Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 24, Issue 5 (2009)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 24, Issue 5 (2009)

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Research Article

Article
Inhibition of dipeptidyl peptidase IV (DPP IV) is one of the mechanisms explaining the hypoglycemic effect of berberine
Ihab M. Al-masri, Mohammad K. Mohammad & Mutasem O. Tahaa
Pages: 1061-1066
Published online: 29 Jul 2009
AbstractforInhibition of dipeptidyl peptidase IV (DPP IV) is one of the mechanisms explaining the hypoglycemic effect of berberine | Full Text | References | PDF (1.2 MB)
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Article
Design, synthesis and evaluation of 3-(imidazol- 1-ylmethyl)indoles as antileishmanial agents. Part II
Francis Giraud, Cedric Loge, Fabrice Pagniez, Damien Crepin, Sophie Barres, Carine Picot, Patrice Le Pape & Marc Le Borgne
Pages: 1067-1075
Published online: 20 Mar 2009
AbstractforDesign, synthesis and evaluation of 3-(imidazol- 1-ylmethyl)indoles as antileishmanial agents. Part II | Full Text | References | PDF (1 MB)
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Article
Dual effects of aliphatic carboxylic acids on cresolase and catecholase reactions of mushroom tyrosinase
N. Gheibi, A.A. Saboury, K. Haghbeen, F. Rajaei & A.A. Pahlevan
Pages: 1076-1081
Published online: 19 Mar 2009
AbstractforDual effects of aliphatic carboxylic acids on cresolase and catecholase reactions of mushroom tyrosinase | Full Text | References | PDF (857.5 KB)
  • 620 Views
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Article
Kinetics of jack bean urease inhibition by 2,3-dichloro-1,4-naphthoquinone. Elucidation of the mechanism: redox cycling and sulfhydryl arylation
Wiesława Zaborska, Mirosława Kot & Agnieszka Bala
Pages: 1082-1087
Published online: 21 Jul 2009
AbstractforKinetics of jack bean urease inhibition by 2,3-dichloro-1,4-naphthoquinone. Elucidation of the mechanism: redox cycling and sulfhydryl arylation | Full Text | References | PDF (971.2 KB)
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Article
Design, synthesis, spectral analysis and in vitro microbiological evaluation of 2-phenyl-3-(4,6-diarylpyrimidin-2-yl)thiazolidin-4-ones
M. Gopalakrishnan, J. Thanusu & V. Kanagarajan
Pages: 1088-1094
Published online: 19 Mar 2009
AbstractforDesign, synthesis, spectral analysis and in vitro microbiological evaluation of 2-phenyl-3-(4,6-diarylpyrimidin-2-yl)thiazolidin-4-ones | Full Text | References | PDF (738.3 KB)
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Article
Microwave assisted, one-pot synthesis of 5-nitro- 2-aryl substituted-1H-benzimidazole libraries: Screening in vitro for antimicrobial activity
Kallappa Mahadevappa Hosamani, Harisha Reddy Seetharamareddy, Rangappa Sangappa Keri, Manohar Shirugumbi Hanamanthagouda & Mark G. Moloney
Pages: 1095-1100
Published online: 23 Sep 2009
AbstractforMicrowave assisted, one-pot synthesis of 5-nitro- 2-aryl substituted-1H-benzimidazole libraries: Screening in vitro for antimicrobial activity | Full Text | References | PDF (877.3 KB)
  • 836 Views
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Article
Molecular dynamics simulation of Axillaridine–A: A potent natural cholinesterase inhibitor
Zaheer ul-Haq, Hassan Hadi, Syed Tarique Moin & M. Iqbal Choudhary
Pages: 1101-1105
Published online: 07 Apr 2009
AbstractforMolecular dynamics simulation of Axillaridine–A: A potent natural cholinesterase inhibitor | Full Text | References | PDF (1.1 MB)
  • 623 Views
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Article
The pyrostatins A and B do not inhibit N-acetyl-ß-D-glucosaminidase
