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Original Article

In vitro antileishmanial activity of fisetin flavonoid via inhibition of glutathione biosynthesis and arginase activity in Leishmania infantum

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Read on this site (3)

Ingrid T. L. Ramos, Tania M. S. Silva & Celso A. Camara. (2019) Synthesis of new 6- and 8-Alkenyl-3,7,3’,4’-Tetramethoxyquercetin derivatives by microwave-assisted Heck coupling. Synthetic Communications 49:19, pages 2583-2589.
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Bárbara Velame Ferreira Teixeira, André Lacerda Braga Teles, Suellen Gonçalves da Silva, Camila Carane Bitencourt Brito, Humberto Fonseca de Freitas, Acássia Benjamim Leal Pires, Thamires Quadros Froes & Marcelo Santos Castilho. (2019) Dual and selective inhibitors of pteridine reductase 1 (PTR1) and dihydrofolate reductase-thymidylate synthase (DHFR-TS) from Leishmania chagasi. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1439-1450.
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Andreza R. Garcia, Danielle M. P. Oliveira, Ana Claudia F. Amaral, Jéssica B. Jesus, Ana Carolina Rennó Sodero, Alessandra M. T. Souza, Claudiu T. Supuran, Alane B. Vermelho, Igor A. Rodrigues & Anderson S. Pinheiro. (2019) Leishmania infantum arginase: biochemical characterization and inhibition by naturally occurring phenolic substances. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1100-1109.
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Articles from other publishers (14)

Janay Stefany Carneiro Araújo, Larissa de Mattos Oliveira, Kaio Vinícius Freitas de Andrade, Raquel Guimarães Benevides, Franco Henrique Andrade Leite & Manoelito Coelho dos Santos Junior. (2023) Superoxide Dismutase Inhibitors against Malaria, Leishmaniasis, and Chagas Disease: Systematic Review. Current Drug Targets 24:2, pages 201-210.
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Jacqueline Soto-Sánchez. (2022) Bioactivity of Natural Polyphenols as Antiparasitic Agents and their Biochemical Targets. Mini-Reviews in Medicinal Chemistry 22:20, pages 2661-2677.
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Huseyin Istanbullu & Gulsah Bayraktar. 2022. Leishmaniasis - General Aspects of a Stigmatized Disease. Leishmaniasis - General Aspects of a Stigmatized Disease.
Ana Elena Ahuir-Baraja, María Pilar Ruiz, María Magdalena Garijo & Lola Llobat. (2021) Feline Leishmaniosis: An Emerging Public Health Problem. Veterinary Sciences 8:9, pages 173.
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Beradiye ÇELİKÇİ, Rüstem Anıl UĞAN & Erdem TOKTAY. (2021) Sıçanlarda letrozolün indüklediği polikistik over sendromunda fisetinin etkileriEffects of fisetin to letrozole-induced polycystic ovary syndrome in rats. Cukurova Medical Journal 46:2, pages 508-515.
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María Fernanda García-Bustos, Agustín Moya Álvarez, Cecilia Pérez Brandan, Cecilia Parodi, Andrea Mabel Sosa, Valeria Carolina Buttazzoni Zuñiga, Oscar Marcelo Pastrana, Paula Manghera, Pablo Alejandro Peñalva, Jorge Diego Marco & Paola Andrea Barroso. (2021) Development of a Fluorescent Assay to Search New Drugs Using Stable tdTomato-Leishmania, and the Selection of Galangin as a Candidate With Anti-Leishmanial Activity. Frontiers in Cellular and Infection Microbiology 11.
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Nicola S. Carter, Brendan D. Stamper, Fawzy Elbarbry, Vince Nguyen, Samuel Lopez, Yumena Kawasaki, Reyhaneh Poormohamadian & Sigrid C. Roberts. (2021) Natural Products That Target the Arginase in Leishmania Parasites Hold Therapeutic Promise. Microorganisms 9:2, pages 267.
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Igor A. Rodrigues, Andreza R. Garcia, Mariana M. Paz, Rogério G. D. Grilo Junior, Ana Claudia F. Amaral & Anderson S. Pinheiro. 2022. Antiprotozoal Drug Development and Delivery. Antiprotozoal Drug Development and Delivery 143 180 .
Shweta Raj, Santanu Sasidharan, S. N. Balaji, Vikash Kumar Dubey & Prakash Saudagar. (2020) Review on natural products as an alternative to contemporary anti-leishmanial therapeutics. Journal of Proteins and Proteomics 11:2, pages 135-158.
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Andrea M. Sosa, Agustín Moya Álvarez, Estefanía Bracamonte, Masataka Korenaga, Jorge D. Marco & Paola A. Barroso. (2020) Efficacy of Topical Treatment with (−)-Epigallocatechin Gallate, A Green Tea Catechin, in Mice with Cutaneous Leishmaniasis. Molecules 25:7, pages 1741.
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Marcus Tullius Scotti, Alex France Messias Monteiro, Jéssika de Oliveira Viana, Francisco Jaime Bezerra Mendonça Junior, Hamilton M. Ishiki, Ernestine Nkwengoua Tchouboun, Rodrigo Santos A. De Araújo & Luciana Scotti. (2020) Recent Theoretical Studies Concerning Important Tropical Infections. Current Medicinal Chemistry 27:5, pages 795-834.
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Keivan Adinehbeigi, Minoo Shaddel, Saeed Khalili & Alireza Zakeri. (2020) Suramin could block the activity of Arabinono-1, 4-lactone oxidase enzyme from Leishmania donovani: structure-based screening and molecular dynamics analyses. Transactions of The Royal Society of Tropical Medicine and Hygiene 114:3, pages 162-172.
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Pone Kamdem Boniface & Elizabeth Igne Ferreira. (2019) Flavonoids as efficient scaffolds: Recent trends for malaria, leishmaniasis, Chagas disease, and dengue. Phytotherapy Research 33:10, pages 2473-2517.
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Bilal Ahmad, Arshad Islam, Arif Khan, Mubarak Ali Khan, Ihsan ul Haq, Laila Jafri, Mansoor Ahmad, Shaila Mehwish, Ajmal Khan & Nazif Ullah. (2019) Comprehensive investigations on anti-leishmanial potentials of Euphorbia wallichii root extract and its effects on membrane permeability and apoptosis. Comparative Immunology, Microbiology and Infectious Diseases 64, pages 138-145.
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