References
- Broom AD. J Med Chem 1989;32:2–7.
- Wolfenden R. Accts Chem Res 1972;5:10–18.
- Heller JS, Canellakis ES, Bussolotti DL, Coward JK. Biochem Biophys Acta 1975;403:197–207.
- Shemin D. Methods Enzymol 1970;17:205–11.
- Gacond S, Frère F, Nentwich M, Fauritea JP, Frankenberg-Dinkel N, Neier N. Chem Biodivers 2007;4:189–202.
- Kang K, Fromm HJ. J Biol Chem 1995;270:15539–44.
- Heim DR, Cseke C, Gerwick BC, Murdoch MG, Green SB. Pestic Biochem Physiol 1995;53:138–45.
- Cseke C, Gerwick BC, Crouse GD, Murdoch MG, Green SB, Heim DR. Pestic Biochem Physiol 1996;55:210–17.
- Fonne-Pfister R, Chemla P, Ward E, Girardet M, Kreuz KE, Honzatko RB, et al. Proc Natl Acad Sci USA 1996;93:9431–6.
- Walters EW, Lee S, Niderman T, Bernasconi P, Subramanian MV, Siehl D. Plant Physiol 1997;114:549–55.
- Hatch MD.. Phytochemistry 1967;6:115–19.
- Hanessian S, Lu PP, Sanceau JY, Chemla P, Gohda K, Fonne-Pfister R, et al. Angew Chem Int Ed 1999;38:3160–2.
- Abu-Elheiga L, Matzuk MM, Abo-Hashema KAH, Wakil SJ. Science 2001;291:2613–16.
- Lenhard JM, Gottschalk WK. Adv Drug Delivery Rev 2002;54:1199–212.
- Levert KL, Waldrop GL, Stephens JM. J Biol Chem 2002;277:16347–50.
- Campbell JW, Cronan JE Jr. Annu Rev Microbiol 2001;55:305–32.
- Blanchard CZ, Waldrop GL. J Biol Chem 1998;273:19140–5.
- Levert KL, Grover L, Waldrop GL. Biochem Biophys Res Commun 2002;291:1213–17.
- Ravindranadh VS, Wilson DJ, Bennett EM, Boshoff HI, Celia L, Beck BJ, et al. J Med Chem 2006;49:7623–35.
- Ravindranadh VS, Boshoff HI, Qiao C, Bennett EM, Barry CE, Aldrich CC. J Med Chem 2006;49:31–6.
- Vannada J, Bennett EM, Wilson DJ, Boshoff HI, Barry CE, Aldrich CC. Org Lett 2006;8:4707–10.
- Finking R, Neumuller A, Solsbacher J, Konz D, Kretzschmar G, Schweitzer M, et al. Chem Biol Chem 2003;4:903–6.
- May JJ, Finking R, Wiegeshoff F, Weber TT, Bandur N, Koert U, et al. FEBS J 2005;272:2993–3003.
- Ferreras JA, Ryu JS, Di Lello F, Tan DS, Quadri LE. Nat Chem Biol 2005;1:29–32.
- Miethke M, Bisseret P, Beckerin CL, Vignard D, Eustache J, Marahiel MA. FEBS J 2006;273:409–19.
- Neres JO, Labello PN, Somu RV, Boshoff HI, Wilson DJ, Vannada J, et al. J Med Chem 2008;51:5349–70.
- Wimalasena K, Wimalasena DS, Dharmasena S, Haines DC, Alliston KR. Biochemistry 1997;36:7144–53.
- Kruse LI, Kaiser C, DeWolf WE Jr, Frazee JS, Garvey E, Hilbert EL, et al. J Med Chem 1986;29:2465–72.
- Kruse LI, Kaiser C, DeWolf WE Jr, Frazee JS, Ross ST, Wawro J, et al. J Med Chem 1987;30:486–94.
- Kruse LI, DeWolf WE Jr, Chambers PA, Goodhart PJ. Biochemistry 1986;25:7271–8.
- Ross ST, Kruse LI, Ohlstein EH, Erickson RW, Ezekiel M, Flaim KE, et al. J Med Chem 1987;30:1309–13.
