiemer G., Kremer G., Dietz J., Palm D. Identification and quantification of beta-adrenoceptor sites in red blood cells from rats. Naunyn-Schmiedeberg's Arch. Pharmacol. 1978; 305: 41–50
  • Tobler H. J., Engel G. Affinity spectra: A novel way for the evaluation of equilibrium binding experiments. Naunyn-Schmiedeberg's Arch. Pharmacol. 1983; 322: 183–192
  • Šmisterová J., Šoltés L., Kallay Z. Purification of 3H-dihydroalprenolol by two dimensional thin layer chromatography. J. Label. Comp. Radiopharm. 198; 27: 481–484
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  • Šoltés L., Sébille B., Fügedi A. Evaluation of racemic propranolol binding to human alpha1-acid glycoprotein by means of affinity spectra. Does this approach recognize the affinities of propranolol enantiomers to the protein?. Bio-Sciences 1989; 8: 13–17
  • Klotz I. M. Number of receptor sites from Scatchard and Klotz graph: A constructive critique. Science 1983; 220: 979–981
  • Nahorski S. R., Richardson A. Pitfalls in the assessment of the specific binding of (-) [3H]-dihydroalpreno-lol to beta-adrenoceptors. Br. J. Pharmacol. 1979; 66: 469–470
  • Rademaker B., Kramer K., Stroes J. W., Vlug J., Krielaart M., Zaagsma J. High affinity non β-adrenoceptor binding of β-adrenergic ligands. Eur. J. Pharmacol. 1985; 111: 31–36
  • Tallman J. F., Smith C. C., Henneberry R. C. Induction of functional beta-adrenergic receptors in HeLa cells. Proc. Natl. Acad. Sci. U.S.A. 1977; 74: 873
  • Kerry R., Scrutton M. C. Binding of 3H-dihydroaplrenolol and H-acebutolol to human blood platelets is not related to occupancy of beta-adrenoceptors. Thrombosis Res. 1983; 29: 583
  • Dax E. M., Partilla J. S. Adrenergic ligand liposolubility in membranes. Mol. Pharmacol. 1982; 22: 5

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