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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 24, 2009 - Issue 5
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Research Article

Microwave assisted, one-pot synthesis of 5-nitro- 2-aryl substituted-1H-benzimidazole libraries: Screening in vitro for antimicrobial activity

Kallappa Mahadevappa HosamaniP.G. Department of Studies in Chemistry, Karnatak University, Pavate Nagar, Dharwad-580 003, IndiaCorrespondence[email protected]
,
Harisha Reddy SeetharamareddyP.G. Department of Studies in Chemistry, Karnatak University, Pavate Nagar, Dharwad-580 003, India
,
Rangappa Sangappa KeriP.G. Department of Studies in Chemistry, Karnatak University, Pavate Nagar, Dharwad-580 003, India
,
Manohar Shirugumbi HanamanthagoudaP.G. Department of Studies in Chemistry, Karnatak University, Pavate Nagar, Dharwad-580 003, India
&
Mark G. MoloneyDepartment of Chemistry, Chemistry Research Laboratory, University of Oxford, Oxford, UK
Pages 1095-1100 | Received 26 May 2008, Accepted 28 Oct 2008, Published online: 23 Sep 2009

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Emre Menteşe, Hakan Bektaş, Serdar Ülker, Olcay Bekircan & Bahittin Kahveci. (2014) Microwave-assisted synthesis of new benzimidazole derivatives with lipase inhibition activity. Journal of Enzyme Inhibition and Medicinal Chemistry 29:1, pages 64-68.
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Mohammad Shakirullah, Hanif Ahmad, Muhammad Raza Shah, Imtiaz Ahmad, Muhammad Ishaq, Nematullah Khan, Amir Badshah & Inamullah Khan. (2011) Antimicrobial activities of Conyzolide and Conyzoflavone from Conyza canadensis. Journal of Enzyme Inhibition and Medicinal Chemistry 26:4, pages 468-471.
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Kaan Küçükoğlu, Ulviye Acar Çevik, Hayrunnisa Nadaroglu, Ismail Celik, Ayşen Işık, Hayrani Eren Bostancı, Yusuf Özkay & Zafer Asım Kaplancıklı. (2023) Synthesis and Molecular Docking of New N-Acyl Hydrazones- Benzimidazole as hCA I and II Inhibitors. Medicinal Chemistry 19:5, pages 485-494.
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Christina Zalaru, Florea Dumitrascu, Constantin Draghici, Isabela Tarcomnicu, Maria Marinescu, George Mihai Nitulescu, Rodica Tatia, Lucia Moldovan, Marcela Popa & Mariana Carmen Chifiriuc. (2022) New Pyrazolo-Benzimidazole Mannich Bases with Antimicrobial and Antibiofilm Activities. Antibiotics 11:8, pages 1094.
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Gurumeet C Wadhawa, Sarang Bhagvat, Ramesh Mohite & Yashwant Gaikwad. (2022) An Efficient Synthesis of 2,4,5-Triaryl-1H-Imidazole Derivatives Catalyzed by Boric Acid IN Green Condition. International Journal of Advanced Research in Science, Communication and Technology, pages 255-260.
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Arup K. Kabi, Sattu Sravani, Raghuram Gujjarappa, Aakriti Garg, Nagaraju Vodnala, Ujjawal Tyagi, Dhananjaya Kaldhi, Virender Singh, Sreya Gupta & Chandi C. Malakar. 2022. Nanostructured Biomaterials. Nanostructured Biomaterials 351 378 .
Mohamed Hagar, Kamel Chaieb, Shazia Parveen, H.A. Ahmed & R.B. Alnoman. (2020) N-alkyl 2-pyridone versus O-alkyl 2-pyridol: Ultrasonic synthesis, DFT, docking studies and their antimicrobial evaluation. Journal of Molecular Structure 1199, pages 126926.
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Adele Cheddie, Suhas A. Shintre, Aishwarya Bantho, Chunderika Mocktar & Neil A. Koorbanally. (2019) Synthesis and antibacterial activity of a series of 2‐trifluoromethylbenzimidazole‐thiazolidinone derivatives. Journal of Heterocyclic Chemistry 57:1, pages 299-307.
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Manaswini Raj & Sumanta Kumar Padhi. (2019) Synthesis, Characterization, and Structure of Quinoline‐based Benzimidazole Derivatives. Journal of Heterocyclic Chemistry 56:3, pages 988-997.
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Ding Ma, Xiaoming Ji, Zhuo Wu, Cang Cheng, Bo Zhou & Yanghui Zhang. (2019) Synthesis of Benzimidazoles through Palladium-Catalyzed Amination of 2-Iodobenzimines with Diaziridinone. Advanced Synthesis & Catalysis 361:4, pages 739-746.
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Hojat-Allah Arab, Mohammad Ali Faramarzi, Nasrin Samadi, Hamid Irannejad, Alireza Foroumadi & Saeed Emami. (2018) New 7-piperazinylquinolones containing (benzo[d]imidazol-2-yl)methyl moiety as potent antibacterial agents. Molecular Diversity 22:4, pages 815-825.
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Hakan Bektas, Canan Albay, Bahar Bilgin Sökmen, Sinem Aydın, Emre Menteşe, Gülbahar Aydın & Dilem Şen. (2018) Synthesis, Antioxidant, and Antibacterial Activities of Some New 2-(3-fluorobenzyl)-1 H -benzimidazole Derivatives . Journal of Heterocyclic Chemistry 55:10, pages 2400-2407.
