85
Views
0
CrossRef citations to date
0
Altmetric
Research Article

Expert Design and Desirability Function Approach for the Development of Diazepam Thermally Sensitive Rectal Gel

, , , &
Pages 813-830 | Received 23 Oct 2019, Accepted 26 Nov 2019, Published online: 18 Dec 2019

References

  • Vijay DH , AdhikraoVY , RemethJDet al. Rectal suppository as an effective alternative for oral administration. Res. J. Pharm. Tech.8(6), 759–766 (2015).
  • Alejandro S , Josedas N , BrunoS. Mucoadhesive polymers in the design of nano-drug-delivery systems for administration by non-parenteral routes: a review. Prog. Poly. Sci.39(12), 2030–2075 (2014).
  • Younsoo B , KazunoriK. Intelligent polymeric micelles from functional poly(ethylene glycol)-poly(amino acid) block copolymers. Adv. Drug Deliv. Rev.61(10), 768–784 (2009).
  • Enrica C , VitaliyVKH. Biomedical applications of hydrogels: a review of patents and commercial products. Eur. Poly. J.65, 252–267 (2015).
  • Fang L , SejalR , HannahKBet al. Patient-centered pharmaceutical design to improve acceptability of medicines: similarities and differences in paediatric and geriatric populations. Drugs74(16), 1871–1889 (2014).
  • Barar FSK . Essentials of Pharmacotherapeutics.S. Chand Publishing. Rum Nagar, New Dehli, 540–555 (2000).
  • Bruce JA . Novel formulation strategies for improving oral bioavailability of drugs with poor membrane permeation or presystemic metabolism. J. Pharm. Sci.82(10), 979–987 (1993).
  • Han-Gon C , Jae-HeeJ , Jei-ManR , Sung-JuneY , Yu-KyoungO , Chong-KookK. Development of in situ-gelling and mucoadhesive acetaminophen liquid suppository. Int. J. Pharm.165(1), 33–44 (1998).
  • Keny RV , LourencoCF. Gelling and mucoadhesive diltiazem hydrochloride liquid suppository. Int. J. Pharm. Bio. Sci.1, 1 (2010).
  • El-Leithy ES , ShakerDS , GhorabMK , Abdel-RashidRS. Evaluation of mucoadhesive hydrogels loaded with diclofenac sodium–chitosan microspheres for rectal administration. AAPS Pharm. Sci. Tech.11(4), 1695–1702 (2010).
  • Dodov MG , GoracinovaK , SimonoskaM , Trajkovic-JolevskaS , RibarskaJT , MitevskaMD. Formulation and evaluation of diazepam hydrogel for rectal administration. ACTA Pharm. Zagreb.55(3), 251 (2005).
  • Christian EE , DieterS. Modern management of epilepsy: a practical approach. Epilepsy Behav.12(4), 501–539 (2008).
  • Rashmin BP , MrunaliRP , KashyapKB , BharatGP. Formulation consideration and characterization of microemulsion drug-delivery system for transnasal administration of carbamazepine. Bull. Fac. Pharm. Cairo Univ.51(2), 243–253 (2013).
  • Judith J , GillesLF , DouglasBCet al. Clinical practice guidelines for the sustained use of sedatives and analgesics in the critically ill adult. Crit. Car. Med.30(1), 119–141 (2002).
  • Ghada A , RaniaHF. Diazepam-loaded solid lipid nanoparticles: design and characterization. AAPS Pharm. Sci. Tech.10(1), 211–219 (2009).
  • Matthew M , DavidB , AmyS , KathrynB , LondonK , HyunahC. Hydrogel-based drug-delivery systems for poorly water-soluble drugs. Molecules20(11), 20397–20408 (2015).
  • Eve RG , Jean-ChristopheL. In situ-forming hydrogels – review of temperature-sensitive systems. Eur. J. Pharm. Biopharm.58(2), 409–426 (2004).
  • Schmolka IR . Artificial skin. I. Preparation and properties of pluronic F-127 gels for treatment of burns. J. Biom. Mater. Res.6(6), 571–582 (1972).
  • Yun M , ChoiH , JungJ , KimC. Development of a thermo-reversible insulin liquid suppository with bioavailability enhancement. Int. J. Pharm.189(2), 137–145 (1999).
  • Chul Soon Y , JinSuck C , Qi-ZheQet al. Effect of sodium chloride on the gelation temperature, gel strength and bioadhesive force of poloxamer gels containing diclofenac sodium. Int. J. Pharm.226(1-2), 195–205 (2001).
  • Muruganantham V. Design and evaluation of buccal tablets of drug loaded microspheres. Vinayaka Missions University, Tamil nadu, India (2016).
  • Lorenzo L , RobertoM , FrancoP , CarloV. Pharmaceutical compositions comprising imidazoquinolin (amines) and derivatives thereof suitable for local administration. Google Patents, US14/752,358 (2015).
  • Susan RM , GaryDS , PeterELet al. Formulation and in-vitro and in-vivo evaluation of a mucoadhesive gel containing freeze dried black raspberries: implications for oral cancer chemoprevention. Pharm. Res.24(4), 728–737 (2007).
  • Seung-Kyum C , RamanaG , RobertAC. Reliability-Based Structural Design. Springer Science & Business Media, London, UK (2006).
  • Mohd Yusof N , VasishtCV , SharifS , EltingS , AbuA. Application of response surface methodology in describing the performance of coated carbide tools when turning AISI 1045 steel. J. Mat. Pro. Tech.145(1), 46–58 (2004).
