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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 33, 2018 - Issue 1
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Research Paper

Design, synthesis, in vitro antiproliferative activity and apoptosis-inducing studies of 1-(3′,4′,5′-trimethoxyphenyl)-3-(2′-alkoxycarbonylindolyl)-2-propen-1-one derivatives obtained by a molecular hybridisation approach

Delia PretiDepartment of Chemical and Pharmaceutical Sciences, University of Ferrara, Ferrara, Italy; View further author information
,
Romeo RomagnoliDepartment of Chemical and Pharmaceutical Sciences, University of Ferrara, Ferrara, Italy; Correspondence[email protected]
View further author information
,
Riccardo RondaninDepartment of Chemical and Pharmaceutical Sciences, University of Ferrara, Ferrara, Italy; View further author information
,
Barbara CacciariDepartment of Chemical and Pharmaceutical Sciences, University of Ferrara, Ferrara, Italy; View further author information
,
Ernest HamelScreening Technologies Branch, Developmental Therapeutics Program, Division of Cancer Treatment and Diagnosis, Frederick National Laboratory for Cancer Research, National Cancer Institute, National Institutes of Health, Frederick, MD, USA; View further author information
,
Jan BalzariniRega Institute for Medical Research, KU Leuven, Laboratory of Virology and Chemotherapy, Leuven, Belgium; View further author information
,
Sandra LiekensRega Institute for Medical Research, KU Leuven, Laboratory of Virology and Chemotherapy, Leuven, Belgium; View further author information
,
Dominique ScholsRega Institute for Medical Research, KU Leuven, Laboratory of Virology and Chemotherapy, Leuven, Belgium; View further author information
,
Francisco Estévez-SarmientoDepartment of Biochemistry and Molecular Biology, Research Institute in Biomedical and Health Sciences (IUIBS), University of Las Palmas de Gran Canaria (ULPGC), SpainView further author information
,
José QuintanaDepartment of Biochemistry and Molecular Biology, Research Institute in Biomedical and Health Sciences (IUIBS), University of Las Palmas de Gran Canaria (ULPGC), SpainView further author information
&
Francisco EstévezDepartment of Biochemistry and Molecular Biology, Research Institute in Biomedical and Health Sciences (IUIBS), University of Las Palmas de Gran Canaria (ULPGC), SpainView further author information
 show all
Pages 1225-1238 | Received 23 Apr 2018, Accepted 21 Jun 2018, Published online: 24 Aug 2018

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