- Miyano K, Koshigoe T, Sakasai T, Hamano H. Chem Pharm Bull 1978;26:1465–72.
- Kruse LI, Kaiser C, Dewolf WE Jr, Finkelstein JA, Frazee JS, Hilbert EL, et al. J Med Chem 1990;33:781–9.
- Salituro FG, Demeter DA, Weintraub HJR, Lippert BJ, Resvick RJ, McDonald IA. J Med Chem 1994;37:4076–8.
- Kaustov L, Kababya S, Belakhov V, Baasov T, Shoham T, Schmidt A. J Am Chem Soc 2003;125:4662–9.
- Du S, Faiger H, Belakhov V, Baasov T. Bioorg Med Chem 1999;7:2671–82.
- Anderson L, Unger FM, eds. Bacterial Lipopolysaccharides. ACS Symposium, Series 231. Washington DC: American Chemical Society, 1983.
- Inouye M. Bacterial Outer Membrane: Biogenesis and Function. New York: Wiley, 1979.
- Ray PH. J Bacteriol 1980;141:635–44.
- Hedstrom L, Abeles R. Biochem Biophys Res Commun 1988;157:816–20.
- Sheffer-Dee-Noor S, Belakhov V, Baasov T. Bioorg Med Chem Lett 1993;3:1583–8.
- Baasov T, Sheffer-Dee-Noor S, Kohen A, Jakob A, Belakhov V. Eur J Biochem 1993;217:991–9.
- Dotson GD, Dua RK, Clemens JC, Wooten EW, Woodard RW. J Biol Chem 1995;270:13698–705.
- Korolev S, Ikeguchi Y, Skarina T, Beasley S, Arrowsmith C, Edwards A, et al. Nat Struct Biol 2001;9:27–31.
- Woster PM, Black AY, Duff KJ, Coward JK, Pegg AE. J Med Chem 1989;32:1300–7.
- Tang KC, Mariuzza R, Coward JK. J Med Chem 1981;24:1277–84.
- Orr GR, Danz DW, Pontoni G, Prabhakaran PC, Gould SJ, Coward JK. J Am Chem Soc 1988;110:5791–9.
- Jencks WP. Adv Enzymol Relat Areas Mol Biol 1975;45:219–23.
- Lakanen JR, Pegg AE, Coward JK. J Med Chem 1995;38:2714–27.
- Dev IK, Harvey RJ. J Biol Chem 1978;253:4242–4.
- Beardsley GP, Taylor EC, Shih C, Poore GA, Grindey GB, Moran RG. Proc AACR 1986;27:259 (abstr 1027).
- Inglese J, Blatchly RA, Benkovic SJ. J Med Chem 1989;32:937–40.
- Greasley SE, Yamashita M, Kai H, Benkovic SJ, Boger DL, Wilson IA. Biochemistry 1999;38:16783–93.
- Greasley SE, Marsilje TH, Kai H, Baker S, Benkovic SJ, Boger DL, et al. Biochemistry 2001;40:13538–47.
- Wall N, Shim JH, Benkovic SJ. J Med Chem 1999;42:3421–4.
- Klein C, Chen P, Arevalo JH, Stura EA, Marolewski A, Warren MS, et al. J Mol Biol 1995;249:153–75.
- Diasio RB, Schuetz JD, Banks W, Wallace H. Proc Am Assoc Cancer Res 1982;23:214.
- Cohen SS. Ann NY Acad Sci 1971;186:292–301.
- Srinivasan A, Amarnath V, Broom AD, Zou FC, Cheng YC. J Med Chem 1984;27:1710–17.
- Koyama H, Ayusawa D, Tsuji M, Seno T. Mutat Res 1982;105:433–8.
- Park JS, Chang CTC, Mertes MP. J Med Chem 1979;22:1134–7.
- Yang IY, Slusher RM, Broom AD, Ueda T, Cheng YC. J Med Chem 1988;31:2126–38.
- Lovelace LL, Gibson LM, Lebioda L. Biochemistry 2007;46:2823–30.
- Enkvist E, Lavogina D, Raidaru G, Vaasa A, Viil I, Lust M, et al. J Med Chem 2006;49:7150–9.
