Development of a novel bi-coated combination capsule containing mosapride and probiotics for irritable bowel syndrome

References

• Brandt L, Chey W, Foxx-Orenstein A, et al. An evidence-based systematic review on the management of irritable bowel syndrome. Am J Gastroenterol 2009;104:S1–S35
   PubMed Web of Science ®Google Scholar
• El-Serag B, Olden K, Bjorkaman D. Health-related quality of life among persons with irritable bowel syndrome: a systematic review. Aliment Pharmacol Ther 2002;16:1171–1185
   PubMed Web of Science ®Google Scholar
• Gralnek M, Hays D, Kilbourne A, et al. The impact of irritable bowel syndrome on health-related quality of life. Gastroenterology 2000;119:654–660
   PubMed Web of Science ®Google Scholar
• Camilleri M, Lasch K, Zhou W. Irritable bowel syndrome: methods, mechanisms, and pathophysiology. The confluence of increased permeability, inflammation, and pain in irritable bowel syndrome. Am J Physiol Gastrointest Liver Physiol 2012;303:775–785
   PubMed Web of Science ®Google Scholar
• Mayer A, Naliboff D, Chang L. Evolving pathophysiological model of functional gastrointestinal disorders: implications for treatment. Eur J Surg Suppl 2002;587:3–9
   Google Scholar
• Neal R, Hebden J, Spiller R. Prevalence of gastrointestinal symptoms six months after bacterial gastroenteritis and risk factors for development of the irritable bowel syndrome: postal survey of patients. BMJ 1997;314:779–782
   PubMed Web of Science ®Google Scholar
• McKendrick W, Read W. Irritable bowel syndrome-post salmonella infection. J Infect 1994;29:1–3
   PubMed Web of Science ®Google Scholar
• Sanders S, Carter J, Hurlstone P, et al. Association of adult coeliac disease with irritable bowel syndrome: a case control study in patients fulfilling ROME II criteria referred to secondary care. Lancet 2001;3:1504–1508
   Google Scholar
• Guyonnet D, Chassany O, Ducrotte P. Effect of a fermented milk containing Bifidobacterium animalis DN-173 010 on the health-related quality of life and symptoms in irritable bowel syndrome in adults in primary care: a multicentre, randomized, double blind, controlled trial. Aliment Pharmacol Ther 2007;26:475–486
   PubMed Web of Science ®Google Scholar
• Kim J, Vazquez Roque I, Camilleri M. A randomized controlled trial of a probiotic combination VSL#3 and placebo in irritable bowel syndrome with bloating. Neurogastroenterol Motil 2005;17:687–696
   PubMed Web of Science ®Google Scholar
• Fuller R. Probiotics in man and animals. J Appl Bacteriol 1989;66:365–378
   PubMedGoogle Scholar
• O'Mahony L, Feeney M, O'Halloran S, et al. Probiotic impact on microbial flora, inflammation and tumour development in IL-10 knockout mice. Aliment Pharmacol Ther 2001;15:1219–1225
   PubMed Web of Science ®Google Scholar
• McCarthy J, O'Mahony L, O'Callaghan L, et al. Double blind, placebo controlled trial two probiotic strains in interleukin 10 knockout mice and mechanistic link with cytokine balance. Gut 2003;52:975–980
   PubMed Web of Science ®Google Scholar
• Andersson H, Asp G, Bruce A, et al. Health effects of probiotics and prebiotics: a literature review on human studies. Scand J Nutr 2001;45:58–75
   Google Scholar
• O'Mahony L, McCarthy J, Kelly P, et al. Lactobacillus and bifidobacterium in irritable bowel syndrome: symptom responses and relationship to cytokine profiles. Gastroenterology 2005;128:541–551
   PubMed Web of Science ®Google Scholar
• Susanna R, Pirjo R. Protecting probiotic bacteria by microencapsulation: challenges for industrial applications. Eur Food Res Technol 2010;231:1–12
   Web of Science ®Google Scholar
• Aguirre M, Collins D. Lactic acid bacteria and human clinical infection. J Appl Bacteriol 1993;75:95–107
   PubMedGoogle Scholar
• Hilton E, Isenberg D, Alperstein P, et al. Ingestion of yogurt containing Lactobacillus acidophilus as prophylaxis for candidal vaginitis. Ann Intern Med 1992;116:353–357
   PubMed Web of Science ®Google Scholar
• De Roos M, Katan B. Effects of probiotic bacteria on diarrhea, lipid metabolism, and carcinogenesis: a review of papers published between 1988 and 1998. Am J Clin Nutr 2000;71:405–411
