References
- Lecaille F, Kaleta J, Brömme D. Chem Rev 2002;102:4459–88.
- Powers JC, Asgian JL, Ekici öD, James KE. Chem Rev 2002;102:4639–750.
- Vicik R, Busemann M, Baumann K, Schirmeister T. Curr Top Med Chem 2006;6:331–53.
- Schaschke N, Assfalg-Machleidt I, Machleidt W, Turk D, Moroder L. Bioorg Med Chem 1997;5:1789–97.
- Schirmeister T. J Med Chem 1999;42:560–72.
- Shaw E. Methods Enzymol 1994;244:649–56.
- Brömme D, Klaus JL, Okamoto K, Rasnick D, Palmer JT. Biochem J 1996;315:85–9.
- Darkins P, Gilmore BF, Hawthorne SJ, Healy A, Moncrieff H, McCarthy N, McKervey MA, Brömme D, Pagano M, Walker B. Chem Biol Drug Des 2007;69:170–9.
- Santos MMM, Moreira R. Mini-Rev Med Chem 2007;7:1040–50.
- Moon JB, Coleman RS, Hanzlik RP. J Am Chem Soc 1986;108:1350–1.
- Löser R, Frizler M, Schilling K, Gütschow M. Angew Chem Int Ed Engl 2008;47:4331–4.
- Wright SW, Ammirati MJ, Andrews KM, Brodeur AM, Danley DE, Doran SD, Lillquist JS, McClure LD, McPherson RK, Orena SJ, Parker JC, Polivkova J, Qiu X, Soeller WC, Soglia CB, Treadway JL, VanVolkenburg MA, Wang H, Wilder DC, Olson TV. J Med Chem 2006;49:3068–76.
- Gütschow M, Powers JC. J Org Chem 2001;66:4723–7.
- Tietze LF. Chem Rev 1996;96:115–36.
- Linnevers CJ, McGrath ME, Armstrong R, Mistry FR, Barnes MG, Klaus JL, Palmer JT, Katz BA, Brömme D. Protein Sci 1997;6:919–21.
- Snyder HR, Sekleton JF, Lewis CD. J Am Chem Soc 1945;67:310–12.
- Singh P, Berlinguet L. Can J Chem 1964;42:605–9.
- Boomgaarden M, Heinrich G, Henklein P. Pharmazie 1992;47:710–11.
- Johnson HE, Crosby DG. J Org Chem 1962;27:798–802.
- Löser R, Schilling K, Dimmig E, Gütschow M. J Med Chem 2005;48:7688–707.
- Copeland RA. Enzymes: A Practical Indroduction to Structure, Mechanism and Data Analysis. New York: Wiley-VCH, 2005:282–3.
- Cheng YC, Prusoff WH. Biochem Pharmacol 1973;22:3099–108.
- Loughlin WA, Tyndall JDA, Glenn MP, Fairlie DP. Chem Rev 2004;104:6085–117.
- Olah GA, Narang SC, Fung AP, Gupta BGB. Synthesis 1980:657–8.
- Tyndall JDA, Nall T, Fairlie DP. Chem Rev 2005;105:973–99.
- Wilson SR, Cui W. Biopolymers 1990;29:225–35.
- van Gunsteren W, Berendsen HJC. Angew Chem Int Ed Engl 1990;29:992–1023.
- Sewald N, Jakubke HD.Peptides: Chemistry and Biology. Weinheim: Wiley-VCH, 2002:40.
- DeLano WL. The PyMOL Molecular Graphics System. San Carlos, CA: DeLano Scientific, 2005.
- Scheidt KA, Roush WA, McKerrow JH, Selzer PM, Hansell E, Rosenthal PJ. Bioorg Med Chem 1998;6:2477–94.
- Turk D, Guncar G, Podobnik M, Turk B. Biol Chem 1998;379:137–47.
- Elnagdi MH, Khalifa MAE, Ibraheim MKA, Elmoghayar MRH. J Heterocyclic Chem 1981;18:877–9.
- Clayden J, Greeves N, Warren S, Wothers P. Organic Chemistry. Oxford: Oxford University Press, 2001:1140–3.
- Freidinger RM, Perlow DS, Veber DF. J Org Chem 1982;47:104–9.
- Tian WX, Tsou CL. Biochemistry 1982;21:1028–32.
- Copeland RA. Evaluation of Enzyme Inhibitors in Drug Discovery. Hoboken: Wiley-Interscience, 2005:215–19.
- Ward YD, Thomson DS, Frye LL, Cywin CL, Morwick T, Emmanuel MJ, Zindell R, McNeil D, Bekkali Y, Girardot M, Hrapchak M, DeTuri M, Crane K, White D, Pav S, Wang Y, Hao M-H, Grygon CA, Labadia ME, Freeman DM, Davidson W, Hopkins JL, Brown ML, Spero DM. J Med Chem 2002;45:5471–82.