- Goldberg AR, Wong TW. Adv Enzyme Regul 1984;22:289–308.
- Kruse CH, Holden KG, Offen PH, Pritchard JAF, Reiman DJ, Bender PE, et al. J Med Chem 1988;31:1768–72.
- Traxler PM, Wacker O, Bach HL, Geissler JF, Kump W, Meyer T, et al. J Med Chem 1991;34:2328–37.
- Russo MW, Lukas TJ, Cohen S, Staros JV. J Biol Chem 1985;160:5205.
- Zoller MN, Nelson NC, Taylor SS. J Biol Chem 1981;256:10837–42.
- Kamps MP, Taylor SS, Sefton BM. Nature 1984;310:589–92.
- Baginski, I, Commerçon A, Tocqué B, Colson G, Zerial A. Biochem Biophys Res Commun 1989;165:1324–30.
- Imoto M, Umezawa K, Sawa T, Takeuchi T, Umezawa H. Biochem Int 1987;15:989–95.
- Lienhard GE, Secemski II. J Biol Chem 1973;248:1121–3.
- Miron S, Munier-Lehmann H, Craescu CT. Biochemistry 2004;43:67–77.
- Lavie A, Konrad M, Brundiers R, Goody RS, Schlichting I, Reinstein J. Biochemistry 1998;37:3677–86.
- Bone R, Cheng YC, Wolfenden R. J Biol Chem 1986;261:5731–5.
- Bone R, Cheng YC, Wolfenden R. J Biol Chem 1986;261:16410–13.
- Ikeda S, Chakravarty R, Ives DH. J Biol Chem 1986;261:15836–43.
- Shen W, Willis D, Zhang Y, Schlattner U, Wallimann T, Molloy GR. Biochem J 2002;367:369–80.
- Min K-L, Steghens J-P, Henry R, Doutheau A, Collombel C. Biochim Biophys Acta 1997;1342:83–9.
- Williams DM, Jakeman DL, Vyle JS, Williamson MP, Blackbum GM. Bioorg Med Chem Lett 1998;8:2603–8.
- Blackburn GM, Jakeman DL, Ivory AJ, Williamson MP. Bioorg Med Chem Lett 1994;4:2573–8.
- Jakeman DL, Ivory AJ, Williamson MP, Blackburn GM. J Med Chem 1998;41:4439–52.
- Shiota T. Chemistry and Biochemistry of Folates. New York: John Wiley & Sons, 1984:121.
- Shi G, Blaszczyk J, Ji X, Yan H. J Med Chem 2001;44:1364–71.
- Nakadate T, Jeng AY, Blumberg PM. Biochem Pharmacol 1988;8:1541–5.
- Ricouart A, Gesquiere JC, Tartar A, Sergheraert C. J Med Chem 1991;34:73–8.
- Hidaka H, Inagaki M, Kawamoto S, Sasaki Y. Biochemistry 1984;23:5036–41.
- Hines AC, Cole PA. Bioorg Med Chem Lett 2004;14:2951–4.
- Hjelmquist G, Andersson J, Edlund B, Engstroom L. Biochem Biophys Res Commun 1974;61:559–63.
- de la Houssaye BA, Masaracchia RA. Anal Biochem 1983;128:54–9.
- Parang K, Till JH, Ablooglu AJ, Kohanski RA, Hubbard SR, Cole PA.Nat Struct Biol 2001;8:37–41.
- Kelly JL, Mclean EW, Crouth RC, Averett DR, Tuttle JV. J Med Chem 1995;38:1005–14.
- Wielgus-Kutrowska B, Antosiewicz JM, Dlugosz M, Holý A, Bzowska A. Biophys Chem 2007;125:260–8.
- Parks RE Jr, Stoeckler JD, Cambor C, Savarese TM, Crabtree GW, Chu S-H. Purine nucleoside phosphorylase and 5′-methylthioadenosine phosphorylase: targets of chemotherapy. In: Sartorelli A, Lazo JS, Bertino JR, eds. Molecular Actions and Targets for Cancer Chemotherapeutic Agents. New York: Academic Press, 1981:229.