   PubMed Web of Science ®Google Scholar
• Islam A, Yun H, Choi J, Cho S. Microencapsulation of live probiotic bacteria. Microbiol Biotechnol 2010;20:1367–1377
   Google Scholar
• Kailasapathy K, Chin J. Survival and therapeutic potential of probiotic organisms with reference to Lactobacillus acidophilus and Bifidobacterium species. Immunol Cell Biol 2000;78:80–88
   PubMed Web of Science ®Google Scholar
• Charalampopoulos D, Pandiella SS, Webb C. Growth studies of potentially probiotic lactic acid bacteria in cereal-based substrates. J Appl Microbiol 2002;92:851–859
   PubMed Web of Science ®Google Scholar
• Chang S. Therapeutic applications of polymeric artificial cells. Nat Rev Drug Discov 2005;4:221–235
   PubMed Web of Science ®Google Scholar
• Sun M, Goosen F, O'Shea G. Microencapsulated cells as hormone delivery systems. Crit Rev Ther Drug Carrier Syst 1987;4:1–12
   PubMed Web of Science ®Google Scholar
• Kim G, Moon T, Lee M. The effects of probiotics on symptoms of irritable bowel syndrome. Korean J Gastroenterol 2006;47:413–419
   PubMedGoogle Scholar
• Kanaizumi T, Nakano H, Matsui Y, et al. Prokinetic effect of AS-4370 on gastric emptying in healthy adults. Eur J Clin Pharmacol 1991;42:335–337
   Google Scholar
• Yoshida N, Kato S, Ito T. Oral bioavailability was 8% of the dose in dogs and 14% in monkeys, suggesting the extensive first-pass metabolism of mosapride. Drugs Future 1993;18:513–515
   Google Scholar
• Yoshida N, Omoya H, Oka M, et al. AS-4370, a novel gastrokinetic agent free of dopamine D2 receptor antagonist properties. Arch Int Pharmacodyn Ther 1989;300:51–67
   PubMedGoogle Scholar
• Karasawa T, Yoshida N, Furukawa K, et al. Comparison of gastrokinetic effects of AS-4370, cisapride and BRL 24924. Eur J Pharmacol 1990;183:2181
   Web of Science ®Google Scholar
• Liu Z, Sakakibara R, Odaka T, et al. Mosapride citrate, a novel 5-HT4 agonist and partial 5-HT3 antagonist, ameliorates constipation in parkinsonian patients. Mov Disord 2005;20:680–686
   PubMed Web of Science ®Google Scholar
• Young N. How to increase serotonin in the human brain without drugs. J Psychiatry Neurosci 2007;32:394–399
   PubMed Web of Science ®Google Scholar
• Gershon D, Tack J. The serotonin signaling system: from basic understanding to drug development for functional GI disorders. Gastroenterology 2007;132:397–414
   PubMed Web of Science ®Google Scholar
• Sakashita M, Mizuki Y, Yamaguchi T, et al. Pharmacokinetics of the gastrokinetic agent mosapride citrate after intravenous and oral administrations in dogs and monkeys. Arzneimittelforschung 1993;43:864–866
   PubMed Web of Science ®Google Scholar
• Society of Toxicology (SOT). Guiding principles in the use of animals in toxicology. 2008. Available from: http://www.toxicology.org/ai/fa/guidingprinciples.pdf [last accessed 20 June 2012]
   Google Scholar
• Newa M, Bhandari H, Li K, et al. Preparation, characterization and in vivo evaluation of ibuprofen binary solid dispersions with poloxamer 188. Int J Pharm 2007;343:228–237
   PubMed Web of Science ®Google Scholar
• Costa P, Sousa Lobo M. Influence of dissolution medium agitation on release profiles of sustained-release tablets. Drug Dev Ind Pharm 2001;27:811–817
   PubMed Web of Science ®Google Scholar
• Keller A, Czerniuk P, Bertuola R, et al. Relative bioavailability of a 5 mg mosapride/10 mg rabeprazole fixed dose combination tablet versus separate single tablets in healthy volunteers: a single-dose randomized open-label crossover study. Curr Med Res Opin 2011;27:2203–2211
   PubMed Web of Science ®Google Scholar
• Kim Y, Kim K, Suh K, et al. New clopidogrel napadisilate salt and its solid dispersion with improved stability and bioequivalence to the commercial clopidogrel bisulphate salt in beagle dogs. Int J Pharm 2011;415:129–139
   PubMed Web of Science ®Google Scholar
• Oh D, Park Y, Kang J, et al. Physicochemical characterization and in vivo evaluation of flurbiprofen-loaded solid dispersion without crystalline change. Drug Deliv 2011;18:46–53
   PubMed Web of Science ®Google Scholar