Supplemental material
Open access
991
Views
4
CrossRef citations to date
0
Altmetric
Research Paper
Further validation of strecker-type α-aminonitriles as a new class of potent human carbonic anhydrase II inhibitors: hit expansion within the public domain using differential scanning fluorimetry leads to chemotype refinement
Mikhail Krasavina Saint Petersburg State University, Saint Petersburg, Russian FederationCorrespondence[email protected]
View further author information
, View further author information
Stanislav Kalinina Saint Petersburg State University, Saint Petersburg, Russian FederationView further author information
, Sergey Zozulyab Enamine Ltd, Kyiv, Ukraine;c Taras Shevchenko National University, Kyiv, UkraineView further author information
, Anastasia Griniukovab Enamine Ltd, Kyiv, UkraineView further author information
, Petro Boryskob Enamine Ltd, Kyiv, UkraineView further author information
, Andrea Angelid Neurofarba Department, Universita degli Studi di Firenze, Florence, Italy
https://orcid.org/0000-0002-1470-7192View further author information
Claudiu T. Supurand Neurofarba Department, Universita degli Studi di Firenze, Florence, ItalyCorrespondence[email protected]
https://orcid.org/0000-0003-4262-0323View further author information
Pages 165-171
|
Received 16 Oct 2019, Accepted 11 Nov 2019, Published online: 22 Nov 2019
Related Research Data
The coumarin-binding site in carbonic anhydrase accommodates structurally diverse inhibitors: the antiepileptic lacosamide as an example and lead molecule for novel classes of carbonic anhydrase inhibitors
Source:
American Chemical Society (ACS)
Evaluation of fluorescence-based thermal shift assays for hit identification in drug discovery.
Source:
Elsevier BV
Non-zinc mediated inhibition of carbonic anhydrases: coumarins are a new class of suicide inhibitors
Source:
American Chemical Society (ACS)
Discovery of Strecker-type α-aminonitriles as a new class of human carbonic anhydrase inhibitors using differential scanning fluorimetry.
Source:
Informa UK Limited
Carbon Dioxide Hydration Activity of Carbonic Anhydrase: Kinetics of Alkylated Anhydrases B and C from Humans
Source:
Proceedings of the National Academy of Sciences
Universal screening methods and applications of ThermoFluor.
Source:
SAGE Publications
Multiple Binding Modes of Inhibitors to Carbonic Anhydrases: How to Design Specific Drugs Targeting 15 Different Isoforms?
Source:
American Chemical Society (ACS)
Crystal structure of the catalytic domain of the tumor-associated human carbonic anhydrase IX
Source:
National Academy of Sciences
Related research
People also read lists articles that other readers of this article have read.
Recommended articles lists articles that we recommend and is powered by our AI driven recommendation engine.
Cited by lists all citing articles based on Crossref citations.
Articles with the Crossref icon will open in a new tab.