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Research Article

Preparation and Analgesic Activity of Eudragit RS100® Microparticles Containing Diflunisal

Pages 35-45 | Published online: 29 Sep 2008

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Mahmoud A. Younis, Marwa R. El-Zahry, Mahmoud A. Tallat & Hesham M. Tawfeek. (2020) Sulpiride gastro-retentive floating microsponges; analytical study, in vitro optimization and in vivo characterization. Journal of Drug Targeting 28:4, pages 386-397.
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Rosario Pignatello, Tiziana M. G. Pecora, Giuseppa G. Cutuli, Alfio Catalfo, Guido De Guidi, Barbara Ruozi, Giovanni Tosi, Simona Cianciolo & Teresa Musumeci. (2019) Antioxidant activity and photostability assessment of trans-resveratrol acrylate microspheres. Pharmaceutical Development and Technology 24:2, pages 222-234.
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Nazila Jafari-Aghdam, Khosro Adibkia, Shahriar Payab, Mohammad Barzegar-Jalali, Alireza Parvizpur, Ghobad Mohammadi & Araz Sabzevari. (2016) Methylprednisolone acetate–Eudragit® RS100 electrospuns: Preparation and physicochemical characterization. Artificial Cells, Nanomedicine, and Biotechnology 44:2, pages 497-503.
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Tatiele Katzer, Paula Chaves, Andressa Bernardi, Adriana Pohlmann, Silvia S. Guterres & Ruy Carlos Ruver Beck. (2014) Prednisolone-loaded nanocapsules as ocular drug delivery system: development, in vitro drug release and eye toxicity. Journal of Microencapsulation 31:6, pages 519-528.
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Sachin S. Pandit, Dinesh P. Hase, Manish M. Bankar, Arun T. Patil & Naresh J. Gaikwad. (2009) Ketoprofen-loaded Eudragit RSPO microspheres: An influence of sodium carbonate on in vitro drug release and surface topology. Journal of Microencapsulation 26:3, pages 195-201.
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Grant Heinicke & Joseph B. Schwartz. (2007) The Influence of Surfactants and Additives on Drug Release from a Cationic Eudragit Coated Multiparticulate Diltiazem Formulation. Pharmaceutical Development and Technology 12:4, pages 381-389.
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Padma V. Devarajan & Ganeshchandra S. Sonavane. (2007) Preparation and In Vitro/In Vivo Evaluation of Gliclazide Loaded Eudragit Nanoparticles as a Sustained Release Carriers. Drug Development and Industrial Pharmacy 33:2, pages 101-111.
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Rosario Pignatello, Daniela Spadaro, Maria Angela Vandelli, Flavio Forni & Giovanni Puglisi. (2004) Characterization of the Mechanism of Interaction in Ibuprofen‐Eudragit RL100® Coevaporates. Drug Development and Industrial Pharmacy 30:3, pages 277-288.
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Ghobad Mohammadi, Elham Namadi, Ali Mikaeili, Pardis Mohammadi & Khosro Adibkia. (2017) Preparation, physicochemical characterization and anti-fungal evaluation of the Nystatin-loaded Eudragit RS100/PLGA nanoparticles. Journal of Drug Delivery Science and Technology 38, pages 90-96.
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Utpal Jana, Anjan Kumar Mohanty, Prabal Kumar Manna & Guru Prasad Mohanta. (2014) Preparation and characterization of nebivolol nanoparticles using Eudragit® RS100. Colloids and Surfaces B: Biointerfaces 113, pages 269-275.
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S. Payab, N. Jafari-Aghdam, M. Barzegar-Jalali, G. Mohammadi, F. Lotfipour, T. Gholikhani & K. Adibkia. (2014) Preparation and physicochemical characterization of the azithromycin-Eudragit RS100 nanobeads and nanofibers using electrospinning method. Journal of Drug Delivery Science and Technology 24:6, pages 585-590.
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Estefanía Vega, M. Antònia Egea, M. Luisa Garduño-Ramírez, M. Luisa García, Elena Sánchez, Marta Espina & Ana Cristina Calpena. (2013) Flurbiprofen PLGA-PEG nanospheres: Role of hydroxy-β-cyclodextrin on ex vivo human skin permeation and in vivo topical anti-inflammatory efficacy. Colloids and Surfaces B: Biointerfaces 110, pages 339-346.
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Swarnali Das, Preeti K. Suresh & Rohitas Desmukh. (2010) Design of Eudragit RL 100 nanoparticles by nanoprecipitation method for ocular drug delivery. Nanomedicine: Nanotechnology, Biology and Medicine 6:2, pages 318-323.
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Ki-Seok Kim & Soo-Jin Park. (2010) Characterization and release behaviors of porous PCL/Eudragit RS microcapsules containing tulobuterol. Colloids and Surfaces B: Biointerfaces 76:2, pages 404-409.
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Rosario Pignatello, Nadia Ricupero, Claudio Bucolo, Francesco Maugeri, Adriana Maltese & Giovanni Puglisi. (2017) Preparation and characterization of Eudragit Retard nanosuspensions for the ocular delivery of cloricromene. AAPS PharmSciTech 7:1, pages E192-E198.
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R. Pignatello, C. Bucolo & G. Puglisi. (2002) Ocular Tolerability of Eudragit RS100® and RL100® Nanosuspensions as Carriers for Ophthalmic Controlled Drug Delivery. Journal of Pharmaceutical Sciences 91:12, pages 2636-2641.
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Rosario Pignatello, Claudio Bucolo, Piera Ferrara, Adriana Maltese, Antonina Puleo & Giovanni Puglisi. (2002) Eudragit RS100® nanosuspensions for the ophthalmic controlled delivery of ibuprofen. European Journal of Pharmaceutical Sciences 16:1-2, pages 53-61.
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