Daniel Appel & Georg Lentzen
Pages: 1106-1108
Published online: 19 Mar 2009
AbstractforThe pyrostatins A and B do not inhibit N-acetyl-ß-D-glucosaminidase | Full Text | References | PDF (717 KB)
  • 548 Views
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Article
QSAR studies on 4-anilino-3-quinolinecarbonitriles as Src kinase inhibitors using robust PCA and both linear and nonlinear models
Min Sun, Youguang Zheng, Hongtao Wei, Junqing Chen & Min Ji
Pages: 1109-1116
Published online: 07 Apr 2009
AbstractforQSAR studies on 4-anilino-3-quinolinecarbonitriles as Src kinase inhibitors using robust PCA and both linear and nonlinear models | Full Text | References | PDF (870.2 KB)
  • 519 Views
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Article
Compounds with neuroprotective activity from the medicinal plant Machilus thunbergii
Choong Je Ma, Young Choong Kim & Sang Hyun Sung
Pages: 1117-1121
Published online: 19 Mar 2009
AbstractforCompounds with neuroprotective activity from the medicinal plant Machilus thunbergii | Full Text | References | PDF (641.2 KB)
  • 999 Views
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Article
A comparative study on the effect of homobrassinolide and gibberellic acid on lipid peroxidation and antioxidant status in normal and diabetic rats
P. Muthuraman & K. Srikumar
Pages: 1122-1127
Published online: 21 Jul 2009
AbstractforA comparative study on the effect of homobrassinolide and gibberellic acid on lipid peroxidation and antioxidant status in normal and diabetic rats | Full Text | References | PDF (596.8 KB)
  • 891 Views
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Article
Galinsosides A and B, bioactive flavanone glucosides from Galinsoga parviflora
Sadia Ferheen, Aziz-Ur-Rehman , Nighat Afza, Abdul Malik, Lubna Iqbal, Muhammad Azam Rasool, Muhammad Irfan Ali & Rasool Bakhsh Tareen
Pages: 1128-1132
Published online: 23 Sep 2009
AbstractforGalinsosides A and B, bioactive flavanone glucosides from Galinsoga parviflora | Full Text | References | PDF (627.7 KB)
  • 1599 Views
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Article
PTP1B inhibitory effects of tridepside and related metabolites isolated from the Antarctic lichen Umbilicaria antarctica
Changon Seo, Yun-Hyeok Choi, Jong Seog Ahn, Joung Han Yim, Hong Kum Lee & Hyuncheol Oh
Pages: 1133-1137
Published online: 21 Jul 2009
AbstractforPTP1B inhibitory effects of tridepside and related metabolites isolated from the Antarctic lichen Umbilicaria antarctica | Full Text | References | PDF (714.8 KB)
  • 1013 Views
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Article
Chemical constituents isolated from Paeonia lactiflora roots and their neuroprotective activity against oxidative stress in vitro
Seung Hyun Kim, Mi Kyeong Lee, Ki Yong Lee, Sang Hyun Sung, Jinwoong Kim & Young Choong Kim
Pages: 1138-1140
Published online: 23 Sep 2009
AbstractforChemical constituents isolated from Paeonia lactiflora roots and their neuroprotective activity against oxidative stress in vitro | Full Text | References | PDF (610.1 KB)
  • 2105 Views
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Article
Screening and evaluation of antioxidant activity of some amido-carbonyl oxime derivatives and their radical scavenging activities
Tevfik Özen & Murat Taş
Pages: 1141-1147
Published online: 23 Sep 2009
AbstractforScreening and evaluation of antioxidant activity of some amido-carbonyl oxime derivatives and their radical scavenging activities | Full Text | References | PDF (717.1 KB)
  • 934 Views
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Article
Synthesis, inhibition of NO production and antiproliferative activities of some indole derivatives
