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Research Article
Novel N-Arylmethyl-aniline/chalcone hybrids as potential VEGFR inhibitors: synthesis, biological evaluations, and molecular dynamic simulations
Hesham Haffeza Biochemistry and Molecular Biology Department, Faculty of Pharmacy, Helwan University, Cairo, Ain Helwan, Egypt;b Center of Scientific Excellence “Helwan Structural Biology Research, (HSBR)”, Helwan University, Cairo, Egypthttps://orcid.org/0000-0002-9924-2063
, Nosaiba A. Elsayedc Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Helwan University, Cairo, Ain Helwan, Egypt
, Marwa F. Ahmedc Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Helwan University, Cairo, Ain Helwan, Egypt
, Samar S. Fatahalad Pharmaceutical Organic Chemistry Department, Faculty of Pharmacy, Helwan University, Cairo, Egypt
, Eman F. Khaleele Department of Medical Physiology, College of Medicine, King Khalid University, Asir, Saudi Arabia
, Rehab Mustafa Badie Department of Medical Physiology, College of Medicine, King Khalid University, Asir, Saudi Arabia
, Eslam B. Elkaeedf Department of Pharmaceutical Sciences, College of Pharmacy, AlMaarefa University, Riyadh, Saudi Arabia
, Mahmoud A. El Hassabg Department of Medicinal Chemistry, Faculty of Pharmacy, King Salman International University (KSIU), South Sinai, Egypt
, Sherif F. Hammadc Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Helwan University, Cairo, Ain Helwan, Egypt;h Medicinal Chemistry Department, PharmD Program, Egypt-Japan University of Science and Technology (E-JUST), New Borg El-Arab City, Egypt Alexandria
, Wagdy M. Eldehnai Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, Egypthttps://orcid.org/0000-0001-6996-4017
, Nicolas Masurierj Institut des Biomolécules Max Mousseron (IBMM), UMR 5247, CNRS, Université de Montpellier, ENSCM, Montpellier, Francehttps://orcid.org/0000-0001-9169-8149
& Radwan El-Haggarc Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Helwan University, Cairo, Ain Helwan, EgyptCorrespondence[email protected]
https://orcid.org/0000-0002-3878-9890
show allhttps://orcid.org/0000-0002-3878-9890
Article: 2278022
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Received 25 Aug 2023, Accepted 25 Oct 2023, Published online: 20 Nov 2023
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