- Kazmers IS, Mitchell BS, Dadonna PE, Watring LL, Townsend LB, Kelley WN. Science 1981;214:1137–9.
- Tuttle JV, Krenitsky TA. J Biol Chem 1984;259:4065–9.
- Krenitsky TA, Tuttle JV, Miller WH, Moorman AR, Orr GF, Beauchamp L. J Biol Chem 1990;265:3066–9.
- Nakamura CE, Chu S-H, Stoeckler JD, Parks RE Jr. Nucleos Nucleot Nucl 1989;8:1039–43.
- Halazy S, Ehrhard A, Danzin C. J Am Chem Soc 1991;113:315–17.
- Ealick SE, Babu YS, Bugg CE, Erion MD, Guida WC, Montgomery JA, et al. Proc Natl Acad Sci USA 1991;88:11540–4.
- Kelley JL, Linn JA, McLean EW, Tuttle JV. J Med Chem 1993;36:3455–63.
- Mannisto PT, Ulmanen I, Lundström K, Taskinen J, Tenhunen J, Tilgmann C, et al. Prog Drug Res 1992;39:291–350.
- Nackley AG, Tan KS, Fecho K, Flood P, Diatchenko L, Maixner W. Pain 2007;128:199–208.
- Anderson GL, Bussolitti DL, Coward JK. J Med Chem1981;24:1271–7.
- Burns MR, Coward JK. Bioorg Med Chem 1996;4:1455–70.
- Borgulya J, Da Prada M, Dingemanse R, Scherschlich B, Schläppi B, Zücher G. Drugs Future 1991;16:719–21.
- Masjost B, Ballmer P, Borroni E, Zürcher G, Winkler FK, Jakob-Roetne R, et al. Chem Eur J 2000;6:971–82.
- Vidgren J, Svensson LA, Liljas A. Nature 1994;368:354–8.
- Lerner C, Masjost B, Ruf A, Gramlich V, Jakob-Roetne R, Zürcher G, et al. Org Biomol Chem 2003;1:42–9.
- Lerner C, Ruf A, Gramlich V, Masjost B, Zürcher G, Jakob-Roetne R, et al. Angew Chem 2001;40:4040–2.
- Paulini R, Lerner C, Jakob-Roetne R, Zürcher G, Borroni E, Diederich F. Chembiochem 2004;5:1270–4.
- Smith KS, Smith PL, Heady TN, Trugman JM, Harman WD, Macdonald TL. Chem Res Toxicol 2003;16:123–8.
- Korlipara LVP, Cooper JM, Schapira AHV. Neuropharmacology 2004;46:562–9.
- Bonifacio MJ, Archer M, Rodrigues ML, Matias PM, Learmonth DA, Carrondo MA, et al. Mol Pharmacol 2002;62:795–805.
- Kappler F, Hai TT, Hampton A. J Med Chem 1986;29:318–22.
- Kappler F, Vrudhula VM, Hampton A. J Med Chem 1987;30:1599–603.
- Vrudhula VM, Kappler F, Afshar C, Ginell SL, Lessinger L, Hampton A. J Med Chem 1989;32:885–90.
- Kappler F, Vrudhula VM, Hampton A. J Med Chem 1988;31:384–9.
- Kappler F, Hampton A. J Med Chem 1990;33:2545–51.
- Benghiat E, Crooks PA. J Med Chem 1983;26:1470–7.
- Cole C, Foster AJ, Freeman S, Jaffar M, Murray PE, Stratford IJ. Anticancer Drug Des 1999;14:383–92.
- Haraguchi M, Miyadera K, Uemura K, Sumizawa T, Furukawa T, Yamada K, et al. Nature 1994;368:198.
- Takeuchi M, Otsuka T, Matsui N, Asai K, Hirano T, Moriyama A, et al. Arthritis Rheum 1994;37:662–72.
- Creamer D, Jaggar R, Allen M, Bicknell R, Barker J. Br J Dermatol 1997;137:851–5.
- Iltzsch MH, el Kouni MH, Cha S. Biochemistry 1985;24:6799–807.
- Balzarini J, Degrève B, Estan-Gamboa A, Esnouf R, De Clercq E, Engelborghs Y, et al. FEBS Lett 2000;483:181–5.