Maria Stefania Sinicropi, Anna Caruso, Filomena Conforti, Mariangela Marrelli, Hussein El Kashef, Jean-charles Lancelot, Sylvain Rault, Giancarlo A. Statti & Francesco Menichini
Pages: 1148-1153
Published online: 19 Mar 2009
AbstractforSynthesis, inhibition of NO production and antiproliferative activities of some indole derivatives | Full Text | References | PDF (762 KB)
  • 808 Views
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Article
Tyrosinase inhibitory effect and inhibitory mechanism of tiliroside from raspberry
Yan-hua Lu, Juan Chen, Dong-zhi Wei, Zheng-tao Wang & Xin-yi Tao
Pages: 1154-1160
Published online: 23 Sep 2009
AbstractforTyrosinase inhibitory effect and inhibitory mechanism of tiliroside from raspberry | Full Text | References | PDF (737.6 KB)
  • 2129 Views
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Article
Synthesis, antimicrobial and antiviral activity of substituted benzimidazoles
Deepika Sharma, Balasubramanian Narasimhan, Pradeep Kumar, Vikramjeet Judge, Rakesh Narang, Erik De Clercq & Jan Balzarini
Pages: 1161-1168
Published online: 23 Sep 2009
AbstractforSynthesis, antimicrobial and antiviral activity of substituted benzimidazoles | Full Text | References | PDF (692.7 KB)
  • 1608 Views
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Article
Anticancer and immunomodulatory activities of novel 1,8-naphthyridine derivatives
Vivek Kumar, Alka Madaan, Vinod K. Sanna, Manupriya Vishnoi, Narendra Joshi, Anu T. Singh, Manu Jaggi, Pramod K. Sharma, Raghuveer Irchhaiya & Anand C. Burman
Pages: 1169-1178
Published online: 21 Apr 2009
AbstractforAnticancer and immunomodulatory activities of novel 1,8-naphthyridine derivatives | Full Text | References | PDF (2.8 MB)
  • 871 Views
  • 9 CrossRef citations
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Article
Synthesis and biological evaluation of O-methyl and O-ethyl NSAID hydroxamic acids
Zrinka Rajić, Ivana Perković, Ivan Butula, Branka Zorc, Dimitra Hadjipavlou-Litina, Eleni Pontiki, Stjepan Pepeljnjak & Ivan Kosalec
Pages: 1179-1187
Published online: 23 Sep 2009
AbstractforSynthesis and biological evaluation of O-methyl and O-ethyl NSAID hydroxamic acids | Full Text | References | PDF (1.1 MB)
  • 1034 Views
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Article
Kukoamine A analogs with lipoxygenase inhibitory activity
Dimitra Hadjipavlou-Litina, Thomas Garnelis, Constantinos M. Athanassopoulos & Dionissios Papaioannou
Pages: 1188-1193
Published online: 23 Sep 2009
AbstractforKukoamine A analogs with lipoxygenase inhibitory activity | Full Text | References | PDF (641.4 KB)
  • 1033 Views
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Article
A series of cinnamic acid derivatives and their inhibitory activity on intestinal α-glucosidase
Sirichai Adisakwattana, Praew Chantarasinlapin, Haruthai Thammarat & Sirintorn Yibchok-Anun
Pages: 1194-1200
Published online: 23 Sep 2009
AbstractforA series of cinnamic acid derivatives and their inhibitory activity on intestinal α-glucosidase | Full Text | References | PDF (890.9 KB)
  • 5041 Views
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Article
Synthesis, spectroscopic, and antibacterial activity of tetraazamacrocyclic complexes of trivalent chromium, manganese, and iron
D.P. Singh, Vandna Malik, Ramesh Kumar & Jitender Singh
Pages: 1201-1206
Published online: 23 Sep 2009
AbstractforSynthesis, spectroscopic, and antibacterial activity of tetraazamacrocyclic complexes of trivalent chromium, manganese, and iron | Full Text | References | PDF (703.5 KB)
  • 558 Views
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