References
- Gill S, Sinicrope FA. Colorectal cancer prevention: Is an ounce of prevention worth a pound of cure? Semin Oncol 2005;32(1 Spec. issue):24–34.
- Phillips RKS, Wallace MH, Lynch PM, Hawk E, Gordon GB, Saunders BP, Wakabayashi N, Shen Y, Zimmerman S, Godio L, Rodrigues-Bigas M, Su L-K Sherman, J, Kelloff G, Levin B, Steinbach G, Abbruzzese J, Dubois Jr, R, Fujimura T, Hittleman W, Jester S, King K, Patterson S, Schumacher M. A randomised, double blind, placebo controlled study of celecoxib, a selective cyclooxygenase 2 inhibitor, on duodenal polyposis familial adenomatous polyposis. Gut 2002;50(6):857–860.
- Maljaars PWJ, Peters HPF, Mela DJ, Masclee AAM. Ileal brake: A sensible food target for appetite control. A review. Physiol Behav 2008;95(3):271–281.
- McConnell EL, Liu F, Basit AW. Colonic treatments and targets: Issues and opportunities. J Drug Target 2009;17(5):335–363.
- Haupt S, Rubinstein A. The colon as a possible target for orally administered peptide and protein drugs. Crit Rev Ther Drug Carrier Syst 2002;19(6):499–551.
- Ibekwe VC, Liu L, Fadda HM, Khela MK, Evans DF, Parsons GE, Basit AW. An investigation into the in vivo performance variability of pH responsive polymers for ileo-colonic drug delivery using gamma scintigraphy in humans. J Pharm Sci 2006;95:2760–2766.
- Ibekwe VC, Fadda HM, Parsons GE, Basit AW. A comparative in vitro assessment of the drug release performance of pH-responsive polymers for ileo-colonic delivery. Int J Pharm 2006;308:52–60.
- Siew LF, Man SM, Newton JM, Basit AW. Amylose formulations for drug delivery to the colon: A comparison of two fermentation models to assess colonic targeting performance in vitro. Int J Pharm 2004;273:129–134.
- Al-Saidan SM, Krishnaiah YS, Satyanarayana V, Rao GS. In vitro and in vivo evaluation of guar gum-based matrix tablets of rofecoxib for colonic drug delivery. Curr Drug Deliv 2005;2:155–163.
- Ramdas M, Dileep KJ, Anitha Y, Paul W, Sharma CP, Alginate encapsulated bioadhesive chitosan microspheres for intestinal drug delivery. J Biomater Appl 1999;13:290–296.
- Bigucci F, Luppi B, Monaco L, Cerchiara T, Zecchi V. Pectin-based microspheres for colon-specific delivery of vancomycin. J Pharm Pharmacol 2009;61:41–46.
- Hu Z, Mawatari S, Shimokawa T, Kimura G, Yoshikawa Y, Shibata N, Takada K. Colon delivery efficiencies of intestinal pressure-controlled colon delivery capsules prepared by a coating machine in human subjects. J Pharm Pharmacol 2000;52:1187–1193.
- Hu Z, Kimura G, Mawatari S, Shimokawa T, Yoshikawa Y, Takada K. New preparation method of intestinal pressure-controlled colon delivery capsules by coating machine and evaluation in beagle dogs. J Control Release 1998;56:293–302.
- Schellekens RCA, Stellaard F, Mitrovic D, Stuurman FE, Kosterink JGW, Frijlink HW. Pulsatile drug delivery to ileo-colonic segments by structured incorporation of disintegrants in pH-responsive polymer coatings. J Control Release 2008;132:91–98.
- Schellekens RCA, Olsder GG, Langenberg SMCH, Boer T, Woerdenbag HJ, Frijlink HW, Kosterink JGW, Stellaard F. Proof-of-concept study on the suitability of 13C-urea as a marker substance for assessment of in vivo behaviour of oral-targeted dosage forms. BJP 2009;158:532–540.
- Schellekens RCA, Stuurman FE, Van der Weert FHJ, Kosterink JGW, Frijlink HW. A novel dissolution method relevant to intestinal behaviour and its application in the evaluation of modified release mesalazine products. Eur J Pharm Sci 2007;30:15–20.
- EMEA/CPMP. Note for guidance on process validation. QWP 848/96, 2001.
- Vadas EB, Down GR, Miller RA. Effect of compressional force on tablets containing cellulosic disintegrators; I-Dimensionless disintegration values. J Pharm Sci 1984;73:781–783.
- Bauer KH, Lehman K, Osterwald HP, Rothgang G. Coated pharmaceutical dosage forms. Stuttgart: Medpharma GmbH Scientific Publishers; 1998:26.
- Rowe RC. The adhesion of film coatings to tablet surfaces – the effect of some direct compression excipients and lubricants. J Pharm Pharmaceut 1977;29:723–726.
- List PH, Muazzam UA. Quellung-Die treibende kraft beim Tablettenzerfall. Pharm Ind 1981;43:480–484.
- Colombo P, Caramella C, Conte U, La Manna A. Disintegrating force and tablet properties. DDIP 1981;7:135–153.
- Van Kamp HV, Bolhuis GK, Lerk CF. Improvement by superdisintegrants of the properties of tablets containing lactose, prepared by wet granulation. PW Sci Ed 1983;5:165–171.
- Van Kamp HV, Bolhuis GK, De Boer AH, Lerk CF, Lie-A-Huen L. The role of water uptake on tablet disintegration. Pharm Acta Helv 1986;61:22–29.