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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 25, 2010 - Issue 3
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Research Article

Evaluation of the antifungal and plasma membrane H+-ATPase inhibitory action of ebselen and two ebselen analogs in S. cerevisiae cultures

Blase BillackSt. John’s University, Jamaica, NY, USACorrespondence[email protected]
,
Magdalena Piętka-OttlikWrocław University of Technology, Wrocław, Poland
,
Michelle SantoroSt. John’s University, Jamaica, NY, USA
,
Stacia NicholsonSt. John’s University, Jamaica, NY, USA
,
Jacek MłochowskiWrocław University of Technology, Wrocław, Poland
&
Cesar Lau-CamSt. John’s University, Jamaica, NY, USA
Pages 312-317 | Received 24 Feb 2009, Accepted 01 Jun 2009, Published online: 09 Mar 2010

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Hemanta C. Rao Tumu, Benedette J. Cuffari, Maria A. Pino, Jerzy Palus, Magdalena Piętka-Ottlik & Blase Billack. (2020) Ebselen oxide attenuates mechlorethamine dermatotoxicity in the mouse ear vesicant model. Drug and Chemical Toxicology 43:4, pages 335-346.
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Articles from other publishers (25)

Margaret R. Young, Sabine Heit & Maike Bublitz. (2024) Structure, function and biogenesis of the fungal proton pump Pma1. Biochimica et Biophysica Acta (BBA) - Molecular Cell Research 1871:1, pages 119600.
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Truong‐Thanh Tung & John Nielsen. (2022) Drug Discovery and Development on Pma1, Where Are We Now? A Critical Review from 1995 to 2022. ChemMedChem 17:19.
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Sebastian Gnat, Dominik Łagowski, Mariusz Dyląg, Grzegorz Jóźwiak, Aleksandra Trościańczyk & Aneta Nowakiewicz. (2022) In Vitro Activity of Ebselen and Diphenyl Diselenide Alone and in Combination with Drugs against Trichophyton mentagrophytes Strains. Pharmaceutics 14:6, pages 1158.
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Suvidha Menon, Richa Vartak, Ketankumar Patel & Blase Billack. (2021) Evaluation of the antifungal activity of an ebselen-loaded nanoemulsion in a mouse model of vulvovaginal candidiasis. Nanomedicine: Nanotechnology, Biology and Medicine 37, pages 102428.
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Hemanta C Rao Tumu, Benedette J. Cuffari & Blase Billack. (2021) Combination of ebselen and hydrocortisone substantially reduces nitrogen mustard-induced cutaneous injury. Current Research in Toxicology 2, pages 375-385.
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Jun Wang, Peng Wang, Chuanjiang Dong, Ying Zhao, Jingxuan Zhou, Chunling Yuan & Lili Zou. (2020) Mechanisms of ebselen as a therapeutic and its pharmacology applications. Future Medicinal Chemistry 12:23, pages 2141-2160.
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Richa Vartak, Manali Patki, Suvidha Menon, Joseph Jablonski, Sonia Mediouni, Yige Fu, Susana T. Valente, Blase Billack & Ketan Patel. (2020) β-cyclodextrin polymer/Soluplus® encapsulated Ebselen ternary complex (EβpolySol) as a potential therapy for vaginal candidiasis and pre-exposure prophylactic for HIV. International Journal of Pharmaceutics 589, pages 119863.
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Richa Vartak, Suvidha Menon, Manali Patki, Blase Billack & Ketan Patel. (2020) Ebselen nanoemulgel for the treatment of topical fungal infection. European Journal of Pharmaceutical Sciences 148, pages 105323.
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Nadine M.S. Araújo, Lucas P. Dias, Helen P.S. Costa, Daniele O.B. Sousa, Ilka M. Vasconcelos, Glaucia A. de Morais & Jose T.A. Oliveira. (2019) ClTI, a Kunitz trypsin inhibitor purified from Cassia leiandra Benth. seeds, exerts a candidicidal effect on Candida albicans by inducing oxidative stress and necrosis. Biochimica et Biophysica Acta (BBA) - Biomembranes 1861:11, pages 183032.
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Sabine Ottilie, Gregory M. Goldgof, Andrea L. Cheung, Jennifer L. Walker, Edgar Vigil, Kenneth E. Allen, Yevgeniya Antonova-Koch, Carolyn W. Slayman, Yo Suzuki & Jacob D. Durrant. (2018) Two inhibitors of yeast plasma membrane ATPase 1 (ScPma1p): toward the development of novel antifungal therapies. Journal of Cheminformatics 10:1.
