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Research Article

LIPID-BASED FORMULATIONS FOR ORAL ADMINISTRATION: OPPORTUNITIES FOR BIOAVAILABILITY ENHANCEMENT AND LIPOPROTEIN TARGETING OF LIPOPHILIC DRUGS

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Pages 215-257 | Published online: 31 Aug 2001

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Chunxi Liu, Donghua Liu, Fan Bai, Jian Zhang & Na Zhang. (2010) In vitro and in vivo studies of lipid-based nanocarriers for oral N3-o-toluyl-fluorouracil delivery. Drug Delivery 17:5, pages 352-363.
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Jigar P Patel & Dion R Brocks. (2009) The effect of oral lipids and circulating lipoproteins on the metabolism of drugs. Expert Opinion on Drug Metabolism & Toxicology 5:11, pages 1385-1398.
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Marc Muchow, Philippe Maincent & Rainer H. Müller. (2008) Lipid Nanoparticles with a Solid Matrix (SLN®, NLC®, LDC®) for Oral Drug Delivery. Drug Development and Industrial Pharmacy 34:12, pages 1394-1405.
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S. Khaleel Basha, R. Dhandayuthabani, M. Syed Muzammil & V. Sugantha Kumari. (2021) Solid lipid nanoparticles for oral drug delivery. Materials Today: Proceedings 36, pages 313-324.
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Abdulwahab Barakat, Ranjita Shegokar, Michael Dittgen & Rainer H. Müller. (2013) Coenzyme Q10 oral bioavailability: effect of formulation type. Journal of Pharmaceutical Investigation 43:6, pages 431-451.
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Kathy Wai Yu Lee, Christopher J. H. Porter & Ben J. Boyd. (2013) A Simple Quantitative Approach for the Determination of Long and Medium Chain Lipids in Bio-relevant Matrices by High Performance Liquid Chromatography with Refractive Index Detection. AAPS PharmSciTech 14:3, pages 927-934.
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Hywel D. Williams, Natalie L. Trevaskis, Susan A. Charman, Ravi M. Shanker, William N. Charman, Colin W. Pouton & Christopher J. H. Porter. (2013) Strategies to Address Low Drug Solubility in Discovery and Development. Pharmacological Reviews 65:1, pages 315-499.
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Jaime A. Yáñez, Stephen W.J. Wang, Ian W. Knemeyer, Mark A. Wirth & Kevin B. Alton. (2011) Intestinal lymphatic transport for drug delivery. Advanced Drug Delivery Reviews 63:10-11, pages 923-942.
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Stephen R. Dueker, Le T. Vuong, Peter N. Lohstroh, Jason A. Giacomo & John S. Vogel. (2011) Quantifying exploratory low dose compounds in humans with AMS. Advanced Drug Delivery Reviews 63:7, pages 518-531.
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Karen L. White, Gary Nguyen, William N. Charman, Glenn A. Edwards, W. A. (Fried) Faassen & Christopher J. H. Porter. (2009) Lymphatic Transport of Methylnortestosterone Undecanoate (MU) and the Bioavailability of Methylnortestosterone Are Highly Sensitive to the Mass of Coadministered Lipid after Oral Administration of MU. Journal of Pharmacology and Experimental Therapeutics 331:2, pages 700-709.
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Rishi Paliwal, Shivani Rai, Bhuvaneshwar Vaidya, Kapil Khatri, Amit K. Goyal, Neeraj Mishra, Abhinav Mehta & Suresh P. Vyas. (2009) Effect of lipid core material on characteristics of solid lipid nanoparticles designed for oral lymphatic delivery. Nanomedicine: Nanotechnology, Biology and Medicine 5:2, pages 184-191.
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Arik Dahan & Amnon Hoffman. (2008) Rationalizing the selection of oral lipid based drug delivery systems by an in vitro dynamic lipolysis model for improved oral bioavailability of poorly water soluble drugs. Journal of Controlled Release 129:1, pages 1-10.
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Shaoling Li, Rong (Ron) Liu & Nuo (Nolan) Wang. 2008. Water-Insoluble Drug Formulation, Second Edition. Water-Insoluble Drug Formulation, Second Edition 609 636 .
Ping Li & Luwei Zhao. (2007) Developing early formulations: Practice and perspective. International Journal of Pharmaceutics 341:1-2, pages 1-19.
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Rochele C. Rossi, Carolina L. Dias, Eliane M. Donato, Laura A. Martins, Ana M. Bergold & Pedro E. Fröehlich. (2007) Development and validation of dissolution test for ritonavir soft gelatin capsules based on in vivo data. International Journal of Pharmaceutics 338:1-2, pages 119-124.
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David M. Shackleford, Christopher J. H. Porter & William N. Charman. 2007. Prodrugs. Prodrugs 653 682 .
Natalie L. Trevaskis, Christopher J.H. Porter & William N. Charman. (2006) AN EXAMINATION OF THE INTERPLAY BETWEEN ENTEROCYTE-BASED METABOLISM AND LYMPHATIC DRUG TRANSPORT IN THE RAT. Drug Metabolism and Disposition 34:5, pages 729-733.
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William N. Charman, Susan A. Charman & Christopher J. H. Porter. 2006. Optimizing the “Drug-Like” Properties of Leads in Drug Discovery. Optimizing the “Drug-Like” Properties of Leads in Drug Discovery 131 150 .
Kopparam Manjunath & Vobalaboina Venkateswarlu. (2005) Pharmacokinetics, tissue distribution and bioavailability of clozapine solid lipid nanoparticles after intravenous and intraduodenal administration. Journal of Controlled Release 107:2, pages 215-228.
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