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Research Article

Inhibition of Serine Proteinases by P-Carbethoxyphenyl Esters of ϵ-Guanidino- And ϵ-Amino Caproic Acid: Thermodynamic and Molecular Modeling Study

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Pages 249-259 | Received 30 Mar 1988, Published online: 27 Sep 2008

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  • Amino acid residues have been identified by their three-letter code and by their sequence number. The numbering of human Lys77-plasmin refers to that of the complete form (Glu1) of human plasminogen.13 The numbering of bovine factor xa refers to that of its heavy chain.12 The numbering of bovine α-thrombin, bovineβ-trypsin, porcine pancreatic β-kallikrein-B and human urinary kallikrein refers to that of bovine chymotrypsinogens A and B.11. The numbering of the Mr 54,000 species of human urokinase refers to that of the single-chain pro-urokinase.15
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