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Alejandra Vázquez-Raygoza, Lucia Cano-González, Israel Velázquez-Martínez, Pedro Trejo-Soto, Rafael Castillo, Alicia Hernández-Campos, Francisco Hernández-Luis, Jesús Oria-Hernández, Adriana Castillo-Villanueva, Claudia Avitia-Domínguez, Erick Sierra-Campos, Mónica Valdez-Solana & Alfredo Téllez-Valencia. (2017) Species-Specific Inactivation of Triosephosphate Isomerase from Trypanosoma brucei: Kinetic and Molecular Dynamics Studies. Molecules 22:12, pages 2055.
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Rangappa S. Keri, Asha Hiremathad, Srinivasa Budagumpi & Bhari Mallanna Nagaraja. (2015) Comprehensive Review in Current Developments of Benzimidazole-Based Medicinal Chemistry. Chemical Biology & Drug Design 86:1, pages 19-65.
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Geeta Yadav & Swastika Ganguly. (2015) Structure activity relationship (SAR) study of benzimidazole scaffold for different biological activities: A mini-review. European Journal of Medicinal Chemistry 97, pages 419-443.
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Alexey N. Rodionov, Kira Ya. Zherebker, Lubov′ V. Snegur, Alexander A. Korlyukov, Dmitry E. Arhipov, Alexander S. Peregudov, Mikhail M. Ilyin, Mikhail M. IlyinJr.Jr., Oleg M. Nikitin, Nataliya B. Morozova & Alexander A. Simenel. (2015) Synthesis, structure and enantiomeric resolution of ferrocenylalkyl mercaptoazoles. Antitumor activity in vivo. Journal of Organometallic Chemistry 783, pages 83-91.
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Kallappa. M. Hosamani, Dinesh S. Reddy & Hirihalli. C. Devarajegowda. (2015) Microwave-assisted synthesis of new fluorinated coumarin–pyrimidine hybrids as potent anticancer agents, their DNA cleavage and X-ray crystal studies. RSC Advances 5:15, pages 11261-11271.
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Rangappa S. Keri, Kallappa M. Hosamani & Ramya V. Shingalapur. (2010) RETRACTED ARTICLE: Synthesis, anti-bacterial, anti-fungal and cytotoxic properties of novel pyrimidine derivatives from chromen-2-one moiety. Medicinal Chemistry Research 23:8, pages 3927-3927.
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Bahittin Kahveci, Fatih Yılmaz, Emre Menteşe, Musa Özil & Şengül Alpay Karaoğlu. (2014) Microwave-Assisted Synthesis of Some Novel Benzimidazole Derivatives Containing Imine Function and Evaluation of Their Antimicrobial Activity. Journal of Heterocyclic Chemistry 51:4, pages 982-990.
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E. Menteşe, I. S. Doğan & B. Kahveci. (2013) Green Protocol: Solvent- and Catalyst-Free Synthesis of Benzimidazole Derivatives via Microwave Technique. Chemistry of Heterocyclic Compounds 49:8, pages 1136-1140.
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Asif Husain, Mohd Rashid, Ravinesh Mishra, Shama Parveen, Dong-Soo Shin & Deepak Kumar. (2012) Benzimidazole bearing oxadiazole and triazolo-thiadiazoles nucleus: Design and synthesis as anticancer agents. Bioorganic & Medicinal Chemistry Letters 22:17, pages 5438-5444.
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Mohd Rashid, Asif Husain & Ravinesh Mishra. (2012) Synthesis of benzimidazoles bearing oxadiazole nucleus as anticancer agents. European Journal of Medicinal Chemistry 54, pages 855-866.
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Rangappa S. Keri, Kallappa M. Hosamani, Ramya V. Shingalapur & Mallinath H. Hugar. (2010) Analgesic, anti-pyretic and DNA cleavage studies of novel pyrimidine derivatives of coumarin moiety. European Journal of Medicinal Chemistry 45:6, pages 2597-2605.
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Kavitha C.S. Achar, Kallappa M. Hosamani & Harisha R. Seetharamareddy. (2010) In-vivo analgesic and anti-inflammatory activities of newly synthesized benzimidazole derivatives. European Journal of Medicinal Chemistry 45:5, pages 2048-2054.
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Ramya V. Shingalapur, Kallappa M. Hosamani, Rangappa S. Keri & Mallinath H. Hugar. (2010) Derivatives of benzimidazole pharmacophore: Synthesis, anticonvulsant, antidiabetic and DNA cleavage studies. European Journal of Medicinal Chemistry 45:5, pages 1753-1759.
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Rangappa S. Keri, Kallappa M. Hosamani, Harisha S. Reddy & Ramya V. Shingalapur. (2010) Synthesis, in‐vitro Antimicrobial and Cytotoxic Studies of Novel Azetidinone Derivatives . Archiv der Pharmazie 343:4, pages 237-247.
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