Citations (44)
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Vladimir N. Koshelev, Olga V. Primerova, Ludmila V. Ivanova & Vladimir G. Kutcherov. (2021) Synthesis of Triazole Derivatives with Sterically Hindered Phenol Fragments. Organic Preparations and Procedures International 53:1, pages 9-17.
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Thuc Dinh Ngoc. (2020) Synthesis and characterization of some new 1,2,3-thiadiazole and 1,2,3-selenadiazole triterpene derivatives from allobetulone and 2-oxoallobetulin. Synthetic Communications 50:11, pages 1665-1671.
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Georgeta Serban, Oana Stanasel, Eugenia Serban & Sanda Bota. (2018) 2-Amino-1,3,4-thiadiazole as a potential scaffold for promising antimicrobial agents. Drug Design, Development and Therapy 12, pages 1545-1566.
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Bakr F. Abdel-Wahab, Abdelbasset A. Farahat & Mohamed S. Bekheit. (2017) Synthetic profile of thiadiazoloquinazolines. Phosphorus, Sulfur, and Silicon and the Related Elements 192:11, pages 1165-1170.
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Sadaf J. Gilani, Suroor A. Khan, Nadeem Siddiqui, Suraj P. Verma, Pooja Mullick & Ozair Alam. (2011) Synthesis and in vitro antimicrobial activity of novel N-(6-chlorobenzo[d]thiazol-2-yl) hydrazine carboxamide derivatives of benzothiazole class. Journal of Enzyme Inhibition and Medicinal Chemistry 26:3, pages 332-340.
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Articles from other publishers (39)
Mahmut GÜR, Merve ZURNACI, Eda ALTINÖZ, Nesrin ŞENER, Çiğdem ŞAHİN, Merve ŞENTURAN, İzzet ŞENER, Muhammet ÇAVUŞ & Ergin Murat ALTUNER. (2023) Novel 1,3,4-Thiadiazole Derivatives as Antibiofilm, Antimicrobial, Efflux Pump Inhibiting Agents and Their ADMET Characterizations. Hittite Journal of Science and Engineering 10:2, pages 99-116.
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Crossref
Gizem Erensoy, Kai Ding, Chang-Guo Zhan, Gamze Çiftçi, Kemal Yelekçi, Merve Duracık, Özlem Bingöl Özakpınar, Esra Aydemir, Zübeyde Nur Yılmaz, Fikrettin Şahin, Necla Kulabaş, Esra Tatar & İlkay Küçükgüzel. (2023) Synthesis, in vitro and in silico studies on novel 3-aryloxymethyl-5-[(2-oxo-2-arylethyl)sulfanyl]-1,2,4-triazoles and their oxime derivatives as potent inhibitors of mPGES-1. Journal of Molecular Structure 1272, pages 134154.
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İrem BozbeyMerde, Gülce Taşkor Önel, Burçin Türkmenoğlu, Şule Gürsoy & Esra Dilek. (2022)
(
p
‐Chlorophenyl)‐3(2
H
)pyridazinone Derivatives: Synthesis,
in Silico
, and AChE/BChE Inhibitory Activity
. ChemistrySelect 7:38.
Crossref
Crossref
Tejaswini D. Patil & Sunil V. Amrutkar. (2022) Novel Benzotriazole Acetamide Derivatives as Benzo-Fused Five-
Membered Nitrogen-Containing Heterocycles - In silico Screening, Molecular
Docking, and Synthesis. Letters in Drug Design & Discovery 19:4, pages 337-349.
Crossref
Crossref
Ihsan A. Shehadi, Mohamad T. Abdelrahman, Mohamed Abdelraof & Huda R. M. Rashdan. (2022) Solvent-Free Synthesis, In Vitro and In Silico Studies of Novel Potential 1,3,4-Thiadiazole-Based Molecules against Microbial Pathogens. Molecules 27:2, pages 342.
Crossref
Crossref
Kishor R. Desai & Bhavin R. Patel. 2022. N-Heterocycles. N-Heterocycles
221
274
.
Merve Zurnacı, Merve Şenturan, Nesrin Şener, Mahmut Gür, Eda Altınöz, İzzet Şener & Ergin Murat Altuner. (2021) Studies on Antimicrobial, Antibiofilm, Efflux Pump Inhibiting, and ADMET Properties of Newly Synthesized 1,3,4‐Thiadiazole Derivatives**. ChemistrySelect 6:45, pages 12571-12581.
