References
- Dohlman H. G., Caron M. G., Lefkowitz R. J. A family of receptors coupled to guanine nucleotide regulatory proteins. Biochemistry 1987; 26: 2657–2664
- Khorana H. G. photoreceptor of the rod cell. J. Biol. Chem. 1992; 267: 1–4
- Lefkowitz R. J., Cotecchia S., Samama P., Costa T. Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins. Trends Pharmacol. Sci. 1993; 14: 303–307
- Unger V. M., Schertler G. F. X. Low resolution structure of bovine rhodopsin determined by electron cryo-microscopy. Biophys. J. 1995; 68: 1776–1786
- Strader C. D., Fong T. M., Tota M. R., Underwood D., Dixon R. A. F. Structure and function of G protein coupled receptors. Ann. Rev. Biochem. 1994; 63: 101–132
- Tota M. R., Strader C. D. Characterization of the binding domain of the beta-adrenergic receptor with the fluorescent antagonist carazolol. J. Biol. Chem. 1990; 265: 16891–16897
- Fong T. M., Strader C. D. Functional mapping of the ligand binding sites of G-protein coupled receptors. Med. Res. Rev. 1994; 14: 387–399
- Schwartz T. W. Locating ligand-binding sites in 7TM receptors by protein engineering. Curr. Opin. Biotechnol. 1994; 5: 434–444
- Li Y. M., Marnerakis M., Stimson E. R., Maggio J. E. Mapping peptide-binding domains of the substance P (NK1) receptor from P388D1 cells with photolabile agonists. J. Biol. Chem. 1995; 270: 1213–1220
- Boyd N. D., Kage R., Dumas J. J., Krause J. E., Leeman S. E. The peptide binding site of the substance P (NK1) receptor localized by a photoreactive analog of substance P: presence of a disulfide bond. Proc. Nat. Acad. Sci. 1996; 93: 433–437
- Fong T. M., Yu H., Huang R. R. C., Strader C. D. The extracellular domain of the human neurokinin-1 receptor is required for the high affinity binding of peptides. Biochemistry 1992; 31: 11806–11811
- Gether U., Johansen T. E., Schwartz T. W. Chimeric NK1/NK3 receptors: identification of domains determining the binding specificity of tachykinin agonists. J. Biol. Chem. 1993; 268: 7893–7898
- Huang R. R. C., Yu H., Strader C. D., Fong T. M. Interaction of substance P with the second and seventh transmembrane domains of the neurokinin-1 receptor. Biochemistry 1994; 33: 3007–3013
- Yokota Y., Akazawa C., Ohkubo H., Nakanishi S. Delineation of structural domains involved in the subtype specificity of tachykinin receptors through chimeric formation of substance P/substance K receptors. EMBOJ. 1992; 11: 3585–3591
- Brodbeck R. M., Sachais B. S., Krause J. E. Residue 78 in the second transmembrane domain of the neurokinin-1 receptor is important in coupling high affinity agonist binding to multiple second messenger responses. Mol. Pharmacol. 1995; 47: 1065–1071
- Helke C. J., Krause J. E., Mantyh P. W., Couture R., Bannon M. J. Diversity in mammalian tachykinin peptidergic neurons: multiple peptides, receptors and regulatory mechanisms. FASEB J. 1990; 4: 1606–1615
- Iversen L. L., Watling K. J., McKnight A. T., Williams B. J., Lee C. M. Multiple receptors for substance P and related tachykinins. Topics in Medicinal Chemistry, P. R. Leeming. Royal Soc. Chem., London 1987; 1–9
- Nakanishi S. Mammalian tachykinin receptors. Ann. Rev. Neurosci. 1991; 14: 123–136
- Benovic J. L., Shorr R. G., Caron M. G., Lefkowitz R. J. The mammalian beta 2-adrenergic receptor: purification and characterization. Biochemistry 1984; 23: 4510–4518
- Senogles S. E., Amlaiky N., Falardeau P., Caron M. G. Purification and characterization of the D2-dopamine receptor from bovine anterior pituitary. J. Biol. Chem. 1988; 263: 18996–19002
- Hochuli E., Dobeli H., Schacher A. New metal chelate adsorbent selective for proteins and peptides containing neighbouring histidine residues. J. Chromatogr 1987; 411: 177–184
- Cascieri M. A., Ber E., Fong T. M., Sadowski S., Bansal A., Swain C., Seward E., Francis B., Burns D., Strader C. D. Characterization of the binding of a potent, selective radioiodinated antagonist to the human neurokinin-1 receptor. Mol. Pharmacol. 1992; 42: 458–463
- Francis B. E., Swain C., Sabin V., Burns H. D. Radioiodinated L-703,606: a potent, selective antagonist to the human NK1 receptor. Applied Radiation and Isotopes 1994; 45: 97–103
- Mazina K. E., Strader C. D., Fong T. M. Expression and solubilization of a recombinant human neurokinin-1 receptor in insect cells. J. Receptor Res 1994; 14: 63–73
- DeBlasi A., O'Reilly K., Motulsky H. J. Calculating receptor number from binding experiments using same compound as radioligand and competitor. Trends Pharmacol. Sci. 1989; 10: 227–229
- Swillens S. How to estimate the total receptor concentration when the specific radioactivity of the ligand is unknown. Trends Pharmacol. Sci. 1992; 13: 430–434
- Taussig R., Quarmby L. M., Gilman A. G. Regulation of purified type I and type II adenylylcyclases by G protein beta gamma subunits. J. Biol. Chem. 1993; 268: 9–12
- Kwatra M. M., Schwin D. A., Schreurs J., Blank J. L., Kim C. M., Benovic J. L., Krause J. E., Caron M. G., Lefkowitz R. J. The substance P receptor, which couples to Gq/11, is a substrate of beta-adrenergic receptor kinase 1 and 2. J. Biol. Chem. 1993; 268: 9161–9164
- Fong T. M., Anderson S. A., Yu H., Huang R. R.C., Strader C. D. Differential activation of intracellular effectors by two isoforms of human neurokinin-1 receptor. Mol. Pharmacol. 1992; 41: 24–30