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Drug Evaluations

Tanespimycin: the opportunities and challenges of targeting heat shock protein 90

Pages 861-868 | Published online: 25 May 2009

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Rahagir Salekeen, Michael S. Lustgarten, Umama Khan & Kazi Mohammed Didarul Islam. (2023) Model organism life extending therapeutics modulate diverse nodes in the drug-gene-microbe tripartite human longevity interactome. Journal of Biomolecular Structure and Dynamics 0:0, pages 1-19.
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Anna Bentke, Jędrzej Małecki, Barbara Ostrowska, Katarzyna Krzykowska-Petitjean & Piotr Laidler. (2013) Tanespimycin and Tipifarnib Exhibit Synergism in Inducing Apoptosis in Melanoma Cell Lines From Later Stages of Tumor Progression. Cancer Investigation 31:8, pages 545-549.
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TaeHun Kim, Gyochang Keum & Ae Nim Pae. (2013) Discovery and development of heat shock protein 90 inhibitors as anticancer agents: a review of patented potent geldanamycin derivatives. Expert Opinion on Therapeutic Patents 23:8, pages 919-943.
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