Crossref
Crossref
Sachin Kumar, Sukhbir Lal Khokra & Akash Yadav. (2021) Triazole analogues as potential pharmacological agents: a brief review. Future Journal of Pharmaceutical Sciences 7:1.
Crossref
Crossref
Yevhen Karpun, Volodymyr Parchenko, Tetiana Fotina, Denys Demianenko, Anatolii Fotin, Volodymyr Nahornyi & Natalia Nahorna. (2021) The investigation of antimicrobial activity of some s-substituted bis-1,2,4-triazole-3-thiones. Pharmacia 68:4, pages 797-804.
Crossref
Crossref
Deepali Dixit, Prabhakar Kumar Verma & Rakesh Kumar Marwaha. (2021) A review on ‘triazoles’: their chemistry, synthesis and pharmacological potentials. Journal of the Iranian Chemical Society 18:10, pages 2535-2565.
Crossref
Crossref
Tejaswini D. Patil, Sunil V. Amrutkar & Amol S. Jagdale. (2021) Design, in silico Analysis, Synthesis and Evaluation of Novel Benzofused Nitrogen Containing
Heterocyclic N-Substituted Mercaptobenzimidazole Derivatives as Potential Antimicrobial Agent. Asian Journal of Organic & Medicinal Chemistry 6:2, pages 121-127.
Crossref
Crossref
Zhi-Ming Cui, Bo-Hang Zhou, Chao Fu, Liu Chen, Juan Fu, Fang-Jun Cao, Xin-Juan Yang & Le Zhou. (2020)
Simple Analogues of Quaternary Benzo[
c
]phenanthridine Alkaloids: Discovery of a Novel Antifungal 2-Phenylphthalazin-2-ium Scaffold with Excellent Potency against Phytopathogenic Fungi
. Journal of Agricultural and Food Chemistry 68:52, pages 15418-15427.
Crossref
Crossref
N. R. Darekar, B. K. Karale, H. N. Akolkar & A. S. Burungale. (2020) Microwave Assisted Synthesis and Antibacterial Activity of New
1,3,4-Thiadiazoles and 1,2,4-Triazoles Derived from
2-{2-[2-(4-Fluorophenyl)-4-methylthiazol-5-yl]-1H-benzo[d]imidazol-1-yl}acetohydrazide. Russian Journal of General Chemistry 90:9, pages 1721-1726.
Crossref
Crossref
Georgiana-Oana Turcan-Trofin, Mirela-Fernanda Zaltariov, Gheorghe Roman, Sergiu Shova, Nicoleta Vornicu, Mihaela Balan-Porcarasu, Dragos Lucian Isac, Andrei Neamtu & Maria Cazacu. (2019) Amphiphilic silicone-bridged bis-triazoles as effective, selective metal ligands and biologically active agents in lipophilic environment. Journal of Molecular Liquids 294, pages 111560.
Crossref
Crossref
Muhammad Taha, Noor Barak Almandil, Umer Rashid, Muhammad Ali, Mohamed Ibrahim, Mohammed Gollapalli, Ashik Mosaddik & Khalid Mohammed Khan. (2019) 2,5-Disubstituted thiadiazoles as potent β-glucuronidase inhibitors; Synthesis, in vitro and in silico studies. Bioorganic Chemistry 91, pages 103126.
Crossref
Crossref
Ankit Jain & Poonam Piplani. (2019) Exploring the Chemistry and Therapeutic Potential of Triazoles: A Comprehensive Literature Review. Mini-Reviews in Medicinal Chemistry 19:16, pages 1298-1368.
Crossref
Crossref
Batirbay Torambetov, Shaxnoza Kadirova, Turdibek Toshmurodov, Jamshid Mengnorovich Ashurov, Nusrat Agzamovich Parpiev & Abdukhakim Ziyaev. (2019)
Crystal structure of tetra-μ-acetato-bis[(5-amino-2-methylsulfanyl-1,3,4-thiadiazole-κ
N
1
)copper(II)]
. Acta Crystallographica Section E Crystallographic Communications 75:8, pages 1239-1242.