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Holly C. May, Jieh-Juen Yu, M. N. Guentzel, James P. Chambers, Andrew P. Cap & Bernard P. Arulanandam. (2018) Repurposing Auranofin, Ebselen, and PX-12 as Antimicrobial Agents Targeting the Thioredoxin System. Frontiers in Microbiology 9.
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Truong-Thanh Tung, Trong T. Dao, Marta G. Junyent, Michael Palmgren, Thomas Günther-Pomorski, Anja T. Fuglsang, Søren B. Christensen & John Nielsen. (2018) LEGO-Inspired Drug Design: Unveiling a Class of Benzo[ d ]thiazoles Containing a 3,4-Dihydroxyphenyl Moiety as Plasma Membrane H + -ATPase Inhibitors . ChemMedChem 13:1, pages 37-47.
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Bruna G. BatistaDaiane F. Dalla LanaGustavo P. SilveiraMarcus M. SáMisael FerreiraTheo V. C. RussoRômulo F. S. CantoFlavio A. R. BarbosaAntônio L. BragaTaís F. A. KaminskiLuís F. S. de OliveiraMichel M. MachadoWilliam LopesMarilene H. VainsteinMário L. TeixeiraSaulo F. AndradeAlexandre M. Fuentefria. (2017) Allylic Selenocyanates as New Agents to Combat Fusarium Species Involved with Human Infections . ChemistrySelect 2:35, pages 11926-11932.
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Lasse Kjellerup, Sandra Gordon, Karen O'Hanlon Cohrt, William Dalby Brown, Anja Thoe Fuglsang & Anne-Marie L. Winther. (2017) Identification of Antifungal H + -ATPase Inhibitors with Effect on Plasma Membrane Potential . Antimicrobial Agents and Chemotherapy 61:7.
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Mirosław Giurg, Anna Gołąb, Jakub Suchodolski, Rafał Kaleta, Anna Krasowska, Egbert Piasecki & Magdalena Piętka-Ottlik. (2017) Reaction of bis[(2-chlorocarbonyl)phenyl] Diselenide with Phenols, Aminophenols, and Other Amines towards Diphenyl Diselenides with Antimicrobial and Antiviral Properties. Molecules 22:6, pages 974.
Crossref
Natalie N. Orie, Andrew R. Warren, Jovana Basaric, Cesar Lau-Cam, Magdalena Piętka-Ottlik, Jacek Młochowski & Blase Billack. (2017) In vitro assessment of the growth and plasma membrane H + -ATPase inhibitory activity of ebselen and structurally related selenium- and sulfur-containing compounds in Candida albicans . Journal of Biochemical and Molecular Toxicology 31:6, pages e21892.
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Shankar Thangamani, Hassan E. Eldesouky, Haroon Mohammad, Pete E. Pascuzzi, Larisa Avramova, Tony R. Hazbun & Mohamed N. Seleem. (2017) Ebselen exerts antifungal activity by regulating glutathione (GSH) and reactive oxygen species (ROS) production in fungal cells. Biochimica et Biophysica Acta (BBA) - General Subjects 1861:1, pages 3002-3010.
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Magdalena Piętka-Ottlik, Agnieszka Lewińska, Anna Jaromin, Anna Krasowska & Kazimiera A. Wilk. (2016) Antifungal organoselenium compound loaded nanoemulsions stabilized by bifunctional cationic surfactants. Colloids and Surfaces A: Physicochemical and Engineering Aspects 510, pages 53-62.
Crossref
Trong Tuan Dao, Pankaj Sehgal, Truong Thanh Tung, Jesper Vuust Møller, John Nielsen, Michael Palmgren, Søren Brøgger Christensen & Anja Thoe Fuglsang. (2016) Demethoxycurcumin Is A Potent Inhibitor of P-Type ATPases from Diverse Kingdoms of Life. PLOS ONE 11:9, pages e0163260.
Crossref
Nikhat Manzoor. 2016. Regulation of Ca2+-ATPases,V-ATPases and F-ATPases. Regulation of Ca2+-ATPases,V-ATPases and F-ATPases 519 530 .
Gajendra Kumar Azad & Raghuvir S. Tomar. (2014) Ebselen, a promising antioxidant drug: mechanisms of action and targets of biological pathways. Molecular Biology Reports 41:8, pages 4865-4879.
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Mikhail V. Keniya, Richard D. Cannon, ẤnBình Nguyễn, Joel D.A. Tyndall & Brian C. Monk. (2013) Heterologous expression of Candida albicans Pma1p in Saccharomyces cerevisiae . FEMS Yeast Research 13:3, pages 302-311.
Crossref
Ann R. Holmes, Mikhail V. Keniya, Irena Ivnitski-Steele, Brian C. Monk, Erwin Lamping, Larry A. Sklar & Richard D. Cannon. (2012) The Monoamine Oxidase A Inhibitor Clorgyline Is a Broad-Spectrum Inhibitor of Fungal ABC and MFS Transporter Efflux Pump Activities Which Reverses the Azole Resistance of Candida albicans and Candida glabrata Clinical Isolates. Antimicrobial Agents and Chemotherapy 56:3, pages 1508-1515.
Crossref
Zvi RappoportCristina W. Nogueira & João B. T. Rocha. 2010. Patai's Chemistry of Functional Groups. Patai's Chemistry of Functional Groups.
. (2010) Current awareness on yeast. Yeast 27:9, pages 777-784.
Crossref

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