181
Views
3
CrossRef citations to date
0
Altmetric
Research Article

A novel bile salts–lipase polymeric film-infused minitablet system for enhanced oral delivery of cholecalciferol

, , , , &
Pages 832-846 | Received 24 Apr 2015, Accepted 24 Jun 2015, Published online: 27 Aug 2015

References

  • Sharma P, Varma MVS, Chawls HPS, Panchagnula R. Absorption enhancement, mechanistic and toxicity studies of medium chain fatty acids, cyclodextrins and bile salts and peroral absorption enhancers. Il Farmaco 2005;60:884–893
  • Charkoftaki G, Dokoumetzidis A, Valsami G, Macheras P. Supersaturated dissolution data and their interpretation: the TPGS-carbamazepine model case. J Pharm Pharmacol 2011;63:352–361
  • Maestrelli F, Cirri M, Mennini N, et al. Improvement in oxaprozin solubility and permeability by the combined use of cyclodextrin, chitosan, and bile components. Eur J Pharm Sci 2011;78:385–393
  • Bernabeu E, Helguera G, Legaspi MJ, et al. Paclitaxel-loaded PCL-TPGS nanoparticles: in vitro and in vivo performance compared to abraxane. Colloid Surface B 2014;113:43–50
  • Nair, HB, Sung B, Yadav VR, et al. Delivery of anti-inflammatory nutraceuticals by nanoparticles for the prevention and treatment of cancer. Biochem Pharmacol 2010;80:1833–1843
  • Garti N, Libster D, Aserin A. Lipid polymorphism in lyotropic liquid crystals for triggered release of bioactives. Food Funct 2012;3:700–713
  • Xia S, Tan C, Xue J, et al. Chitosan/tripolyphosphate-nanoliposomes core-shell nanocomplexes as vitamin E carriers: shelf-life and thermal properties. Int J Food Sci Technol 2014;49:1367–1374
  • Samstein RM, Perica K, Balderrama F, et al. The use of deoxycholic acid to enhance the oral bioavailability of biodegradable nanoparticles. Biomaterials 2008;29:703–708
  • Fieker A, Philpott J, Armand M. Enzyme replacement therapy for pancreatic insufficiency: present and future. J Clin Exp Gastroenterol 2011;4:55–73
  • Braithwaite MC, Kumar P, Tyagi C, et al. Vitamin D therapy and related metabolomics: is the calciferol dose and form the only requirements for successful clinical therapeutics? Med Hypotheses 2013;81:656–663
  • Nandy BC, Roy Sandipan R, Mazumder B, et al. In vitro–in vivo correlation: application in pharmaceutical development of various dosage forms. J Chem Pharm Res 2011;3:550–564
  • Mercê ALR, Nicolini J, Khan MA, Bouet G. Qualitative study of supramoleculkar assemblies of β-cyclodextrin and cholecalciferol and the cobalt (II), copper (II) and zinc (II) ions. Carbohyd Polym 2009;77:402–409
  • Giannola LI, De Caro V, Giandalia G, et al. Release of naltrexone on bucal mucosa: permeation studies, histological aspects and matrix system design. Eur J Pharm Biopharm 2007;67:425–433
  • Xue X, You J, He P. Simultaneous determination of five fat-soluble vitamins in feed by high-performance liquid chromatography following solid-phase extraction. J Chromatogr Sci 2008;46:345–349
  • Zhang Y, Huo M, Zhou J, et al. DDSolver: an add-in program for modelling and comparison of drug dissolution profiles. AAPS J 2010;12:263–271
  • Medina JR, Salazar DK, Hurtado M, et al. Comparative in vitro dissolution study of carbamazepine immediate-release products using the USP paddles method and the flow-through cell system. Saudi Pharm J 2014;22:141–147
  • Wang J, Cao Y, Sun B, Wang C. Physicochemical and release characterization of garlic oil-b-cyclodextrin inclusion complexes. Food Chem 2011;127:1680–1685
  • Teng Z, Luo Y, Wang Q. Carboxymethyl chitosan–soy protein complex nanoparticles for the encapsulation and controlled release of vitamin D3. Food Chem 2013;141:524–532
  • Yuan T, Qin L, Wang Z, et al. Solid dispersion of calcitriol with enhanced dissolution and stability. Asian J Pharm Sci 2013;8:39–47
  • Hu X, Wei B, Wu C, et al. Preparation of the β-cyclodextrin-vitamin C (β-CD-Vc) inclusion complex under high hydrostatic pressure (HHP). Carbohyd Polym 2012;90:1193–1196
  • Shin S, Kim J. Physicochemical characterization of solid dispersion of furosemide with TPGS. Int J Pharm 2003;251:79–84
  • Yang L, Xu Y, Su Y, et al. FT-IR spectroscopic study on the variations of molecular structures of some carboxyl acids induced by free electron laser. Spectrochim Acta A 2005;62:1209–1215
  • Ahmed MK, McLeod MP, Nezivar J, Giuliani AW. Fourier transform infrared and near-infrared spectroscopic methods for the detection of toxic diethylene glycol contaminant in glycerin based cough syrup. Spectroscopy 2010;24:601–608
  • Pongjanyakul T, Puttipipatkhorn S. Alginate-magnesium aluminium silicate films: effect of plasticizers on film properties, drug permeation and drug release from coated tablets. Int J Pharm 2007;333:34–44