Crossref
Crossref
Kristiana T. Santoso, Chen‐Yi Cheung, Kiel Hards, Gregory M. Cook, Bridget L. Stocker & Mattie S. M. Timmer. (2019) Synthesis and Investigation of Phthalazinones as Antitubercular Agents. Chemistry – An Asian Journal 14:8, pages 1278-1285.
Crossref
Crossref
Maria Shafique, Shahid Hameed, Muhammad Moazzam Naseer & Najim Aboud Al-Masoudi. (2018) Synthesis of new chiral 1,3,4-thiadiazole-based di- and tri-arylsulfonamide residues and evaluation of in vitro anti-HIV activity and cytotoxicity. Molecular Diversity 22:4, pages 957-968.
Crossref
Crossref
Anna A. Hoser, Daniel M. Kamiński, Alicja Skrzypek, Arkadiusz Matwijczuk, Andrzej Niewiadomy, Mariusz Gagoś & Krzysztof Woźniak. (2018) Interplay of Inter- and Intramolecular Interactions in Crystal Structures of 1,3,4-Thiadiazole Resorcinol Derivatives. Crystal Growth & Design 18:7, pages 3851-3862.
Crossref
Crossref
Mahmut Gür, Nesrin Şener, Çiğdem A. Kaştaş, Osman Emre Özkan, Halit Muğlu & Magboule A. M. Elmaswari. (2017) Synthesis and Characterization of Some New Heteroaromatic Compounds Having Chirality Adjacent to a 1,3,4-Thiadiazole Moiety and Their Antimicrobial Activities. Journal of Heterocyclic Chemistry 54:6, pages 3578-3590.
Crossref
Crossref
Olfat Abiad Nief. (2015) Photostabilization of polyvinyl chloride by some new thiadiazole derivatives. European Journal of Chemistry 6:3, pages 242-247.
Crossref
Crossref
Noemí Vila, Pedro Besada, Tamara Costas, Mª Carmen Costas-Lago & Carmen Terán. (2015) Phthalazin-1(2H)-one as a remarkable scaffold in drug discovery. European Journal of Medicinal Chemistry 97, pages 462-482.
Crossref
Crossref
Ş.Güniz Küçükgüzel & Pelin Çıkla-Süzgün. (2015) Recent advances bioactive 1,2,4-triazole-3-thiones. European Journal of Medicinal Chemistry 97, pages 830-870.
Crossref
Crossref
Hany S. Ibrahim, Wagdy M. Eldehna, Hatem A. Abdel-Aziz, Mahmoud M. Elaasser & Marwa M. Abdel-Aziz. (2014) Improvement of antibacterial activity of some sulfa drugs through linkage to certain phthalazin-1(2H)-one scaffolds. European Journal of Medicinal Chemistry 85, pages 480-486.
Crossref
Crossref
Mashooq Ahmad Bhat, Abdul Arif Khan, Shahanavaj Khan, Mohamed A. Al-Omar, Mohammad Khalid Parvez, Mohammed Salem Al-Dosari & Abdullah Al-Dhfyan. (2014) Synthesis and anti-Candidal activity of N-(4-aryl/cyclohexyl)-2-(pyridine-4-yl carbonyl) hydrazinecarbothioamide. Bioorganic & Medicinal Chemistry Letters 24:5, pages 1299-1302.
Crossref
Crossref
Ahmed Kamal, Vangala Santhosh Reddy, Karnewar Santosh, G. Bharath Kumar, Anver Basha Shaik, Rasala Mahesh, Sumit. S. Chourasiya, Ibrahim Bin Sayeed & Srigiridhar Kotamraju. (2014) Synthesis of imidazo[2,1-b][1,3,4]thiadiazole–chalcones as apoptosis inducing anticancer agents. Med. Chem. Commun. 5:11, pages 1718-1723.
Crossref
Crossref
R.K. Dani, M.K. Bharty, S.K. Kushawaha, S. Paswan, Om Prakash, Ranjan K. Singh & N.K. Singh. (2013) Syntheses, spectral, X-ray and DFT studies of 5-benzyl-N-phenyl-1,3,4-thiadiazol-2-amine, 2-(5-phenyl-1,3,4-thiadiazol-2-yl) pyridine and 2-(5-methyl-1,3,4-thiadiazole-2-ylthio)-5-methyl-1,3,4-thiadiazole obtained by Mn(II) catalyzed reactions. Journal of Molecular Structure 1054-1055, pages 251-261.