- Allan AL, Gladstone PL, Price ML, Hopkins SA, Juarez JC, Donate F, et al..J Med Chem 2006;49:7807–15.
- Matsushita S, Nitanda T, Furukawa T, Sumizawa T, Tani A, Nishimoto K, et al. Cancer Res 1999;59:1911–16.
- Palcic MM, Heerze LD, Srivastava OP, Hindsgaul O. J Biol Chem 1989;264:17174–81.
- Hashimoto H, Endo T, Kajihara Y..xxx.J Org Chem 1997;62:1914–15.
- Gautier-Lefebvre I, Behr JB, Guillerma G, Ryder NS. Bioorg Med Chem Lett 2000;10:1483–6.
- Lau JTY, Wuensch SA. In: Ernst B, Hart GW, Sinaÿ P, eds. Carbohydrates in Chemistry and Biology. Weinheim: Wiley-VCH, 2000;3:213–26.
- Stolz F, Blume A, Hinderlich S, Reutter W, Schmidt RR. Eur J Org Chem 2004;15:3304–12.
- Schafer A, Thiem J. J Org Chem 2000;65:24–9.
- Luengo JI, Gleason JG. Tetrahedron Lett 1992;33:6911–14.
- Orbe M, Claesson A. Eur J Med Chem 1989;24:447–51.
- Norbeck DW, Kramer JB, Lartey PA. J Org Chem 1987;52:2174–9.
- Schmidt RR, Frische K. Bioorg Med Chem Lett 1993;3:1747–50.
- Vaghefi MM, Bernacki RJ, Dalley NK, Wilson BE, Robins RK. J Med.Chem 1987;30:1383–91.
- Schworer R, Schmidt RR. J Am Chem Soc 2002;124:1632–7.
- Hinou H, Sun X-L, Ito Y. J Org Chem 2003;68:5602–13.
- Izumi M, Wada K, Yuasa H, Hashimoto H. J Org Chem 2005;70:8817–24.
- Izumi M, Kaneko S, Yuasa H, Hashimoto H. Org Biomol Chem 2006;4:681–90.
- Brockhausen I, Carver JP, Schachter H. Biochem Cell Biol 1988;66:1134–51.
- Cummings RD, Trowbridge IS, Kornfeld S. J Biol Chem 1982;257:13421–7.
- Dennis JW, Granovsky M, Warren CE. Biochim Biophys Acta 1999;1473:21–34.
- Dennis JW, Laferte S, Waghorne C, Breitman ML, Kerbel RS. Science 1987;236:582–5.
- Ihara S, Miyoshi E, Ko J, Murata K, Nakahara S, Honke K, et al. J Biol Chem 2002;277:16960–7.
- Demetriou M, Nabi IR, Oppolino M, Dedhar S, Dennis JW. J Cell Biol 1995;130:383–92.
- Guo HB, Lee I, Kamar M, Akiyama SK, Pierce M. Cancer Res 2002;62:6837–45.
- Saito T, Miyoshi E, Sasai K, Nakano N, Eguchi H, Honke K, et al. J BiolChem 2002;277:17002–8.
- Hanashima S, Manabe S, Inamori KI, Taniguchi N, Ito Y. Chem Eur J 2006;12:3449–62.
- Tvaroska I, André I, Carver JP. J Am Chem Soc 2000;122:8762–76.
- Tahir SH, Hindsgaul O. Can J Chem 1986;64:1771–80.
- De Angelis J, Gastel J, Klein DC, Cole PA. J Biol Chem 1998;273:3045–50.
- Kim CM, Cole PA. J Med Chem 2001;44:2479–85.
- Khalil EM, Cole PA. J Am Chem Soc 1998;120:6195–6.
- Khalil EM, De Angelis J, Ishii M, Cole PA. Proc Natl Acad Sci USA 1999;96:12418–23.
- Zheng W, Cole PA. Bioorg Chem 2003;31:398–411.
- Frisch SM, Mymryk JS. Nat Rev Mol Cell Biol 2002;3:441–52.
- Timmermann S, Lehrmann H, Polesskaya A, Harel-Bellan A. Cell Mol Life Sci 2001;58:728–36.
