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Research Article

Itraconazole Formulation Studies of the Melt-Extrusion Process with Mixture Design

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Pages 641-652 | Published online: 06 Dec 2003

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M. Maniruzzaman, M. M. Rana, J. S. Boateng, J. C. Mitchell & D. Douroumis. (2013) Dissolution enhancement of poorly water-soluble APIs processed by hot-melt extrusion using hydrophilic polymers. Drug Development and Industrial Pharmacy 39:2, pages 218-227.
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Parinda Srinarong, Hans de Waard, Henderik W Frijlink & Wouter LJ Hinrichs. (2011) Improved dissolution behavior of lipophilic drugs by solid dispersions: the production process as starting point for formulation considerations. Expert Opinion on Drug Delivery 8:9, pages 1121-1140.
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L.S. Ranzani, J. Font, F. Galimany, A. Santanach, A.M. Gomez-Gomar, G. Casadevall & A. Gryczke. (2011) Enhanced in vivo absorption of CB-1 antagonist in rats via solid solutions prepared by hot-melt extrusion. Drug Development and Industrial Pharmacy 37:6, pages 694-701.
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Dave A. Miller, James C. DiNunzio, Wei Yang, James W. McGinity & Robert O. Williams$suffix/text()$suffix/text(). (2008) Enhanced In Vivo Absorption of Itraconazole via Stabilization of Supersaturation Following Acidic-to-Neutral pH Transition. Drug Development and Industrial Pharmacy 34:8, pages 890-902.
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Alfred Fahr & Xiangli Liu. (2007) Drug delivery strategies for poorly water-soluble drugs. Expert Opinion on Drug Delivery 4:4, pages 403-416.
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Stacy M. Trey, Douglas A. Wicks, Praveen K. Mididoddi & Michael A. Repka. (2007) Delivery of Itraconazole from Extruded HPC Films. Drug Development and Industrial Pharmacy 33:7, pages 727-735.
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Xin Zheng, Rui Yang, Xing Tang & Liangyuan Zheng. (2007) Part I: Characterization of Solid Dispersions of Nimodipine Prepared by Hot-melt Extrusion. Drug Development and Industrial Pharmacy 33:7, pages 791-802.
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Edmund J. Elder, Jonathan C. Evans, Brian D. Scherzer, James E. Hitt, Gary B. Kupperblatt, Shakil A. Saghir & Dan A. Markham. (2007) Preparation, Characterization, and Scale-up of Ketoconazole with Enhanced Dissolution and Bioavailability. Drug Development and Industrial Pharmacy 33:7, pages 755-765.
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Jiahui Hu, Keith P. Johnston & Robert O. Williams$suffix/text()$suffix/text(). (2004) Nanoparticle Engineering Processes for Enhancing the Dissolution Rates of Poorly Water Soluble Drugs. Drug Development and Industrial Pharmacy 30:3, pages 233-245.
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David Engers, Jing Teng, Jonathan Jimenez-Novoa, Philip Gent, Stuart Hossack, Cheryl Campbell, John Thomson, Igor Ivanisevic, Alison Templeton, Stephen Byrn & Ann Newman. (2010) A Solid-State Approach to Enable Early Development Compounds: Selection and Animsal Bioavailability Studies of an Itraconazole Amorphous Solid Dispersion. Journal of Pharmaceutical Sciences 99:9, pages 3901-3922.
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Roger Vandecruys, Jef Peeters, Geert Verreck & Marcus E. Brewster. (2007) Use of a screening method to determine excipients which optimize the extent and stability of supersaturated drug solutions and application of this system to solid formulation design. International Journal of Pharmaceutics 342:1-2, pages 168-175.
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Mi‐Jin Park, Shan Ren & Beom‐Jin Lee. (2007) In vitro and in vivo comparative study of itraconazole bioavailability when formulated in highly soluble self‐emulsifying system and in solid dispersion . Biopharmaceutics & Drug Disposition 28:4, pages 199-207.
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Shankar Swaminathan, P. R. Vavia, Francesco Trotta & Satyen Torne. (2007) Formulation of betacyclodextrin based nanosponges of itraconazole. Journal of Inclusion Phenomena and Macrocyclic Chemistry 57:1-4, pages 89-94.
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Sang-Young Shim, Chang-Won Ji, Hongkee Sah, Eun-Seok Park & Beom-Jin Lee. (2006) Characterization of itraconazole semisolid dosage forms prepared by hot melt technique. Archives of Pharmacal Research 29:11, pages 1055-1060.
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Liang Wang, Fu De Cui, Tomokazu Hayase & Hisakazu Sunada. (2005) Preparation and Evaluation of Solid Dispersion for Nitrendipine–Carbopol and Nitrendipine–HPMCP Systems Using a Twin Screw Extruder. CHEMICAL & PHARMACEUTICAL BULLETIN 53:10, pages 1240-1245.
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