Crossref
Crossref
Abhishek Kumar Jain, Simant Sharma, Ankur Vaidya, Veerasamy Ravichandran & Ram Kishore Agrawal. (2013) 1,3,4-Thiadiazole and its Derivatives: A Review on Recent Progress in Biological Activities. Chemical Biology & Drug Design 81:5, pages 557-576.
Crossref
Crossref
Bhawna Sharma, Amita Verma, Sunil Prajapati & Upendra Kumar Sharma. (2013) Synthetic Methods, Chemistry, and the Anticonvulsant Activity of Thiadiazoles. International Journal of Medicinal Chemistry 2013, pages 1-16.
Crossref
Crossref
Agata Siwek, Joanna Stefańska, Katarzyna Dzitko & Artur Ruszczak. (2012) Antifungal effect of 4-arylthiosemicarbazides against Candida species. Search for molecular basis of antifungal activity of thiosemicarbazide derivatives. Journal of Molecular Modeling 18:9, pages 4159-4170.
Crossref
Crossref
Keriman Özadalı, Fügen Özkanlı, Sarthak Jain, Praveen P.N. Rao & Carlos A. Velázquez-Martínez. (2012) Synthesis and biological evaluation of isoxazolo[4,5-d]pyridazin-4-(5H)-one analogues as potent anti-inflammatory agents. Bioorganic & Medicinal Chemistry 20:9, pages 2912-2922.
Crossref
Crossref
Agata Siwek, Katarzyna Świderek & Stefan Jankowski. (2011) Problems with molecular mechanics implementations on the example of 4-benzoyl-1-(4-methyl-imidazol-5-yl)-carbonylthiosemicarbazide. Journal of Molecular Modeling 18:3, pages 843-849.
Crossref
Crossref
Irena Wawrzycka-Gorczyca & Agata Siwek. (2011)
Synthesis, X-ray crystal structure and theoretical study of 4-ethyl-5-(2-thienyl)-2,4-dihydro-3
H
-1,2,4-triazole-3-thione; structural comparison with its aromatic analogs
. Zeitschrift für Kristallographie 226:11, pages 861-868.
Crossref
Crossref
Agata Siwek, Paweł Stączek & Joanna Stefańska. (2011) Synthesis and structure–activity relationship studies of 4-arylthiosemicarbazides as topoisomerase IV inhibitors with Gram-positive antibacterial activity. Search for molecular basis of antibacterial activity of thiosemicarbazides. European Journal of Medicinal Chemistry 46:11, pages 5717-5726.
Crossref
Crossref
Agata Siwek, Paweł Stączek, Monika Wujec, Joanna Stefańska, Urszula Kosikowska, Anna Malm, Stefan Jankowski & Piotr Paneth. (2010) Biological and docking studies of topoisomerase IV inhibition by thiosemicarbazides. Journal of Molecular Modeling 17:9, pages 2297-2303.
Crossref
Crossref
Irena Wawrzycka-Gorczyca, Agata Siwek, Urszula Kosikowska & Anna Malm. (2011)
Synthesis and crystal structure of
N
-butyl-5-(4-methyl-1,2,3-thiadiazol-5-yl)-1,3,4-thiadiazol-2-amine and 5-isoquinolin-3-yl-
N
-(2-methylphenyl)-1,3,4-thiadiazol-2-amine
. Zeitschrift für Kristallographie 226:3, pages 297-302.
Crossref
Crossref
Agata Siwek, Monika Wujec, Tomasz Plech, Edyta Kuśmierz, Ewa Jagiełło‐Wójtowicz & Anna Chodkowska. (2010)
Structure–activity relationship of
s
‐triazoles and thiadiazoles as analgesics
. Heteroatom Chemistry 21:4, pages 256-264.
Crossref
Crossref
Agata Siwek, Joanna Stefańska, Irena Wawrzycka‐Gorczyca & Monika Wujec. (2010) Synthesis and in vitro antibacterial evaluation of 1‐substituted‐4‐ethoxycarbonylmethylthiosemicarbazides and products of their dehydrocyclization. Heteroatom Chemistry 21:3, pages 131-138.
Crossref
Crossref