- Gayther SA, Batley SJ, Linger L, Bannister A, Thorpe K, Chin SF, et al. Nat Genet 2000;24:300–3.
- Deguchi K, Ayton PM, Carapeti M, Kutok JL, Snyder CS, Williams IR, et al. Cancer Cell 2003;3:259–71.
- Lau OD, Kundu TK, Soccio RE, Ait-Si-Ali S, Khalil EM, Vassilev A, et al. Mol Cell 2000;5:589–95.
- Lau OD, Courtney AD, Vassilev A, Marzilli LA, Cotter RJ, Nakatani Y, et al. J Biol Chem 2000;275:21953–9.
- Thompson PR, Kurooka H, Nakatani Y, Cole PA. J Biol Chem 2001; 276:33721–9.
- Sagar V, Zheng W, Thompson PR, Cole PA. Bioorg Med Chem 2004;12:3383–90.
- Cebrat M, Kim CM, Thompson PR, Daugherty M, Cole PA. Bioorg Med Chem 2003;11:3307–13.
- Wright GD, Berghuis AM, Mobashery S. Aminoglycoside antibiotics: structures, functions and resistance. In: Rosen BP, Mobashery S, eds. Resolving the Antibiotic Paradox: Progress in Understanding Drug Resistance and Development of New Antibiotics. New York: Plenum, 1998:27.
- Magnet S, Blanchard JS. Chem Rev 2005;105:477–97.
- Auclair K, Gao F, Yan X. US Patent Application 11/359 274, filed February 21 2006.
- Gao F, Yan X, Baettig OM, Berghuis AM, Auclair K. Angew Chem Int Ed 2005;44:6859–62.
- Wright GD, Ladak P. Antimicrob Agents Chemother 1997;41:956–60.
- Gao F, Yan X, Shakya T, Baettig OM, Ait-Mohand-Brunet S, Berghuis AM, et al. J Med Chem 2006;49:5273–81.
- Liu M, Haddad J, Azucena E, Kotra LP, Kirzhner M, Mobashery S. J Org Chem 2000;65:7422–31.
- Lipscomb WN. Adv Enzymol Relat Areas Mol Biol 1994;68:67–151.
- Laing N, Chan WW-C, Hutchinson DW, öberg B. FEBS Lett 1990;260:206–8.
- Dutta PL, Foye WO. J Pharm Sci 1990;79:447–52.
- Swyryd EA, Seaver SS, Starkv GR. J Biol Chem 1974;246:6945–50.
- Collins KD, Startk GR. J Biol Chem1971;246:6599–605.
- Newell JO, Markby DW, Schachman HK. J Biol Chem 1989;264:2476–81.
- Howlett GJ, Schachman HK. Biochemistry 1977;16:5077–83.
- Endrizzi JA, Beernink PT, Alber T, Schachman HK. Proc Natl Acad Sci USA 2000;97:5077–82.
- Van Boxstael S, Cunin R, Khan S, Maes D. J Mol Biol 2003;326:203–16.
- Krause KL, Volz KW, Lipscomb WN. Proc Natl Acad Sci USA 1985;82:1643–7.
- Grison C, Coutrot P, Comoy C, Balas L, Joliez S, Lavecchia G, et al. Eur J Med Chem 2004;39:333–44.
- Bowman KG, Bertozzi CR. Chem Biol 1999;6:R9–22.
- Kehoe JW, Bertozzi CR. Chem Biol 2000;7:R57–61.
- Falany CN. FASEB J 1997;11:206–16.
- Kakuta Y, Pedersen LG, Pedersen LC, Negishi M. Trends Biochem Sci 1998;23:129–30.
- Armstrong JI, Ge X, Verdugo DE, Winans KA, Leary JA, Bertozzi CR. Org Lett 2001;3:2657–60.
- Armstrong JI, Verdugo DE, Bertozzi CR. J Org Chem 2003;68:170–3.
- Zhang FL, Casey PJ. Annu Rev Biochem 1996;65:241–69.
- Fu HW, Casey PJ. Recent Prog Horm Res 1999;54:315–43.