  • Thu H, Ng S. Gelatine enhances drug dispersion in alginate bilayer film via the formation of crystalline microaggregates. Int J Pharm 2013;454:99–106
  • Charusheela A, Arvind L. Enzyme hydrolysis of esters using reversibly soluble polymer conjugated lipases. Enzyme Microb Technol 2002;30:19–25
  • Mu L, Feng SS. A novel controlled release formulation for the anticancer drug paclitaxel (Taxol): PLGA nanoparticles containing vitamin E. J Control Release 2003;86:33–48
  • Guo Y, Luo J, Tan S, et al. The applications of Vitamin E TPGS in drug delivery. Eur J Pharm Sci 2013;49:175–186
  • Dua K, Pabreja K, Ramana MV, Lather V. Dissolution behavior of β-cyclodextrin molecular inclusion complexes of aceclofenac. J Pharm Bioallied Sci 2011;3:417–425
  • Alishahi A, Mirvaghefi A, Tehrani MR, et al. Shelf life and delivery enhancement of vitamin C using chitosan nanoparticles. Food Chem 2011;126:935–940
  • Huq T, Salmieri S, Khan A, et al. Nanocrystalline cellulose (NCC) reinforced alginate based biodegradable nanocomposite film. Carbohyd Polym 2012;90:1757–1763
  • Pereira R, Carvalho A, Vaz DC, et al. Development of novel alginate based hydrogel films for wound healing. Int J Biol Macromol 2013;52:221–230
  • Goddeeris C, Willems T, Van den Mooter G. Formulation of fast disintegrating tablets of ternary solid dispersions consisting of TPGS 1000 and HPMC 2910 or PVPVA 64 to improve the dissolution of the anti-HIV drug UC 781. Eur J Pharm Sci 2008;34:293–302
  • Ostacolo C, Caruso C, Tronino D, et al. Enhancement of corneal permeation of riboflavin-5-phosphate through vitamin E TPGS: a promising approach in corneal trans-epithelial cross linking treatment. Int J Pharm 2013;440:148–153
  • Jin F, Tatavarti A. Tabletability assessment of conventional formulations containing vitamin E tocopheryl polyethylene glycol succinate. Int J Pharm 2010;389:58–65
  • Saphier S, Rosner A, Brandeis R, Karton Y. Gastro intestinal tracking and gastric emptying of solid dosage forms in rats using X-ray imaging. Int J Pharm 2010;388:190–195
  • Cordova H, Guarner-Argente C, Martinez-Palli G, et al. Gastric emptying is delayed in transgastric notes: a randomized study in swine. J Surg Res 2012;174:e61–e67
  • Anderson DL, Bartholomeusz D, Kirkwood ID, et al. Liquid gastric emptying in the pig: effect of concentration of inhaled isoflurane. J Nucl Med 2002;43:968–971
  • Saadati R, Dadashzadeh S. Marked effects of combined TPGS and PVA emulsifiers in the fabrication of etoposide-loaded PLGA-PEG nanoparticles: in vitro and in vivo evaluation. Int J Pharm 2014;464:135–144
  • Zhang Z, Tan S, Feng S. Vitamin E TPGS as a molecular biomaterial for drug delivery. Biomaterials 2012;33:4889–4906
  • Jones G. Pharmacokinetics of vitamin D toxicity. Am J Clin Nutr 2008;88:582S–586S
  • Chen Y, Lu Yi, Chen J, et al. Enhanced bioavailability of the poorly water-soluble drug fenofibrate by using liposomes containing bile salt. Int J Pharm 2009;376:153–160
  • Niu M, Lu Y, Hovgaard L, et al. Hypoglycemic activity and oral bioavailability of insulin-loaded liposomes containing bile salts in rats: the effect of cholate type, particle size and administered dose. Eur J Pharm Biopharm 2012;81:265–272
  • Van Hasselt PM, Janssens GEPJ, Slot TK, et al. The influence of bile acids on the oral bioavailability of vitamin K encapsulated in polymeric micelles. J Control Release 2009;133:161–168
  • Wolpowitz D, Gilchrest BA. The vitamin D questions: how much do you need and how should you get it? J Am Acad Dermatol 2006;54:301–317
  • Haddad JG, Rojanasathit S. Acute administration of 25-hydroxycholecalciferol in man. J Clin Endocrinol Metab 1976;42:284–290
  • Heaney RP, Davies MK, Chen TC, et al. Human serum 25-hydroxycholecalciferol response to extended oral dosing with cholecalciferol. Am J Clin Nutr 2003;77:204–210
  • Stephenson A, Brotherwood M, Rober R, et al. Cholecalciferol significantly increases 25-hydroxyvitamin D concentrations in adults with cystic fibrosis. Am J Clin Nutr 2007;85:1307–1311
  • Horst RL, Reinhardt TA. Chapter 2. Vitamin D metabolism. In: Feldman D, Glorieux FH, Pike JW, eds. Vitamin D. Academic Press: San Diego; 1997:69–85
  • Pointillart A, Fontaine N. Effects of vitamin D on calcium regulation in vitamin-D-deficient pigs given a phytate-phosphorous diet. Brit J Nutr 1986;56:661–669
  • Flohr JR, Tokach MD, Dritz SS, et al. Effects of supplemental vitamin D3 on serum 25-hydroxycholecalciferol and growth of preweaning and nursery pigs. J Anim Sci 2014;92:152–163
  • Brannon PM, Yetley AE, Bailey RL, Picciano MF. Summary of roundtable discussion on vitamin D research needs. Am J Clin Nutr 2008;88:5875S–5892S

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.