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Dipeptidyl peptidase-4 inhibitors for the treatment of type 2 diabetes: comparison, efficacy and safety

, PhD DMSc & , MD DMSc
Pages 2047-2058 | Published online: 07 Aug 2013

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Yunxiang Ma, Junkai Wang, Changhua Wang, Qiong Zhang, Yannan Xu, Huajin Liu, Xia Xiang & Jiangwei Ma. (2019) DPP-4 inhibitor anagliptin protects against hypoxia-induced cytotoxicity in cardiac H9C2 cells. Artificial Cells, Nanomedicine, and Biotechnology 47:1, pages 3823-3831.
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Cristina M. Alcántara & Andrés R. Alcántara. (2018) Biocatalyzed synthesis of antidiabetic drugs: A review. Biocatalysis and Biotransformation 36:1, pages 12-46.
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Takashi Kadowaki, Satsuki Muto, Yoshiumi Ouchi, Ryutaro Shimazaki & Yutaka Seino. (2017) Efficacy and safety of saxagliptin in combination with insulin in Japanese patients with type 2 diabetes mellitus: a 16-week double-blind randomized controlled trial with a 36-week open-label extension. Expert Opinion on Pharmacotherapy 18:18, pages 1903-1919.
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Baptist Gallwitz. (2017) A safety evaluation of empagliflozin plus linagliptin for treating type 2 diabetes. Expert Opinion on Drug Safety 16:12, pages 1399-1405.
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Huan Yu & Vincent C Woo. (2017) Emerging use of combination therapies for the management of type 2 diabetes – focus on saxagliptin and dapagliflozin. Diabetes, Metabolic Syndrome and Obesity 10, pages 317-332.
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Ryuichi Morishita & Hironori Nakagami. (2015) Teneligliptin: expectations for its pleiotropic action. Expert Opinion on Pharmacotherapy 16:3, pages 417-426.
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Jocelyn de Heer & Burkhard Göke. (2014) Are incretin mimetics and enhancers linked to pancreatitis and malignant transformations in pancreas?. Expert Opinion on Drug Safety 13:11, pages 1469-1481.
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Kimberly A Coughlan, Rudy J Valentine, Neil B Ruderman & Asish K Saha. (2014) AMPK activation: a therapeutic target for type 2 diabetes?. Diabetes, Metabolic Syndrome and Obesity 7, pages 241-253.
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Kristin Gonzales & Adrian Vella. 2021. Clinical Dilemmas in Diabetes. Clinical Dilemmas in Diabetes 146 160 .
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R. D. Carr & A. Solomon. (2020) Inhibitors of dipeptidyl peptidase‐4 as therapeutic agents for individuals with type 2 diabetes: a 25‐year journey. Diabetic Medicine 37:8, pages 1230-1233.
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