- Reiss Y, Goldstein JL, Seabra MC, Casey PJ, Brown MS. Cell 1990;62:81–8.
- Gibbs JB. Cell 1991;65:1–4.
- Graham SL, deSolms SJ, Guiliani EA, Kihl NE, Mosser SD, Oliff AI, et al. J Med Chem 1994;37:725–32.
- Pompliano DL, Rands E, Schaber MD, Mosser SD, Anthony NJ, Gibbs JB. Biochemistry 1992;31:3800–7.
- Singh SB, Zink DL, Liesch JM, Goetz MA, Jenkins RG, Nallin-Olmstead M, et al. Tetrahedron 1993;49:5917–26.
- Bhide RS, Patel DV, Patel MM, Robinson SP, Hunihan LW, Gordon EM. Bioorg Med 2Chem Lett 1994;4:2107–12.
- Patel DV, Gordon EM, Schmidt Harold RJ, Weller N, Young MG, Zahler R, et al. J Med Chem 1995;38:435–42.
- Patel DV, Young MG, Robinson SP, Hunihan LW, Dean BJ, Gordon EM. J Med Chem 1996;39:4197–210.
- Reynolds JEF, ed. Martindale: The Extra Pharmacopoeia, 31st ed. London: Royal Pharmaceutical Society of Great Britain, 1996:821.
- Schlitzer M, Sattler I. Eur J Med Chem 2000;35:721–6.
- Schlitzer M, Böhm M, Sattler I, Dahse HM. Bioorg Med Chem 2000;8:1991–2006.
- Schlitzer M, Böhm M, Sattler I. Bioorg Med Chem 2000;8:2399–406.
- Schlitzer M, Sattler I. Bioorg Med Chem 1999;7:2391–5.
- Mitsch A, Bergemann S, Gust R, Sattler I, Schlitzer M. Arch Pharm Pharm Med Chem 2003;336:242–50.
- Schlitzer M, Böhm M, Sattler I. Bioorg Med Chem 2002;10:615–20.
- Zhang H. Structure 2003;11:237–9.
- Reid TS, Terry KL, Casey PJ, Beese LS. J Mol Biol 2004;343:417–33.
- Casey P, Thissen JA, Moomaw JF. Proc Natl Acad Sci USA 1991;88:8631–5.
- Yokoyama K, Goodwin GW, Ghomaschi F, Glomset JA, Gelb MH. Proc Natl Acad Sci USA 1991;88:5302–6.
- El Oualid F, Baktawar J, Leroy IM, van den Elst H, Cohen LH, van der Marel GA, et al. Bioorg Med Chem 2005;13:1463–75.
- El Oualid F, Bruining L, Leroy IM, Cohen LH, van Boom JH, van der Marel GA, et al. Helv Chim Acta 2002;85:3455–72.
- Plaut GWE, Smith CM, Alworth WL. Annu Rev Biochem 1974;43:899–922.
- Plaut GWE. In: Florkin M, Stotz EH, eds. Comprehensive Biochemistry. Amsterdam: Elsevier, 1971;21:11.
- Bacher A, Ladenstein R. In: Müller F, ed. Chemistry and Biochemistry of Flavoenzymes. Boca Raton, FL: Chemical Rubber Co., 1991;II:293.
- Cushman M, Mavandadi F, Yang D, Kugelbrey K, Kis K, Bacher A. J Org Chem 1999;64:4635–42.
- Saridakis V, Christendat D, Kimber MS, Dharamsi A, Edwards AM, Pai EF. J Biol Chem 2001;276:7225–32.
- Sorci L, Cimadamore F, Scotti S, Petrelli R, Cappellacci L, Franchetti P, et al. Biochemistry 2007;46:4912–22.
- Cleland WW. Adv Enzymol Relat Areas Mol Biol 1977;45:273–87.
- Bose R, Holbert MA, Pickin KA, Cole PA. Curr Opin Struct Biol 2006;16:668–75.
- Vazquez J, Tautz L, Ryan JJ, Vuori K, Mustelin T, Pellecchia M. J Med Chem 2007;50:2137–43.
- Hines AC, Parang K, Kohanski RA, Hubbard SR, Cole PA. Bioorg Chem 2005;33:285–97.