  • Margareth RCM , RaimarL , MayA. Simulated biological fluids with possible application in dissolution testing. Disso. Technol.18(3), 15–28 (2011).
  • Saurabh SS , NandhibatlaVS , VinodKA , PremSG. Micellar structure of silicone surfactants in water from surface activity, SANS and viscosity studies. J. Physic. Chem.106(10), 2606–2617 (2002).
  • Susan CM , BernadetteRD. Rheological properties of poloxamer vehicles. Int. J. Pharm.18(3), 269–276 (1984).
  • Carretero MI , ManuelP. Clay and non-clay minerals in the pharmaceutical industry: part I. Excipients and medical applications. Appl. Clay Sci.46(1), 73–80 (2009).
  • Sambhaji SP , AnantRP , KakasahebRM , ShivajiraoSK. Pluronic gels for nasal delivery of vitamin B12. Part I: preformulation study. Int. J. Pharm.270(1-2), 37–45 (2004).
  • Maja Radivojša M , JulijanaK , PegiAhlin G. Thermoresponsive polymers: insights into decisive hydrogel characteristics, mechanisms of gelation, and promising biomedical applications. Int. J. Pharm.472(1-2), 262–275 (2014).
  • Jay L , BenediktV , SergioGDet al. Controlled-release cns modulating compositions and methods for the treatment of otic disorders. Google Patents, W02010011466A2 (2009).
  • Choi YM , JungKC , JoHMet al. Combined effects of potassium lactate and calcium ascorbate as sodium chloride substitutes on the physicochemical and sensory characteristics of low-sodium frankfurter sausage. Meat. Sci.96(1), 21–25 (2014).
  • Jeong B , KimSW , BaeYH. Thermosensitive sol–gel reversible hydrogels. Adv. Drug Deliv. Rev.64, 154–162 (2012).
  • Escobar-Chávez JJ , López-CervantesM , NaïkA , KaliaYN , Quintanar-GuerreroD , Ganem-QuintanarA. Applications of thermo-reversible pluronic F-127 gels in pharmceutical formulations. J. Pharm. Pharm. Sci.9(3), 339–358 (2006).
  • Giulia B , MarcoC , GiovannaM , GianfabioG , GiovanniFilippo P. Thermosensitive self-assembling block copolymers as drug-delivery systems. Polymers3(2), 779–811 (2011).
  • Waikar SS , SabbisettiVS , BonventreJV. Normalization of urinary biomarkers to creatinine during changes in glomerular filtration rate. Kidn. Int.78(5), 486–494 (2010).
  • Jantzen JP , IreneT , PeterKW , AnkeMK. Rectal pH in children. Can. J. Anaesthes.36(6), 665–667 (1989).
  • Chung JOL . Novel injectable interpenetrating polymer network as a semi-permanent injectable implant for soft tissue augmemtation. University of California, Los Angeles, CA, USA (2015).
  • Rafi M , TarunG , AmitKG , GoutamR. Polymeric nanofibers: targeted gastro-retentive drug-delivery systems. J. Drug Tar.23(2), 109–124 (2015).
  • Jaspreet Kaur V , KaustubhT , SanjayG. Bioadhesive microspheres as a controlled drug-delivery system. Int. J. Pharm.255(1-2), 13–32 (2003).
  • Cristina M , AránzazuZ , JoséML. Critical factors in the release of drugs from sustained release hydrophilic matrices. J. Control. Rel.154(1), 2–19 (2011).
  • Peppas NA , BuresP , LeobandungWS , IchikawaH. Hydrogels in pharmaceutical formulations. Eur. J. Pharm. Biopharm.50(1), 27–46 (2000).
  • Laura ME , RichardC , JustinH. Oral drug delivery with polymeric nanoparticles: the gastrointestinal mucus barriers. Adv. Drug Deliv. Rev.64(6), 557–570 (2012).
  • Michele M , AliR , TaherianH , RamaswamyHS. Rheological properties of selected hydrocolloids as a function of concentration and temperature. Food Res. Int.34(8), 695–703 (2001).
  • Byeongtaek O , ChiHL. Nanofiber for cardiovascular tissue engineering. Exp. Opin. Drug Deliv.10(11), 1565–1582 (2013).
  • Qi H , ChenW , HuangCet al. Development of a poloxamer analogs/carbopol-based in situ gelling and mucoadhesive ophthalmic delivery system for puerarin. Int. J. Pharm.337(1-2), 178–187 (2007).
  • Amir F , MartaC , AlexanderS. Thermogelling properties of purified poloxamer 407. Heliyon3(8), E00390 (2017).
  • Kumar R , KatareOP. Lecithin organogels as a potential phospholipid-structured system for topical drug delivery: a review. AAPS Pharm. Sci. Tech.6(2), E298–E310 (2005).
  • Baloglu E , SenyigitZA , KaravanaSY , Bernkop-SchnürchA. Strategies to prolong the intravaginal residence time of drug-delivery systems. J. Pharm. Pharm. Sci.12(3), 312–336 (2009).
  • Sara S . Nanoparticles as potential tools for improved antioxidant enzyme delivery. J. Adv. Chem. Pharm. Mat.1(3), 65–66 (2018).
  • Mohammad M , SaraS , AhmadYKh. Natural low-and high-density lipoproteins as mighty bio-nanocarriers for anticancer drug delivery. Cancer Chemotherap. Pharmaco.82(3), 371–382 (2018).

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.